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1
المؤلفون: Joseph M. Luettgen, Carol A. Watson, Pancras C. Wong, Cailan Wang, Mark R. Harpel, Vidhyashankar Ramamurthy, Ge Zhang, Jeffrey M. Bozarth, Tara L. Peterson, Francis J. Woerner, Dietmar A. Seiffert, Alan R. Rendina, Frank A. Barbera, Karen A. Rossi, Ruth R. Wexler, Randi L. Brown, Joanne M. Smallheer, Paul E. Morin, Mimi L. Quan, Anzhi Wei
المصدر: Journal of Medicinal Chemistry. 57:955-969
مصطلحات موضوعية: Bleeding Time, Stereochemistry, Chemistry, Molecular Conformation, Stereoisomerism, Factor XIa, Pharmacology, Crystallography, X-Ray, Risk profile, Small molecule, Molecular Docking Simulation, Structure-Activity Relationship, Fibrinolytic Agents, Drug Discovery, Antithrombotic, Quinolines, Animals, Humans, Molecular Medicine, Rabbits, Factor Xa Inhibitors
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2
المؤلفون: James A. Johnson, Ramakrishna Seethala, Christine Huang, Michael M. Miller, David S. Taylor, Ji Jiang, Ruth R. Wexler, Mark E. Salvati, Jun Zhang, Xiaohong Yin, Yalei Liu, R. Michael Lawrence, Tatyana Zvyaga, David S. Nirschl, Lalgudi S. Harikrishnan, Tara L. Peterson, Michael A. Poss, Alice Ye A. Chen, Leonard P. Adam, Yufeng Wang, Muthoni G. Kamau
المصدر: Bioorganicmedicinal chemistry letters. 22(20)
مصطلحات موضوعية: Halogenation, Pyridines, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Mice, Drug Discovery, Cholesterylester transfer protein, Moiety, Animals, Humans, Urea, Amines, Molecular Biology, CETP inhibitor, biology, Chemistry, Organic Chemistry, Reverse cholesterol transport, In vitro, Cholesterol Ester Transfer Proteins, Rats, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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3
المؤلفون: R. Michael Lawrence, George C. Morton, Mark E. Salvati, Jonathan O’Connell, Ramakrishna Seethala, Arthur V. Miller, Tara L. Peterson, Cooper Christopher B, Carolyn A. Weigelt, Yalei Liu, Tammy C. Wang, Lalgudi S. Harikrishnan, Timothy F. Herpin, Kingsley K. Appiah, David S. Taylor, Xiaohong Yin, Muthoni G. Kamau, Jennifer X. Qiao, Leonard P. Adam, Alice Ye A. Chen, David S. Nirschl
المصدر: Bioorganicmedicinal chemistry letters. 18(8)
مصطلحات موضوعية: Models, Molecular, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Cholesterylester transfer protein, medicine, Humans, Molecular Biology, CETP inhibitor, Benzoxazoles, biology, Molecular Structure, Chemistry, Organic Chemistry, Benzoxazole, Fluorescence, Coronary heart disease, Cholesterol Ester Transfer Proteins, Pattern synthesis, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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4
المؤلفون: Andrew T. Pudzianowski, William A. Schumacher, Jeffrey M. Bozarth, Karnail S. Atwal, Doree F. Sitkoff, Thomas E. Steinbacher, Sharon N. Bisaha, Chi Li, Eddie C.-K. Liu, Sonia Youssef, Yan Shi, Philip D. Stein, Tara L. Peterson, Karen S. Hartl, Stephen P. O'connor, Ge Zhang, Mengxiao Shi, Steven M. Seiler, Jing Zhang, Robert Zahler, Gregory S. Bisacchi, Alan R. Rendina
المصدر: Bioorganicmedicinal chemistry letters. 15(24)
مصطلحات موضوعية: Models, Molecular, medicine.drug_mechanism_of_action, Lactams, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Molecular Conformation, Pharmaceutical Science, Ketene, Administration, Oral, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Humans, Molecular Biology, Chemistry, Organic Chemistry, Ethylenes, Ketones, Thiourea, Aminal, Lactam, Molecular Medicine, Bioisostere, Factor Xa Inhibitors
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5
المؤلفون: Karen S. Hartl, Jeffrey M. Bozarth, Steven M. Seiler, Karnail S. Atwal, Chi Li, Sharon N. Bisaha, Thomas E. Steinbacher, Philip D. Stein, Yan Shi, Stephen P. O'connor, Andrew T. Pudzianowski, William A. Schumacher, Gregory S. Bisacchi, Doree F. Sitkoff, Alan R. Rendina, Eddie C.-K. Liu, Tara L. Peterson, Sonia Youssef, Ge Zhang, Mengxiao Shi, Jing Zhang, Robert Zahler
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:1449
مصطلحات موضوعية: Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Ketene, Biochemistry, chemistry.chemical_compound, Orally active, Drug Discovery, Aminal, Lactam, Molecular Medicine, Molecular Biology