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1دورية أكاديمية
المصدر: Translational Oncology, Vol 10, Iss 2, Pp 153-157 (2017)
مصطلحات موضوعية: Neoplasms. Tumors. Oncology. Including cancer and carcinogens, RC254-282
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Yi Yu, Ronald E Savage, Sudharshan Eathiraj, Justin Meade, Michael J Wick, Terence Hall, Giovanni Abbadessa, Brian Schwartz
المصدر: PLoS ONE, Vol 10, Iss 10, p e0140479 (2015)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/1932-6203
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المؤلفون: Terence Hall, Yunxia Wang, Bassel F. El-Rayes, Patricia LoRusso, Walid L. Shaib, Jasgit C. Sachdev, Ronald E. Savage, R. D. Harvey, Giovanni Abbadessa, Julia Kazakin, Drew W. Rasco, Amita Patnaik, Brian Schwartz, Kyriakos P. Papadopoulos, Anthony W. Tolcher
المصدر: British Journal of Cancer
مصطلحات موضوعية: 0301 basic medicine, Adult, Male, Cancer Research, medicine.medical_specialty, Pathology, FGFR2 fusion, Nausea, Administration, Oral, Gastroenterology, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Internal medicine, Neoplasms, medicine, Adrenocortical carcinoma, Humans, Dosing, Adverse effect, Protein Kinase Inhibitors, solid tumours, Aged, Aniline Compounds, business.industry, Middle Aged, medicine.disease, Receptors, Fibroblast Growth Factor, FGFR inhibitor, 030104 developmental biology, Oncology, phase 1, 030220 oncology & carcinogenesis, Pharmacodynamics, Toxicity, Cohort, Clinical Study, Quinazolines, Female, medicine.symptom, business
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المؤلفون: Terence Hall, Brian Schwartz, Michael J. Wick, Sudharshan Eathiraj, Giovanni Abbadessa, Yi Yu
المصدر: Anti-Cancer Drugs
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, Cell cycle checkpoint, Cell, Aminopyridines, Bioinformatics, Mice, 0302 clinical medicine, Neoplasms, Antineoplastic Combined Chemotherapy Protocols, Preclinical Reports, Pharmacology (medical), ARQ 087, Mice, Inbred BALB C, Aniline Compounds, FGFR, Imidazoles, Drug Synergism, inhibitor, medicine.anatomical_structure, Oncology, 030220 oncology & carcinogenesis, ComputingMethodologies_DOCUMENTANDTEXTPROCESSING, Female, ARQ 092, kinase, small molecule, Biology, 03 medical and health sciences, In vivo, Cell Line, Tumor, medicine, Animals, Humans, Protein Kinase Inhibitors, Protein kinase B, PI3K/AKT/mTOR pathway, combination, Pharmacology, AKT, Cancer, medicine.disease, Receptors, Fibroblast Growth Factor, Xenograft Model Antitumor Assays, Endometrial Neoplasms, 030104 developmental biology, Apoptosis, Quinazolines, Cancer research, Drug Screening Assays, Antitumor, Ovarian cancer, Proto-Oncogene Proteins c-akt
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::04e80297afd8299ce4ed5e7719e7a826
https://doi.org/10.1097/cad.0000000000000486 -
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المصدر: Translational Oncology, Vol 10, Iss 2, Pp 153-157 (2017)
مصطلحات موضوعية: 0301 basic medicine, Chemotherapy, Cancer Research, Kinase, business.industry, medicine.medical_treatment, Pan FGFR Inhibitor ARQ 087, Pharmacology, lcsh:Neoplasms. Tumors. Oncology. Including cancer and carcinogens, lcsh:RC254-282, Carboplatin, Capecitabine, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, Paclitaxel, Oncology, 030220 oncology & carcinogenesis, medicine, Cytotoxic T cell, Receptor, business, medicine.drug
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المؤلفون: Paula Olaizola, Massimo Roncalli, N. Navari, Karim Fiaccadori, Chiara Raggi, Fabio Marra, Giovanni Abbadessa, B. Piombanti, Gianfranco Alpini, Luca Di Tommaso, Terence Hall, Jesus M. Banales, Annarita Destro, Elisabetta Rovida, Margherita Correnti, Alessandra Elvevi, Pietro Invernizzi, Shannon Glaser, Michele Droz dit Busset, Vincenzo Mazzaferro, Fanyin Meng, Elisa Forti, Sherrie Bhoori, Alessio Gerussi, Mirella Pastore, Caterina Peraldo-Neia
المساهمون: Raggi, C, Fiaccadori, K, Pastore, M, Correnti, M, Piombanti, B, Forti, E, Navari, N, Abbadessa, G, Hall, T, Destro, A, Di Tommaso, L, Roncalli, M, Meng, F, Glaser, S, Rovida, E, Peraldo-Neia, C, Olaizola, P, Banales, J, Gerussi, A, Elvevi, A, Droz Dit Busset, M, Bhoori, S, Mazzaferro, V, Alpini, G, Marra, F, Invernizzi, P
مصطلحات موضوعية: 0301 basic medicine, Epithelial-Mesenchymal Transition, information science, Biology, Fibroblast growth factor, Pathology and Forensic Medicine, Cholangiocarcinoma, 03 medical and health sciences, 0302 clinical medicine, parasitic diseases, Tumor Cells, Cultured, Humans, cardiovascular diseases, Phosphorylation, Receptor, Fibroblast Growth Factor, Type 2, Receptor, Protein Kinase Inhibitors, Protein kinase B, Cell Proliferation, Aniline Compounds, Fibroblast growth factor receptor 2, Cell growth, Fibroblast growth factor receptor 1, fungi, 030104 developmental biology, Bile Duct Neoplasms, Fibroblast growth factor receptor, 030220 oncology & carcinogenesis, Quinazolines, cardiovascular system, Cancer research, Signal transduction, Signal Transduction
وصف الملف: STAMPA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6bab2b025cbe2443ffc855f41a68d0b3
http://hdl.handle.net/10281/240048 -
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المؤلفون: Nevena Damjanov, Sherrie Bhoori, Kyriakos P. Papadopoulos, Terence Hall, Michele Droz dit Busset, Fadi Braiteh, Christian Cotsoglou, Nicola Personeni, William P. Harris, Walid L. Shaib, Yunxia Wang, Brian Schwartz, Vincenzo Mazzaferro, Gianluca Masi, Vittorina Zagonel, Lorenza Rimassa, Julia Kazakin, Bassel F. El-Rayes, Filippo de Braud
المصدر: British Journal of Cancer
مصطلحات موضوعية: Adult, Male, Cancer Research, medicine.medical_specialty, Oncogene Proteins, Fusion, medicine.medical_treatment, Gastroenterology, Article, Cholangiocarcinoma, Fusion gene, 03 medical and health sciences, Hyperphosphatemia, Alkaloids, Targeted therapies, 0302 clinical medicine, Internal medicine, medicine, Humans, In patient, Receptor, Fibroblast Growth Factor, Type 2, Intrahepatic Cholangiocarcinomas, Adverse effect, Protein Kinase Inhibitors, Intrahepatic Cholangiocarcinoma, Aged, Aged, 80 and over, Clinical Trials as Topic, Chemotherapy, Aniline Compounds, business.industry, Bile duct cancer, Middle Aged, medicine.disease, Bile Ducts, Intrahepatic, Bile Duct Neoplasms, Oncology, 030220 oncology & carcinogenesis, Mutation, Toxicity, Quinazolines, Female, Gene Fusion, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8fa956fa25583c496cdf14ed67299e12
http://hdl.handle.net/11568/994323 -
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المؤلفون: Maria Lamar, Terence Hall, Brian Schwartz, Julia Kazakin, Shubham Pant, Ronald E. Savage
المصدر: Molecular Cancer Therapeutics. 18:A034-A034
مصطلحات موضوعية: Cancer Research, business.industry, Insulin, medicine.medical_treatment, Cmax, AKT1, Pharmacology, Oncology, Pharmacokinetics, Pharmacodynamics, medicine, business, Protein kinase B, PI3K/AKT/mTOR pathway, Whole blood
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b10813e62a4002c06d4b28d9d65807c6
https://doi.org/10.1158/1535-7163.targ-19-a034 -
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المؤلفون: Mark A. Ashwell, Jean-Marc Lapierre, Christopher Brassard, Karen Bresciano, Cathy Bull, Susan Cornell-Kennon, Sudharshan Eathiraj, Dennis S. France, Terence Hall, Jason Hill, Eoin Kelleher, Sampada Khanapurkar, Darin Kizer, Steffi Koerner, Jeff Link, Yanbin Liu, Sapna Makhija, Magdi Moussa, Nivedita Namdev, Khanh Nguyen, Robert Nicewonger, Rocio Palma, Jeff Szwaya, Manish Tandon, Uma Uppalapati, David Vensel, Laurie P. Volak, Erika Volckova, Neil Westlund, Hui Wu, Rui-Yang Yang, Thomas C. K. Chan
المصدر: Journal of Medicinal Chemistry. 55:5291-5310
مصطلحات موضوعية: Models, Molecular, Protein Conformation, Pyridines, Administration, Oral, Biological Availability, AKT1, Antineoplastic Agents, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Mice, Structure-Activity Relationship, Adenosine Triphosphate, In vivo, Catalytic Domain, Cell Line, Tumor, Drug Discovery, Animals, Humans, Structure–activity relationship, Phosphorylation, Protein kinase B, Adaptor Proteins, Signal Transducing, Cell Proliferation, Effector, Chemistry, Imidazoles, Ribosomal Protein S6 Kinases, 70-kDa, Small molecule, Biochemistry, Microsomes, Liver, Molecular Medicine, Proto-Oncogene Proteins c-akt, Protein Binding
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المؤلفون: Terence Hall, William P. Harris, Ronald E. Savage, Vincenzo Mazzaferro, Gianluca Masi, Christian Cotsoglou, Brian Schwartz, Nicola Personeni, Maria Lamar, Julia Kazakin, Walid L. Shaib, Lorenza Rimassa, Bassel F. El-Rayes, Sherrie Bhoori, Vittorina Zagonel, Yunxia Wang, Kyriakos P. Papadopoulos, Nevana Damjanov, Michele Droz-Dit-Busset
المصدر: Cancer Research. 78:LB-232
مصطلحات موضوعية: Cancer Research, Cellular differentiation, FGFR Inhibition, Cancer, FGF19, Biology, Fibroblast growth factor, medicine.disease, Receptor tyrosine kinase, Oncology, Fibroblast growth factor receptor, medicine, Cancer research, biology.protein, Receptor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::866d06a8deec5eda3a4742570916cd76
https://doi.org/10.1158/1538-7445.am2018-lb-232