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المصدر: Airway pharmacology and treatment.
مصطلحات موضوعية: Proteases, biology, business.industry, Lung injury, Cathepsin G, Molecular biology, In vitro, chemistry.chemical_compound, chemistry, In vivo, Proteinase 3, Neutrophil elastase, biology.protein, Medicine, business, IC50
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::2b7ea17d0fe41559b33026867fd554db
https://doi.org/10.1183/13993003.congress-2020.3303 -
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المؤلفون: Thorsten Oost, Herbert Nar, Christian A. Kuttruff
المصدر: Medicinal Chemistry Reviews ISBN: 9780996293280
Medicinal Chemistry Reviewsمصطلحات موضوعية: Oncology, medicine.medical_specialty, Sting, business.industry, Internal medicine, medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::167ac6c2f802db5feb2a003767438201
https://doi.org/10.29200/acsmedchemrev-v54.ch9 -
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المؤلفون: Achim Grube, Martin Fleck, Vittoria Zinzalla, Norbert Kraut, Georg Rast, Maria Antonietta Impagnatiello, Sebastian Carotta, Gabriela Gremel, Esther Schmidt, Paolo Chetta, Jonathon Sedgwick, Thorsten Oost, Sophia Blake, Thorsten Laux, Thomas Zichner, Marco H. Hofmann, Tom Bretschneider, Ute Klinkhardt, Kirsten Arndt-Schmitz, Herbert Nar, Otmar Schaaf
المصدر: Cancer Research. 80:4522-4522
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, business.industry, medicine.medical_treatment, medicine.disease, Primary tumor, eye diseases, 03 medical and health sciences, Sting, 030104 developmental biology, 0302 clinical medicine, Immune system, Cytokine, Oncology, In vivo, Interferon, Cancer research, Medicine, Cytokine secretion, business, Ex vivo, 030215 immunology, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c1e8c9ee01a60eb8189bc2e10e183b8a
https://doi.org/10.1158/1538-7445.am2020-4522 -
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المؤلفون: Thorsten Oost, Marcel M. van Gaalen, Liliane Unger, Hervé Geneste, Wilfried Hornberger, Charles W. Hutchins, Astrid Netz, Swati Bhowmik
المصدر: Bioorganicmedicinal chemistry letters. 28(19)
مصطلحات موضوعية: 0301 basic medicine, Vasopressin, Clinical Biochemistry, Pharmaceutical Science, Biological Availability, Pharmacology, 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, 0302 clinical medicine, Microsomes, Drug Discovery, Moiety, Animals, Humans, Oxindole, Receptor, Molecular Biology, Organic Chemistry, Brain, Antidepressive Agents, Bioavailability, Rats, Piperazine, 030104 developmental biology, chemistry, Models, Animal, Microsome, Molecular Medicine, Penetrant (biochemical), Antidiuretic Hormone Receptor Antagonists, Half-Life
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المؤلفون: W. Lubisch, Astrid Netz, Wilfried Hornberger, Swati Bhowmik, Liliane Unger, Hervé Geneste, Wolfgang Wernet, Marcel M. van Gaalen, Thorsten Oost, Gisela Backfisch
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3828-3831
مصطلحات موضوعية: Vasopressin, Indoles, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Drug Discovery, Animals, Moiety, Oxindole, Receptor, Molecular Biology, Oxazole, Arginine vasopressin receptor 1B, Molecular Structure, Organic Chemistry, Biological activity, Antidepressive Agents, Oxindoles, Rats, Disease Models, Animal, chemistry, Lactam, Molecular Medicine, Antidiuretic Hormone Receptor Antagonists, Protein Binding
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المؤلفون: Daniel H. Rich, Chanokporn Sukonpan, Eric A. Johnson, Michael C. Goodnough, Thorsten Oost, William H. Tepp
المصدر: The Journal of Peptide Research. 63:181-193
مصطلحات موضوعية: chemistry.chemical_classification, Dipeptide, Stereochemistry, Substrate (chemistry), Peptide, Biochemistry, chemistry.chemical_compound, Enzyme activator, Endocrinology, Enzyme, chemistry, Tetrahedral carbonyl addition compound, Peptide synthesis, Peptide sequence
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::51e31bef8277232649dece0289781d72
https://doi.org/10.1111/j.1399-3011.2004.00124.x -
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المؤلفون: Thorsten Lehmann, Ralf Lotz, Thorsten Oost, Mueller Stephan Georg, Klaus Rudolf, Dirk Stenkamp, Armin Heckel, Ralph Budzinski, Jörg Kley, Gerd-Michael Maier, Gerald Juergen Roth, Leo Thomas, Martin Lenter, Kirsten Arndt, Michael Markert
المصدر: Bioorganicmedicinal chemistry letters. 25(16)
مصطلحات موضوعية: medicine.medical_specialty, Pyridines, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, In Vitro Techniques, Lipidoses, Biochemistry, Part iii, Structure-Activity Relationship, Internal medicine, Appetite Depressants, Drug Discovery, medicine, Potassium Channel Blockers, Moiety, Animals, Humans, Receptors, Somatostatin, Receptor, Molecular Biology, Phospholipids, Phospholipidosis, biology, Chemistry, Organic Chemistry, Body Weight, Antagonist, Ether-A-Go-Go Potassium Channels, High-Throughput Screening Assays, Rats, Pyridazines, Endocrinology, Design synthesis, Pyrazines, biology.protein, Hepatocytes, Microsomes, Liver, Molecular Medicine, Anti-Obesity Agents, Cyclobutanes, Sibutramine, medicine.drug
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المؤلفون: Gerd-Michael Maier, Thorsten Lehmann, Ralf Lotz, Jörg Kley, Martin Lenter, Michael Markert, Mueller Stephan Georg, Kirsten Arndt, Philipp Lustenberger, Klaus Rudolf, Thorsten Oost, Armin Heckel, Marcus Schindler, Gerald Juergen Roth, Dirk Stenkamp
المصدر: Bioorganicmedicinal chemistry letters. 25(16)
مصطلحات موضوعية: Pyridines, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Receptors, G-Protein-Coupled, Eating, Structure-Activity Relationship, Animal model, In vivo, Drug Discovery, Potency, Animals, Cytochrome P-450 Enzyme Inhibitors, ATP Binding Cassette Transporter, Subfamily B, Member 1, Obesity, Receptors, Somatostatin, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Body Weight, Antagonist, Limiting, High-Throughput Screening Assays, Rats, Design synthesis, Cytochrome P-450 CYP2D6, Alkynes, Drug Design, Molecular Medicine, Efflux, Anti-Obesity Agents
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المؤلفون: Kirsten Arndt, Ralf Lotz, Klaus Rudolf, Thorsten Lehmann, Mueller Stephan Georg, Ralph Budzinski, Gerald Juergen Roth, Leo Thomas, Martin Lenter, Dirk Stenkamp, Armin Heckel, Thorsten Oost, Marcus Schindler, Jörg Kley
المصدر: Bioorganicmedicinal chemistry letters. 25(16)
مصطلحات موضوعية: Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Lipidoses, Biochemistry, Structure-Activity Relationship, Drug Discovery, Potassium Channel Blockers, Animals, Receptor, Serotonin, 5-HT2A, Receptors, Somatostatin, Rats, Wistar, Receptor, Molecular Biology, Phospholipids, G protein-coupled receptor, Phospholipidosis, biology, Chemistry, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Rats, Pyridazines, Safety profile, Design synthesis, biology.protein, Molecular Medicine, Anti-Obesity Agents, Serotonin Antagonists
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المؤلفون: James M. Trevillyan, Charles W. Hutchins, Thorsten Oost, Mike A. Stashko, Gang Liu, Tom Lubben, Cele Abad-Zapatero, Bruce G. Szczepankiewicz, Zhili Xin, Steve J. Ballaron, Philip J. Hajduk, Mike R Jirousek, Zhonghua Pei
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:1887-1890
مصطلحات موضوعية: Phosphoric monoester hydrolases, T-Lymphocytes, Clinical Biochemistry, Pharmaceutical Science, Protein tyrosine phosphatase, Crystallography, X-Ray, Ligands, Benzoates, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Hydrolase, Combinatorial Chemistry Techniques, Enzyme Inhibitors, Phosphotyrosine, Molecular Biology, Protein Tyrosine Phosphatase, Non-Receptor Type 1, chemistry.chemical_classification, Binding Sites, Molecular Structure, biology, Organic Chemistry, Metabolism, Amides, In vitro, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Protein Tyrosine Phosphatases