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1
المؤلفون: Anthone W. Dunah, Thierry Bussiere, Kenneth J. Rhodes, Hairuo Peng, Lin Xu, Mahin Arastu, Gnanasambandam Kumaravel, Joy Wang, Melanie S. Brennan, Pamela A. Snodgrass-Belt, Arthur G. Taveras, Mi-young Jung, Tina Talreja, Sowmya Chollate, Zhili Xin, Diana Fahrer, Robert Dunstan, Robert H. Scannevin, Ellen Rohde, H. Moore Arnold
المصدر: Neuropharmacology. 103:57-68
مصطلحات موضوعية: Male, 0301 basic medicine, Gene isoform, Pathology, medicine.medical_specialty, Central nervous system, BACE1-AS, Plaque, Amyloid, Cleavage (embryo), Mice, 03 medical and health sciences, Cellular and Molecular Neuroscience, 0302 clinical medicine, Alzheimer Disease, Amyloid precursor protein, medicine, Animals, Protein Isoforms, Pharmacology, Aldehydes, Amyloid beta-Peptides, Dose-Response Relationship, Drug, biology, P3 peptide, Brain, medicine.disease, Rats, Inbred F344, Rats, Disease Models, Animal, Macaca fascicularis, 030104 developmental biology, medicine.anatomical_structure, biology.protein, Amyloid Precursor Protein Secretases, Alzheimer's disease, Amyloid precursor protein secretase, 030217 neurology & neurosurgery
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2
المؤلفون: Robert H. Scannevin, Tina Talreja, Lin Xu, Gnanasambandam Kumaravel, David Kocisko, Arthur G. Taveras, Anthone W. Dunah, Hairuo Peng, Kenneth J. Rhodes, Ellen Rohde, H. Moore Arnold, Sowmya Chollate, Pamela A. Snodgrass-Belt, Mi-yong Jung, Andrew Zhang, Zhili Xin, Melanie N. Shackett
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:7277-7280
مصطلحات موضوعية: Scaffold, Carboxylic acid, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Mice, chemistry.chemical_compound, Piperidines, Oral administration, Drug Discovery, Animals, γ secretase, Enzyme Inhibitors, Molecular Biology, Phenylacetates, chemistry.chemical_classification, Amyloid beta-Peptides, Nonsteroidal, Anti-Inflammatory Agents, Non-Steroidal, Organic Chemistry, Brain, Combinatorial chemistry, Peptide Fragments, Rats, chemistry, Drug Design, Molecular Medicine, Amyloid Precursor Protein Secretases
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3
المؤلفون: Tina Talreja, Arthur G. Taveras, Michael Humora, Lawrence Gan, J. Hernan Cuervo, Kenneth J. Rhodes, Hairuo Peng, Lin Xu, Anthone W. Dunah, Gnanasambandam Kumaravel, Pamela A. Snodgrass-Belt, Mi-young Jung, Zhili Xin, Sowmya Chollate, Melanie N. Shackett, Ellen Rohde, H. Moore Arnold, Robert H. Scannevin
المصدر: ACS Medicinal Chemistry Letters. 2:786-791
مصطلحات موضوعية: biology, business.industry, Organic Chemistry, Notch signaling pathway, Pharmacology, Biochemistry, In vitro, Pharmacokinetics, In vivo, Oral administration, Pharmacodynamics, Drug Discovery, biology.protein, Medicine, Potency, business, Amyloid precursor protein secretase
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4
المؤلفون: Teresa A. Soucy, Peter G. Smith, Michael A. Milhollen, Allison J. Berger, James M. Gavin, Sharmila Adhikari, James E. Brownell, Kristine E. Burke, David P. Cardin, Stephen Critchley, Courtney A. Cullis, Amanda Doucette, James J. Garnsey, Jeffrey L. Gaulin, Rachel E. Gershman, Anna R. Lublinsky, Alice McDonald, Hirotake Mizutani, Usha Narayanan, Edward J. Olhava, Stephane Peluso, Mansoureh Rezaei, Michael D. Sintchak, Tina Talreja, Michael P. Thomas, Tary Traore, Stepan Vyskocil, Gabriel S. Weatherhead, Jie Yu, Julie Zhang, Lawrence R. Dick, Christopher F. Claiborne, Mark Rolfe, Joseph B. Bolen, Steven P. Langston
المصدر: Nature. 458:732-736
مصطلحات موضوعية: NEDD8 Protein, Ubiquitin-activating enzyme, Transplantation, Heterologous, Antineoplastic Agents, Cyclopentanes, Ubiquitin-Activating Enzymes, NEDD8, Mice, Ubiquitin, Cell Line, Tumor, Neoplasms, Animals, Humans, Enzyme Inhibitors, Ubiquitins, Cells, Cultured, Multidisciplinary, biology, Cullin Proteins, Cell biology, Pyrimidines, Pevonedistat, Proteasome, Cancer cell, biology.protein, Female, Neddylation, Proteasome Inhibitors, Cullin
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5
المؤلفون: Kevin Guertin, Tonika Bohnert, Tao Wang, Howard Jones, Edward Yin-Shiang Lin, Daliya Banerjee, Tina Talreja, Istvan J. Enyedy, Kurt Van Vloten, Douglas Marcotte, Jianhua Chao, Jason D. Fontenot
المصدر: Bioorganicmedicinal chemistry letters. 25(15)
مصطلحات موضوعية: Models, Molecular, Drug Inverse Agonism, Clinical Biochemistry, Pharmaceutical Science, Inflammation, Pyrazole, Pharmacology, Biochemistry, Autoimmune Diseases, Pathogenesis, chemistry.chemical_compound, Mice, Drug Discovery, Gene expression, medicine, Moiety, Inverse agonist, Animals, Humans, Molecular Biology, Chemistry, Organic Chemistry, Interleukin-17, Nuclear Receptor Subfamily 1, Group F, Member 3, Nuclear receptor, Benzamides, Molecular Medicine, Pyrazoles, Th17 Cells, Interleukin 17, medicine.symptom, Spleen
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6
المؤلفون: Dominique Hebrault, Hairuo Peng, Xianglin Shi, Michael Humora, Zhili Xin, William F. Kiesman, Tina Talreja, Zezhou Wang
المصدر: ChemInform. 43
مصطلحات موضوعية: Reaction rate, Reaction conditions, chemistry.chemical_compound, Salicylaldehyde, Chemistry, Organic chemistry, General Medicine, Molecular sieve, Stereocenter
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7
المؤلفون: William F. Kiesman, Tina Talreja, Michael Humora, Hairuo Peng, Xianglin Shi, Dominique Hebrault, Zhili Xin, Zezhou Wang
المصدر: The Journal of organic chemistry. 77(2)
مصطلحات موضوعية: Reaction conditions, Aldehydes, Magnetic Resonance Spectroscopy, Molecular Structure, Chemistry, Organic Chemistry, Stereoisomerism, Chemistry Techniques, Synthetic, Molecular sieve, Stereocenter, Reaction rate, chemistry.chemical_compound, Salicylaldehyde, Organic chemistry, Amines, Amyloid Precursor Protein Secretases, Chromatography, High Pressure Liquid
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8
المؤلفون: Aleem Gangjee, Yibin Zeng, Tina Talreja, John J. McGuire, Sherry F. Queener, Roy L. Kisliuk
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Antineoplastic Agents, Pneumocystis carinii, Chemical synthesis, Article, chemistry.chemical_compound, Structure-Activity Relationship, Sulfanyl, Cell Line, Tumor, Drug Discovery, Dihydrofolate reductase, parasitic diseases, Escherichia coli, Animals, Humans, Pyrroles, Benzoic acid, Antibacterial agent, Cell Proliferation, chemistry.chemical_classification, biology, Aryl, Rats, Tetrahydrofolate Dehydrogenase, Pyrimidines, chemistry, Drug Resistance, Neoplasm, Drug Design, Antifolate, Thiol, biology.protein, Molecular Medicine, Folic Acid Antagonists, Drug Screening Assays, Antitumor, Toxoplasma, Mycobacterium avium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::52b5a53ff6a15df48292950fd69746c4
https://europepmc.org/articles/PMC3850752/ -
9دورية أكاديمية
المؤلفون: Aleem Gangjee, Yibin Zeng, Tina Talreja, John J. McGuire, Roy L. Kisliuk, Sherry F. Queener
المصدر: Journal of Medicinal Chemistry; Jun2007, Vol. 50 Issue 13, p3046-3053, 8p