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1دورية أكاديمية
المؤلفون: Menglin Chen, Zhengrong Zhu, Tom Wisniewski, Xiaoping Zhang, David G. McLaren, Adam Weinglass, S. Adrian Saldanha
المصدر: SLAS Discovery, Vol 27, Iss 7, Pp 405-412 (2022)
مصطلحات موضوعية: Label-free technologies, LC-MS, Cell-based assays, Affinity binding, Medicine (General), R5-920, Biotechnology, TP248.13-248.65
وصف الملف: electronic resource
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2
المؤلفون: Joe Clemas, Jerry Andrew Taylor, Feroze Ujjainwalla, Jim Tata, Doris F. Cully, Tom Wisniewski, Wei Tang, Charlene Bopp, Clare London, Andreas Verras, Scott B. Hoyt, Andrea Sok, Elaine Tung, Douglas J. MacNeil, Gaochao Zhou, Amjad Ali, Qing Chen, Gino Salituro, Yusheng Xiong, Daniel R. McMasters, Mary Struthers, Ning Ren, Ruth A. Duffy
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:2384-2388
مصطلحات موضوعية: Male, 0301 basic medicine, Aldosterone synthase, Indazoles, Clinical Biochemistry, High selectivity, Pharmaceutical Science, Pharmacology, 01 natural sciences, Biochemistry, Cell Line, Rats, Sprague-Dawley, 03 medical and health sciences, chemistry.chemical_compound, Cricetulus, Pharmacokinetics, Cytochrome P-450 CYP2D6 Inhibitors, Drug Discovery, Animals, Cytochrome P-450 CYP11B2, Humans, Molecular Biology, Antihypertensive Agents, Indazole, biology, Aromatase Inhibitors, Chemistry, Organic Chemistry, Stereoisomerism, Hit to lead, Macaca mulatta, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 030104 developmental biology, Hypertension, biology.protein, Steroid 11-beta-Hydroxylase, Molecular Medicine
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3
المؤلفون: Brent R. Whitehead, Michael M.-C. Lo, Amjad Ali, Min K. Park, Scott B. Hoyt, Yusheng Xiong, Jiaqiang Cai, Emma Carswell, Andrew Cooke, John MacLean, Paul Ratcliffe, John Robinson, D. Jonathan Bennett, Joseph A. Clemas, Tom Wisniewski, Mary Struthers, Doris Cully, Douglas J. MacNeil
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:143-146
مصطلحات موضوعية: Male, Aldosterone synthase, medicine.medical_specialty, Pyridines, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Structure-Activity Relationship, Cricetulus, Internal medicine, Drug Discovery, medicine, Animals, Cytochrome P-450 CYP11B2, Humans, Rats, Wistar, Molecular Biology, biology, 010405 organic chemistry, Chemistry, Organic Chemistry, Imidazoles, Macaca mulatta, humanities, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Endocrinology, Microsomes, Liver, biology.protein, Steroid 11-beta-Hydroxylase, Molecular Medicine
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4
المؤلفون: Chris J. van Koppen, Scott B. Hoyt, Gino Salituro, Elaine Tung, Jim Tata, Joe Clemas, Mark Rosenbach, Jack Gibson, Daphne Szeto, Wei Tang, Andreas Verras, Lee-Yuh Pai, Ning Ren, Carrie Ann Maxwell, Joe Metzger, Jose Castro-Perez, Qing Chen, Lina Yin, Daniel R. McMasters, Yusheng Xiong, Rolf W. Hartmann, Mary Struthers, Gui-Bai Liang, Charlene Bopp, Xiuying Ma, Gaochao Zhou, Richard Hajdu, Tom Wisniewski, Mike E. Lassman, Nicole Buist, Clare London, Andrea Sok, Gail Forrest, Sloan Stribling, Theresa McLaughlin, Qingzhong Hu, Tian-Quan Cai, Whitney Lane Petrilli
المصدر: ACS Medicinal Chemistry Letters. 6:861-865
مصطلحات موضوعية: Aldosterone synthase, medicine.medical_specialty, Aldosterone, Organic Chemistry, Triazole, Hit to lead, Biology, Pharmacology, Biochemistry, chemistry.chemical_compound, Endocrinology, chemistry, Pharmacokinetics, In vivo, Pharmacodynamics, Internal medicine, Drug Discovery, medicine, biology.protein, Cortisol level
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5
المؤلفون: Daphne Szeto, Doris F. Cully, Scott B. Hoyt, Ning Ren, Elaine Tung, Charlene Bopp, Jack Gibson, Gino Salituro, Clare London, Jiaqiang Cai, Amjad Ali, Qing Chen, Andrea Sok, Simone Belshaw, Carrie Ann Maxwell, Mark Rosenbach, Gaochao Zhou, Gail Forrest, Tian-Quan Cai, Daniel R. McMasters, Lee-Yuh Pai, Nelo R. Rivera, Sloan Stribling, Emma Carswell, Richard Hajdu, Robinson John E, Andrew J. Cooke, Jeff Kuethe, Tom Wisniewski, Joe Metzger, Thomas R. Clarkson, Gui-Bai Liang, Mary Struthers, Jim Tata, Mike E. Lassman, Lindsay Brown, Wei Tang, Theresa McLaughlin, Xiuying Ma, Nicole Buist, Kun Liu, Joe Clemas, D. Jonathan Bennett, Andreas Verras, Min K. Park, Yusheng Xiong, John Maclean, Jose Castro-Perez
مصطلحات موضوعية: Aldosterone synthase, Benzimidazole, medicine.medical_specialty, Aldosterone, Organic Chemistry, High selectivity, Biology, Pharmacology, Biochemistry, chemistry.chemical_compound, Endocrinology, chemistry, Pharmacokinetics, In vivo, Internal medicine, Pharmacodynamics, Drug Discovery, medicine, biology.protein, Cortisol level
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::02bdb44414988404f1b182298b88bcd9
https://europepmc.org/articles/PMC4434468/