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1
المؤلفون: Shin-ichi Inoue, Shoko Honzumi, Nagaoka Nobumi, Tomoko Ogiyama, Yuka Yamamoto, Mitsuhiro Yamaguchi, Nobuya Kurikawa, Daisuke Sugiyama, Takako Kimura, Koji Terayama
المصدر: Bioorganic & Medicinal Chemistry. 25:4817-4828
مصطلحات موضوعية: Glycerol, Male, 0301 basic medicine, Aché, Clinical Biochemistry, Cell, Administration, Oral, Pharmaceutical Science, Hormone-sensitive lipase, Inhibitory postsynaptic potential, 01 natural sciences, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Humans, Lipolysis, Enzyme Inhibitors, Rats, Wistar, Molecular Biology, Hypolipidemic Agents, chemistry.chemical_classification, 010405 organic chemistry, Chemistry, Organic Chemistry, food and beverages, Sterol Esterase, Glutathione, Recombinant Proteins, language.human_language, In vitro, Rats, 0104 chemical sciences, Enzyme Activation, 030104 developmental biology, Enzyme, medicine.anatomical_structure, Butyrylcholinesterase, Drug Design, Acetylcholinesterase, language, Molecular Medicine, Lead compound, Half-Life
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2
المؤلفون: Tomoko Ogiyama, Shoko Honzumi, Shin-ichi Inoue, Nobuya Kurikawa, Mitsuhiro Yamaguchi, Daisuke Sugiyama, Yuka Yamamoto
المصدر: Bioorganic & Medicinal Chemistry. 24:3801-3807
مصطلحات موضوعية: Male, 0301 basic medicine, Spectrometry, Mass, Electrospray Ionization, Proton Magnetic Resonance Spectroscopy, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Hormone-sensitive lipase, 01 natural sciences, Biochemistry, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Oral administration, Drug Discovery, Sterol esterase, Animals, Structure–activity relationship, Lipolysis, Enzyme Inhibitors, Rats, Wistar, Molecular Biology, IC50, Dose-Response Relationship, Drug, 010405 organic chemistry, Organic Chemistry, food and beverages, Sterol Esterase, Boronic Acids, Rats, 0104 chemical sciences, 030104 developmental biology, chemistry, Molecular Medicine, Selectivity, Boronic acid
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3
المؤلفون: Toshiyuki Nakanishi, Madoka Hoshino, Yu Ohki, Kazuishi Kubota, Hiroki Shimizu, Hideki Kobayashi, Tomio Ishikawa, Hidetaka Sakurai, Yasunori Muramatsu, Hiroyuki Tsuruoka, Tomoko Ogiyama, Hideki Terashima, Shojiro Miyazaki
المصدر: Cell chemical biology. 26(1)
مصطلحات موضوعية: Male, Proteomics, Clinical Biochemistry, Computational biology, Biology, 01 natural sciences, Biochemistry, Correlation, Small Molecule Libraries, Drug Discovery, Gene silencing, Humans, Gene Silencing, Enzyme Inhibitors, RNA, Small Interfering, Molecular Biology, Intramolecular Transferases, Cells, Cultured, Pharmacology, Molecular Structure, 010405 organic chemistry, Drug discovery, Gene Expression Profiling, Phenotype, Small molecule, 0104 chemical sciences, Molecular targets, biology.protein, Molecular Medicine, Deconvolution, Lanosterol synthase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::665d5079cf04843f0ae211a9a73dd37e
https://pubmed.ncbi.nlm.nih.gov/30449674 -
4
المؤلفون: Nobuya Kurikawa, Hideo Takakusa, Yuka Yamamoto, Daisuke Sugiyama, Shoko Honzumi, Mitsuhiro Yamaguchi, Shin-ichi Inoue, Tomoko Ogiyama
المصدر: Bioorganicmedicinal chemistry. 25(7)
مصطلحات موضوعية: 0301 basic medicine, Male, Spectrometry, Mass, Electrospray Ionization, Proton Magnetic Resonance Spectroscopy, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Hormone-sensitive lipase, Inhibitory postsynaptic potential, 01 natural sciences, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Inhibitory Concentration 50, Oral administration, Drug Discovery, Animals, Enzyme Inhibitors, Rats, Wistar, Molecular Biology, IC50, Dyslipidemias, 010405 organic chemistry, Organic Chemistry, Benzanilide, Sterol Esterase, 0104 chemical sciences, Rats, 030104 developmental biology, chemistry, Reactive metabolite, Molecular Medicine, Linker, Derivative (chemistry)