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1
المؤلفون: Maureen Caligiuri, Grace L. Williams, Jennifer Castro, Linda Battalagine, Erik Wilker, Lili Yao, Shawn Schiller, Angela Toms, Ping Li, Eneida Pardo, Bradford Graves, Joey Azofeifa, Agustin Chicas, Torsten Herbertz, Maria Lai, Joel Basken, Kenneth W. Wood, Qunli Xu, Sylvie M. Guichard
المصدر: Targeted Oncology. 18:269-285
مصطلحات موضوعية: Cancer Research, Oncology, Pharmacology (medical)
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2
المؤلفون: Bruce Follows, Shawn Fessler, Timm Baumeister, Ann-Marie Campbell, Mary Margaret Zablocki, Hongbin Li, Deepali Gotur, Zhongguo Wang, Xiaozhang Zheng, Lisa Molz, Cokey Nguyen, Torsten Herbertz, Liann Wang, Kenneth Bair
المصدر: Bioorganic & Medicinal Chemistry Letters. 29:2375-2382
مصطلحات موضوعية: Models, Molecular, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Drug Discovery, Humans, Myeloid Cell Leukemia Sequence 1 Protein, Molecular Medicine, Molecular Biology
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3
المؤلفون: Grace L. Williams, Shawn Schiller, Monica A. Alvarez Morales, Crystal McKinnon, Matthew W. Martin, George P. Luke, Torsten Herbertz, Adam C. Talbot, Stephen Hubbs, Katherine J. Kayser-Bricker, Daniel Cardillo, Paul Troccolo, David S. Millan, Rachel L. Mendes
المصدر: ACS Medicinal Chemistry Letters. 8:847-852
مصطلحات موضوعية: 0301 basic medicine, Cellular activity, Chemistry, Organic Chemistry, A protein, Biochemistry, Combinatorial chemistry, Small molecule, Bromodomain, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Mouse xenograft, In vivo, Lipophilic efficiency, 030220 oncology & carcinogenesis, Drug Discovery, Binding site
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4
المصدر: ACS Chemical Neuroscience
مصطلحات موضوعية: Drug, Physiology, Research areas, Cognitive Neuroscience, media_common.quotation_subject, Central nervous system, Disease, chemoinformatics, Biochemistry, Brain cancer, chemical substructures, Medicine, solvent accessible surface area, media_common, molecular volume, Drug discovery, business.industry, non-CNS drugs, Cell Biology, General Medicine, physicochemical property profile, aliphatic amine, medicine.anatomical_structure, linear chains, Aliphatic amine, polar hydrogen, CNS, polar surface area, business, CNS drugs, Neuroscience, Research Article
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5
المؤلفون: Randy W. Jackson, Matthew G. LaPorte, Torsten Herbertz, Tandy L. Draper, Janet A. Gaboury, Susan R. Rippin, Ravi Patel, Srinivas K. Chunduru, Christopher A. Benetatos, Dorothy C. Young, Christopher J. Burns, Stephen M. Condon
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3227-3231
مصطلحات موضوعية: Models, Molecular, Indoles, Molecular Structure, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, Crystallography, X-Ray, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, Drug Discovery, Molecular Medicine, Enzyme Inhibitors, Molecular Biology, Allosteric Site, Pyrans
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6
المؤلفون: Deborah Galinis, Sheila J. Miknyoczki, Ted L. Underiner, Damaris Rolon-Steele, Jean Husten, Craig A. Zificsak, Thelma S. Angeles, Torsten Herbertz, Mark S. Albom, Bruce D. Dorsey, Laura S. Kocsis, Kevin J. Wells-Knecht, Jay P. Theroff, Lisa D. Aimone, Kelli S. Zeigler, Candace S. Worrell, Rebecca A. Brown, Christine LoSardo, Seetha Murthy, Jennifer Grobelny
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:660-663
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Metabolite, Clinical Biochemistry, Substituent, Administration, Oral, Mice, Nude, Pharmaceutical Science, Antineoplastic Agents, Carboxamide, Biochemistry, Chemical synthesis, Mice, chemistry.chemical_compound, In vivo, Neoplasms, Drug Discovery, medicine, Animals, Humans, Protein Kinase Inhibitors, Molecular Biology, biology, Bicyclic molecule, Chemistry, Organic Chemistry, Proto-Oncogene Proteins c-met, Xenograft Model Antitumor Assays, Pyrimidines, Diaminopyrimidine, Enzyme inhibitor, biology.protein, Molecular Medicine
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7
المؤلفون: Eugene C. Amparo, Srinivas K. Chunduru, Ariamala Gopalsamy, Christopher A. Benetatos, Lori E. Miller, Tandy L. Draper, Christopher J. Burns, Matthew G. LaPorte, Lara K. Leister, Torsten Herbertz, Dorothy C. Young, Stephen M. Condon, Blackledge Charles W, Gerry Rhodes, Alison R. Hussey
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:2968-2973
مصطلحات موضوعية: Indoles, Stereochemistry, Hepatitis C virus, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Viral Nonstructural Proteins, Crystallography, X-Ray, medicine.disease_cause, Antiviral Agents, Biochemistry, Virus, Structure-Activity Relationship, Drug Discovery, medicine, Structure–activity relationship, Enzyme Inhibitors, Binding site, Molecular Biology, Pyrans, chemistry.chemical_classification, Indole test, Binding Sites, biology, Organic Chemistry, virus diseases, digestive system diseases, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
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8
المؤلفون: Sheila J. Miknyoczki, Torsten Herbertz, Ted L. Underiner
المصدر: Anti-Cancer Agents in Medicinal Chemistry. 10:7-27
مصطلحات موضوعية: Models, Molecular, Pharmacology, Cancer Research, C-Met, Drug discovery, Angiogenesis, Antineoplastic Agents, Proto-Oncogene Proteins c-met, Biology, Ligands, Bioinformatics, Small molecule, Paracrine signalling, chemistry.chemical_compound, chemistry, Drug Discovery, Cancer research, medicine, Animals, Humans, Molecular Medicine, Hepatocyte growth factor, Kinase activity, Autocrine signalling, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a06afc09f2777a1329ec565f923b48a
https://doi.org/10.2174/1871520611009010007 -
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المؤلفون: Daniel C. Pevear, Dorothy C. Young, Christopher A. Benetatos, Glen A. Coburn, Susan R. Rippin, Christopher J. Burns, Marc S. Collett, Christopher J. Rizzo, Joel S. Christensen, Tandy L. Draper, Tiejun Gao, John O'Connell, Stephen M. Condon, Kristin Galie, Alison R. Hussey, Srinivas K. Chunduru, Gerry Rhodes, Norman M. Kneteman, Janet A. Gaboury, Tarek S. Mansour, Randy W. Jackson, D. Lorne Tyrrell, Anita Y. M. Howe, Matthew G. LaPorte, Torsten Herbertz
المصدر: ChemMedChem. 3:1508-1515
مصطلحات موضوعية: Indoles, Allosteric regulation, Mice, Transgenic, Hepacivirus, Mice, SCID, Viral Nonstructural Proteins, Antiviral Agents, Biochemistry, Ns5b polymerase, Inhibitory Concentration 50, Mice, Allosteric Regulation, In vivo, Drug Discovery, Animals, General Pharmacology, Toxicology and Pharmaceutics, Pyrans, Pharmacology, Indole test, Chemistry, Organic Chemistry, RNA-Dependent RNA Polymerase, Virology, RNA, Viral, Molecular Medicine
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10
المصدر: Journal of Medicinal Chemistry. 51:5149-5171
مصطلحات موضوعية: Drug, media_common.quotation_subject, Quantitative Structure-Activity Relationship, Pharmacology, Ligands, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Databases, Protein, Benzamide, Phosphorylase kinase, Protein Kinase Inhibitors, media_common, Binding Sites, biology, Chemistry, Drug discovery, Kinase, Imatinib, Biochemistry, Drug Design, Mitogen-activated protein kinase, biology.protein, Molecular Medicine, Signal transduction, medicine.drug