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1دورية أكاديميةEffect of ASP2151, a Herpesvirus Helicase-Primase Inhibitor, in a Guinea Pig Model of Genital Herpes
المؤلفون: Toru Kontani, Yasuaki Shimizu, Kenji Sudo, Koji Chono, Kiyomitsu Katsumata, Hiroshi Suzuki
المصدر: Molecules, Vol 16, Iss 9, Pp 7210-7223 (2011)
مصطلحات موضوعية: ASP2151, amenamevir, antiviral, HSV, guinea pig, genital herpes, Organic chemistry, QD241-441
وصف الملف: electronic resource
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المؤلفون: Hiroshi Inami, Tsuyoshi Mizutani, Junko Watanabe, Hisashi Hayashida, Tomonori Ito, Takeshi Terasawa, Toru Kontani, Hiroaki Yamagishi, Hiroyuki Usuda, Naohiro Aoyama, Emiko Imamura, Takeshi Ishikawa
المصدر: Bioorganic & Medicinal Chemistry. 87:117302
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry
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المؤلفون: Toru Kontani, Yoshiaki Ohtsu, Kota Kato, Koji Chono, Kiyomitsu Katsumata, Shoji Takakura, Hiroshi Suzuki
المصدر: Antimicrobial Agents and Chemotherapy. 57:1339-1346
مصطلحات موضوعية: viruses, DNA Primase, Herpesvirus 1, Human, Viral Plaque Assay, Biology, Pharmacology, Virus Replication, medicine.disease_cause, Antiviral Agents, Drug Administration Schedule, Mice, Viral Proteins, Pharmacokinetics, medicine, Animals, Pharmacology (medical), Amenamevir, Enzyme Inhibitors, Skin, Mice, Hairless, Oxadiazoles, Dose-Response Relationship, Drug, DNA Helicases, Varicella zoster virus, Dose fractionation, Herpes Simplex, Titer, Dose–response relationship, Infectious Diseases, Herpes simplex virus, Area Under Curve, Pharmacodynamics, Female
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::da69367dc83195739db7085fab4f2e57
https://doi.org/10.1128/aac.01803-12 -
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المؤلفون: Hiroshi Suzuki, Toru Kontani, Kiyomitsu Katsumata, Adriana Weinberg, Shoji Takakura, Koji Chono
المصدر: Antimicrobial Agents and Chemotherapy. 56:3587-3591
مصطلحات موضوعية: Simplexvirus, food.ingredient, viruses, Acyclovir, Phases of clinical research, DNA Primase, HSL and HSV, Biology, medicine.disease_cause, Antiviral Agents, Virus, Viral Proteins, food, medicine, Humans, Pharmacology (medical), Amenamevir, Enzyme Inhibitors, Herpes Genitalis, Pharmacology, Oxadiazoles, DNA Helicases, virus diseases, Virology, Infectious Diseases, Herpes simplex virus, Primase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6188241d14870d4f114ddf3706a4261a
https://doi.org/10.1128/aac.00133-12 -
5Effect of ASP2151, a Herpesvirus Helicase-Primase Inhibitor, in a Guinea Pig Model of Genital Herpes
المؤلفون: Yasuaki Shimizu, Kiyomitsu Katsumata, Toru Kontani, Koji Chono, Hiroshi Suzuki, Kenji Sudo
المصدر: Molecules; Volume 16; Issue 9; Pages: 7210-7223
Molecules
Molecules, Vol 16, Iss 9, Pp 7210-7223 (2011)مصطلحات موضوعية: Herpesvirus 2, Human, viruses, Drug Evaluation, Preclinical, Acyclovir, amenamevir, Pharmaceutical Science, Herpesvirus 1, Human, Viral Plaque Assay, medicine.disease_cause, Analytical Chemistry, Drug Discovery, Oxadiazoles, HSV, virus diseases, Valine, Viral Load, antiviral, Effective dose (pharmacology), Virus Shedding, Chemistry (miscellaneous), Area Under Curve, Valacyclovir, genital herpes, Molecular Medicine, Female, Guinea Pigs, ASP2151, guinea pig, DNA Primase, Antiviral Agents, Article, lcsh:QD241-441, Viral Proteins, lcsh:Organic chemistry, medicine, Animals, Potency, Amenamevir, Physical and Theoretical Chemistry, Viral shedding, Herpes Genitalis, business.industry, Organic Chemistry, DNA Helicases, Varicella zoster virus, Virology, Herpes simplex virus, Vero cell, business
وصف الملف: application/pdf
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المؤلفون: Ayako Moritomo, Mitsuaki Ohta, Shunji Kageyama, Toru Kontani, Osamu Yamamoto, Naoyuki Masuda, Tetsuro Ohgami, Masahiro Fujii
المصدر: Synthetic Communications. 35:2305-2316
مصطلحات موضوعية: chemistry.chemical_classification, chemistry, Organic Chemistry, Regioselectivity, Organic chemistry, General Medicine, Alkylation, Combinatorial chemistry, Sulfonamide
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المؤلفون: Masamichi Sakai, Toru Kontani, Keishi Takeyama, Koki Takanashi, Yoshihisa Obi, Osamu Nakamura, Yoshiya Uwatoko
المصدر: Japanese Journal of Applied Physics. 43:681-687
مصطلحات موضوعية: Physics and Astronomy (miscellaneous), Condensed matter physics, Hydrogen, Carrier scattering, General Engineering, General Physics and Astronomy, chemistry.chemical_element, Yttrium, Thermal conduction, Optical conductivity, chemistry, Electrical resistivity and conductivity, Hall effect, Electrical measurements
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المؤلفون: Ayako Moritomo, Tadatsura Koshika, Toru Kontani, Yuji Matsushima, Hiroshi Nagata, Hisao Hamaguchi, Shinya Nagashima, Makoto Takeuchi
المصدر: Bioorganicmedicinal chemistry. 22(13)
مصطلحات موضوعية: Male, Models, Molecular, medicine.medical_specialty, Quinuclidines, Clinical Biochemistry, Rat model, Pharmaceutical Science, Pharmacology, Biochemistry, Rats, Sprague-Dawley, Structure-Activity Relationship, Internal medicine, Drug Discovery, Muscarinic acetylcholine receptor, medicine, Muscarinic acetylcholine receptor M4, Animals, Molecular Biology, Receptor, Muscarinic M3, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Muscarinic antagonist, Muscarinic acetylcholine receptor M3, Tiotropium bromide, Muscarinic acetylcholine receptor M1, Rats, Endocrinology, Molecular Medicine, Bronchoconstriction, Carbamates, medicine.symptom, medicine.drug
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المؤلفون: Hiroshi Suzuki, Koji Chono, Kimiyasu Shiraki, Kiyomitsu Katsumata, Toru Kontani
المصدر: Biochemical pharmacology. 84(4)
مصطلحات موضوعية: viruses, Herpesvirus 2, Human, Mutant, Molecular Sequence Data, DNA Primase, Herpesvirus 1, Human, Viral Plaque Assay, Biology, medicine.disease_cause, Biochemistry, Antiviral Agents, Virus, Mice, Viral Proteins, Chlorocebus aethiops, Drug Resistance, Viral, medicine, Animals, Humans, Amenamevir, Amino Acid Sequence, Cells, Cultured, Pharmacology, Mice, Hairless, Oxadiazoles, DNA Helicases, Helicase, Herpes Simplex, Virology, Molecular biology, Helicase Gene, Herpes simplex virus, Viral replication, Amino Acid Substitution, Mutation, biology.protein, Female, Primase
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المؤلفون: Tokio Yamaguchi, Tamako Nomura, Shin-ichi Tsukamoto, Ryo Naito, Toshiyasu Mase, Tomoyuki Yasunaga, Toru Kontani
المصدر: ChemInform. 28
مصطلحات موضوعية: Chemistry, Stereochemistry, 5-HT1A receptor, General Medicine, Antagonism, Receptor antagonist activity, Butylamines