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1
المؤلفون: Jeffrey C. Jerman, Derek N. Middlemiss, Martyn C. Coldwell, Darren Smart, Stephen J. Brough, Tracey Gager, Martyn D. Wood
المصدر: European Journal of Pharmacology. 414:23-30
مصطلحات موضوعية: Agonist, medicine.medical_specialty, medicine.drug_class, Receptor expression, Biology, Pharmacology, Partial agonist, Cell Line, chemistry.chemical_compound, Internal medicine, Receptor, Serotonin, 5-HT2B, Receptor, Serotonin, 5-HT2C, medicine, Enzyme-linked receptor, Humans, Inverse agonist, Receptor, Serotonin, 5-HT2A, Receptor, Dose-Response Relationship, Drug, Sodium butyrate, Serotonin Receptor Agonists, Butyrates, Endocrinology, chemistry, Receptors, Serotonin, Serotonin Antagonists, Endogenous agonist
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2
المؤلفون: Derek N. Middlemiss, Helen Newman, Stephen E. Clarke, Graham J. Riley, Carol Routledge, Tracey Gager, Gary W. Price, Steven Mark Bromidge, Warren D. Hirst, Tania O. Stean, Neil Upton, Anthony M. C. Brown, Stephen Moss
المصدر: British Journal of Pharmacology. 130:1606-1612
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, SB-258585, Seizure threshold, medicine.drug_class, Antagonist, Stimulation, Biology, Receptor antagonist, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, SB-271046, 5-HT6 receptor, medicine, Receptor
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3
المؤلفون: Anthony M. C. Brown, Heinz H. Pertz, Tracey Gager, Alberto J. Kaumann
المصدر: Journal of Pharmacy and Pharmacology. 51:319-330
مصطلحات موضوعية: Male, Agonist, Stereochemistry, medicine.drug_class, Inositol Phosphates, Methysergide, Pharmaceutical Science, In Vitro Techniques, Binding, Competitive, Partial agonist, Structure-Activity Relationship, chemistry.chemical_compound, Lysergol, Receptors, Adrenergic, alpha-1, medicine, Animals, Ergolines, Rats, Wistar, Inositol phosphate, Receptor, Pharmacology, chemistry.chemical_classification, Biological activity, Arteries, Rats, Serotonin Receptor Agonists, Ergoline, chemistry, Serotonin Antagonists, Antipsychotic Agents, medicine.drug
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4
المؤلفون: Jeffrey C. Jerman, Derek N. Middlemiss, Martyn C. Coldwell, A. J. Hunter, Jeannette M. Watson, Stephen J. Brough, Graham J. Riley, Anthony M. C. Brown, M. Ho, Tracey Gager
المصدر: British Journal of Pharmacology. 125:1413-1420
مصطلحات موضوعية: Pharmacology, Agonist, medicine.medical_specialty, medicine.drug_class, Partial agonist, Pirenzepine, chemistry.chemical_compound, Endocrinology, chemistry, Himbacine, Internal medicine, Muscarinic acetylcholine receptor, medicine, Xanomeline, Receptor, 5-HT receptor, medicine.drug
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5
المؤلفون: Helen Newman, Stephen E. Clarke, Steven Mark Bromidge, Halina T Serafinowska, Kerry Griffith, Peter J. Lovell, Tracey Gager, Douglas R Smith, Graham J. Riley, Carol Routledge, Andrew John Jennings, Stephen Moss, Phillip Jeffrey, Graham Francis Joiner, Derek C. Rogers, Frank D. King
المصدر: Bioorganicmedicinal chemistry letters. 11(1)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Biological Availability, Biochemistry, Chemical synthesis, Piperazines, Cns penetration, Substrate Specificity, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Structure–activity relationship, Animals, Humans, Serotonin Antagonists, Molecular Biology, Sulfonamides, Molecular Structure, Organic Chemistry, SB-357134, In vitro, Bioavailability, Rats, chemistry, Blood-Brain Barrier, Receptors, Serotonin, Molecular Medicine, Selectivity
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6
المؤلفون: Derek N. Middlemiss, Helen Newman, Tracey Gager, P. Jeffrey, Stephen Moss, Graham J. Riley, Carol Routledge, Wyman Paul Adrian, Anthony M. Brown, Helen L. Grassam, Graham Francis Joiner, Steven Mark Bromidge, Frank King, Kathy Dodgson, Stephen E. Clarke
المصدر: Journal of medicinal chemistry. 42(2)
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonamides, Bicyclic molecule, Stereochemistry, Antagonist, Benzothiophene, Administration, Oral, Biological Availability, Thiophenes, Chemical synthesis, Sulfonamide, Cell Line, Rats, chemistry.chemical_compound, chemistry, Amide, SB-271046, Receptors, Serotonin, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Animals, Humans, Serotonin Antagonists