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1
المؤلفون: Maki Seki, Tsuyoshi Ogiku
المصدر: Tetrahedron. 70:3864-3870
مصطلحات موضوعية: Enantiopure drug, Tandem, Chemistry, Stereochemistry, Organic Chemistry, Drug Discovery, Optically active, Ring (chemistry), Biochemistry, Phenylalanine derivatives
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2
المؤلفون: Hiroshi Sai, Tsuyoshi Ogiku, Hiroshi Miyazaki, Hiroshi Ohmizu, Jun Murakami, Akio Ohtani
المصدر: Bioorganic & Medicinal Chemistry. 18:1968-1979
مصطلحات موضوعية: Serine Proteinase Inhibitors, Clinical Biochemistry, Molecular Conformation, Administration, Oral, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Phenylbutyrate, Molecular conformation, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Fibrinolytic Agents, Bleeding time, Plasminogen Activator Inhibitor 1, Drug Discovery, Antithrombotic, Butadienes, medicine, Animals, Structure–activity relationship, Molecular Biology, Cells, Cultured, medicine.diagnostic_test, Chemistry, Organic Chemistry, Phenylbutyrates, Rats, Plasminogen activator inhibitor-1, Molecular Medicine, Fibrinolytic agent
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3
المؤلفون: Koichi Fukase, Tsuyoshi Ogiku, Kunio Saruta
المصدر: Tetrahedron Letters. 50:4364-4367
مصطلحات موضوعية: chemistry.chemical_classification, Sulfonium, Organic Chemistry, Alkylation, Biochemistry, Combinatorial chemistry, Sulfonamide, chemistry.chemical_compound, Solid-phase synthesis, chemistry, Intramolecular force, Drug Discovery, Microwave irradiation, Organic chemistry
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4
المؤلفون: Tsuyoshi Ogiku, Hiroshi Miyazaki, Hiroshi Ohmizu
المصدر: Organic Process Research & Development. 13:760-763
مصطلحات موضوعية: In situ, chemistry.chemical_compound, chemistry, Stereochemistry, Plasminogen activator inhibitor-1, Organic Chemistry, Physical and Theoretical Chemistry, Selectivity, Isomerization, Plasminogen activator, Derivative (chemistry)
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5
المؤلفون: Akio Ohtani, Hiroshi Miyazaki, Tsuyoshi Ogiku, Jun Murakami, Hiroshi Ohmizu, Hiroshi Sai
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:6419-6422
مصطلحات موضوعية: Chemistry, Pharmaceutical, Clinical Biochemistry, Drug Evaluation, Preclinical, Administration, Oral, Biological Availability, Succinimides, Pharmaceutical Science, Benzylidene Compounds, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Dogs, Oral administration, Plasminogen Activator Inhibitor 1, Drug Discovery, Antithrombotic, Animals, Humans, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Drug Administration Routes, Organic Chemistry, In vitro, Rats, Bioavailability, Enzyme, Models, Chemical, Solubility, Enzyme inhibitor, Drug Design, Plasminogen activator inhibitor-1, biology.protein, Molecular Medicine
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6
المؤلفون: Tsuyoshi Ogiku, James Zapf, Shao-Hui Zhang, Kui Xu, Kei Takedomi, Naoki Sakurai, Guang Yang, Rick Jack, Jie-Fei Cheng, Miguel Barbosa, Chiaki Fukushima
المصدر: Journal of Medicinal Chemistry. 51:2057-2061
مصطلحات موضوعية: Models, Molecular, Benzylamines, Hydrocarbons, Fluorinated, Receptors, Cytoplasmic and Nuclear, Ligands, Benzoates, Structure-Activity Relationship, Phenazocine, Drug Discovery, Coactivator, Computer Simulation, RNA, Messenger, Liver X receptor, Liver X Receptors, Oligonucleotide Array Sequence Analysis, Sulfonamides, Virtual screening, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, biology, Chemistry, Gene Expression Profiling, Orphan Nuclear Receptors, Cell biology, DNA-Binding Proteins, Gene expression profiling, Sterols, ABCG1, Biochemistry, Nuclear receptor, Docking (molecular), ABCA1, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins)
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7
المؤلفون: Tsuyoshi Ogiku, Kunio Saruta
المصدر: Tetrahedron Letters. 49:424-427
مصطلحات موضوعية: chemistry.chemical_compound, Solid-phase synthesis, Chemistry, Sulfonium, Phase (matter), Intramolecular force, Organic Chemistry, Drug Discovery, Alkylation, Biochemistry, Combinatorial chemistry
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8
المؤلفون: Tsuyoshi Ogiku, Hiroshi Ohmizu, Hiroshi Sai
المصدر: Tetrahedron. 63:10345-10353
مصطلحات موضوعية: Reaction mechanism, Chemistry, Organic Chemistry, Biochemistry, Medicinal chemistry, chemistry.chemical_compound, Stereospecificity, Deprotonation, Dehydration reaction, Drug Discovery, Copper(II) chloride, Cinnamates, 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide, Stereoselectivity
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9
المؤلفون: Maki Seki, Tsuyoshi Ogiku
المصدر: ChemInform. 45
مصطلحات موضوعية: Enantiopure drug, Tandem, Stereochemistry, Chemistry, General Medicine, Optically active, Ring (chemistry), Phenylalanine derivatives
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10
المؤلفون: Ming-Wei Wang, Xin Hui, Jie Gao, Tsuyoshi Ogiku, Xin Xie, Naoki Suto
المصدر: Acta Pharmacologica Sinica. 26:1175-1180
مصطلحات موضوعية: Pharmacology, Stereochemistry, Chemistry, Ligand binding assay, High-throughput screening, Kidney metabolism, General Medicine, Wheat germ agglutinin, Cytisine, chemistry.chemical_compound, Nicotinic acetylcholine receptor, Scintillation proximity assay, Biochemistry, Epibatidine, medicine, Pharmacology (medical), medicine.drug