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1دورية أكاديمية
المؤلفون: V.R. Knight-Schrijver, V. Chelliah, L. Cucurull-Sanchez, N. Le Novère
المصدر: Computational and Structural Biotechnology Journal, Vol 14, Iss C, Pp 363-370 (2016)
مصطلحات موضوعية: Quantitative systems pharmacology, QSP, Drug discovery, Modelling, Systems biology, New therapeutic entity, Biotechnology, TP248.13-248.65
وصف الملف: electronic resource
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2
المؤلفون: Charles Lee Jayne, Santhosh Neelamkavil, Alan Hruza, Richard N. Ingram, Samuel Chackalamannil, Mariappan V. Chelliah, Keith Eagen, Teresa Andreani, William J. Greenlee, Kartik M. Keertikar, Steve Fried, Brian Hawes, Yan Xia, Zhuyan Guo, Michael P. Dwyer, Tin-Yau Chan, Paul Reichert, Martin C. Clasby
المصدر: Bioorganicmedicinal chemistry letters. 30(15)
مصطلحات موضوعية: Pyrimidine, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, 01 natural sciences, Biochemistry, Factor IXa, chemistry.chemical_compound, Structure-Activity Relationship, In vivo, Drug Discovery, Structure–activity relationship, Humans, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Chemistry, Organic Chemistry, Plasma levels, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Pyrimidines, Molecular Medicine, Selectivity, Factor Xa Inhibitors
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3
المؤلفون: Mariappan V. Chelliah, Ian W. Davies, Yan Xia, John A. Howe, Srikanth Venkatraman, Shah Unmesh G, Francisco Velazquez, Randy R. Miller, Samuel Chackalamannil, Santhosh Neelamkavil, Zhuyan Guo, Martin C. Clasby, Aileen Soriano
المصدر: ACS Medicinal Chemistry Letters. 7:1173-1178
مصطلحات موضوعية: NS3, Molecular model, 010405 organic chemistry, Stereochemistry, Chemistry, Organic Chemistry, 010402 general chemistry, 01 natural sciences, Biochemistry, 0104 chemical sciences, Genotype 1b, Grazoprevir, Drug Discovery, Moiety, Proline
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4
المؤلفون: Samuel Chackalamannil, Mariappan V. Chelliah
المصدر: Lead Generation
مصطلحات موضوعية: medicine.medical_specialty, business.industry, Fda approval, medicine, Identification (biology), Intensive care medicine, business, Vorapaxar, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c27c782d3362f785bde05a524fbb0f5a
https://doi.org/10.1002/9783527677047.ch19 -
5
المؤلفون: Keith Eagen, Yunsheng Hsieh, Mariappan V. Chelliah, Stan Kurowski, Zhuyan Guo, Madhu Chintala, William J. Greenlee, Hsingan Tsai, Samuel Chackalamannil, Ho-Sam Ahn, Yan Xia, George Boykow
المصدر: ACS Medicinal Chemistry Letters. 5:561-565
مصطلحات موضوعية: Organic Chemistry, Plasma levels, Biochemistry, Combinatorial chemistry, In vitro, chemistry.chemical_compound, Par 1 antagonist, chemistry, Himbacine, Drug Discovery, Thrombin receptor, medicine, Receptor, Vorapaxar, medicine.drug
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6
المؤلفون: Stan Kurowski, Mariappan V. Chelliah, William J. Greenlee, Madhu Chintala, Yunsheng Hsieh, Yan Xia, George Boykow, Ho-Sam Ahn, Samuel Chackalamannil
المصدر: ACS Medicinal Chemistry Letters. 5:183-187
مصطلحات موضوعية: Platelet aggregation, business.industry, education, Organic Chemistry, Pharmacology, Biochemistry, humanities, In vitro binding, chemistry.chemical_compound, Par 1 antagonist, chemistry, Pharmacokinetics, Himbacine, Drug Discovery, Thrombin receptor, medicine, business, Ex vivo, Vorapaxar, medicine.drug
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7دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
8
المؤلفون: Christopher Joseph Sinz, Sarah Souza, Aimie M. Ogawa, Dennis Leung, Eric R. Ashley, Brande Thomas-Fowlkes, Maria Madeira, Mary Ann Powles, Effie Tozzo, Hong D. Chu, Feroze Ujjainwalla, Melissa Kirkland, Matthew Lombardo, Clare London, Jerry Di Salvo, Keith Eagen, John S. Debenham, Jason M. Cox, Ping Lan, Alejandro Crespo, Adam B. Weinglass, Taro E. Akiyama, Nengxue Wang, Henry M. Vaccaro, Michele Pachanski, Shah Unmesh G, Zhongxiang Sun, Mariappan V. Chelliah, James R. Tata, Michael A. Plotkin, Candice Alleyne, Takao Suzuki, Srikanth Venkatraman
المصدر: ACS medicinal chemistry letters. 8(1)
مصطلحات موضوعية: 0301 basic medicine, Agonist, medicine.medical_specialty, medicine.drug_class, Insulin, medicine.medical_treatment, Organic Chemistry, Type 2 Diabetes Mellitus, GPR120, Type 2 diabetes, Biology, medicine.disease, Biochemistry, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Insulin resistance, Endocrinology, 030220 oncology & carcinogenesis, Diabetes mellitus, Internal medicine, Drug Discovery, medicine, Receptor
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9
المؤلفون: Mariappan V. Chelliah, Tze-Ming Chan, Yan Xia, George Boykow, Madhu Chintala, Matthew Bryant, Ho-Sam Ahn, Keith Eagen, Jacqueline Agans-Fantuzzi, William J. Greenlee, Yunsheng Hsieh, Samuel Chackalamannil
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:2544-2549
مصطلحات موضوعية: Blood Platelets, Platelet Aggregation, Metabolite, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Naphthalenes, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Alkaloids, Piperidines, In vivo, Drug Discovery, Thrombin receptor, medicine, Animals, Humans, Structure–activity relationship, Receptor, PAR-1, Furans, Molecular Biology, Vorapaxar, Drug discovery, Organic Chemistry, Thrombin, Rats, Macaca fascicularis, chemistry, Himbacine, Molecular Medicine, Platelet Aggregation Inhibitors, Ex vivo, Protein Binding, medicine.drug
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10
المؤلفون: Charles Lee Jayne, Francisco Velazquez, Zhuyan Guo, Donald M. Sperbeck, Murali Rajagopalan, Duane Burnette, Karen Marcantonio, Shouwu Miao, Sathesh Bhat, Santhosh Neelamkavil, Linda Brockunier, Stacia Kargman, Yan Xia, Rebecca T. Ruck, Vincent J. Colandrea, John A. Howe, Nicole Buist, Andrew Nolting, Yongxin Han, Pinto Patrick A, Thomas Bara, Mark Cartwright, Robert Chase, Martin C. Clasby, Srikanth Venkatraman, Randy R. Miller, Keith Eagen, Samuel Chackalamannil, Josien Hubert B, Chad Bennett, Mariappan V. Chelliah, Ian W. Davies, Austin Chen, Shah Unmesh G, Sony Agrawal, Dipshikha Biswas, Jin Wu, Aileen Soriano
المصدر: ACS medicinal chemistry letters. 7(1)
مصطلحات موضوعية: NS3, Protease, Molecular model, 010405 organic chemistry, Stereochemistry, medicine.medical_treatment, Organic Chemistry, Mutant, Biology, 01 natural sciences, Biochemistry, Protease inhibitor (biology), 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Drug Discovery, Genotype, medicine, Proline, Structural motif, medicine.drug