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1دورية أكاديمية
المؤلفون: Barbora Svobodova, Lenka Pulkrabkova, Dawid Panek, Anna Misiachna, Marharyta Kolcheva, Rudolf Andrys, Jiri Handl, Jan Capek, Pavlina Nyvltova, Tomas Rousar, Lukas Prchal, Vendula Hepnarova, Martina Hrabinova, Lubica Muckova, Daniela Tosnerova, Galina Karabanovich, Vladimir Finger, Ondrej Soukup, Martin Horak, Jan Korabecny
المصدر: International Journal of Molecular Sciences, Vol 24, Iss 11, p 9124 (2023)
مصطلحات موضوعية: Alzheimer’s disease, acetylcholinesterase, enzyme inhibition, N-methyl-d-aspartate receptor, monoamine oxidase A/B, multi-target directed ligands, Biology (General), QH301-705.5, Chemistry, QD1-999
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: David Malinak, Rafael Dolezal, Vendula Hepnarova, Miroslava Hozova, Rudolf Andrys, Petr Bzonek, Veronika Racakova, Jan Korabecny, Lukas Gorecki, Eva Mezeiova, Miroslav Psotka, Daniel Jun, Kamil Kuca, Kamil Musilek
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 478-488 (2020)
مصطلحات موضوعية: acetylcholinesterase, butyrylcholinesterase, organophosphate, reactivator, oxime, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: Barbora Svobodova, Eva Mezeiova, Vendula Hepnarova, Martina Hrabinova, Lubica Muckova, Tereza Kobrlova, Daniel Jun, Ondrej Soukup, María Luisa Jimeno, José Marco-Contelles, Jan Korabecny
المصدر: Biomolecules, Vol 9, Iss 8, p 379 (2019)
مصطلحات موضوعية: tacrine, bis(7)-tacrine, 6-chlorotacrine, 7-methoxytacrine, squaramides, Alzheimer’s disease, cholinesterases, in vitro, in silico, Microbiology, QR1-502
وصف الملف: electronic resource
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4دورية أكاديمية
المؤلفون: Jana Janockova, Rafael Dolezal, Eugenie Nepovimova, Tereza Kobrlova, Marketa Benkova, Kamil Kuca, Jan Konecny, Eva Mezeiova, Michaela Melikova, Vendula Hepnarova, Avi Ring, Ondrej Soukup, Jan Korabecny
المصدر: Molecules, Vol 23, Iss 11, p 2926 (2018)
مصطلحات موضوعية: orexin A, suvorexant, orexin receptor modulators, narcolepsy, structure-based virtual screening, Organic chemistry, QD241-441
وصف الملف: electronic resource
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5
المؤلفون: Vendula Hepnarova, Slavka Hamulakova, Jan Korabecny, Ondrej Soukup, Roman Mezencev, Ladislav Janovec, Martina Hrabinova, Veronika Ihnatova, Yury O. Chernoff, Zachery J. Deckner, Nikola Novakova, Zuzana Kudličková, Kamil Kuca, Petr Bzonek, Jana Janockova, Daniel Jun
المصدر: Future Med Chem
مصطلحات موضوعية: Indoles, Stereochemistry, Drug Evaluation, Preclinical, Molecular Dynamics Simulation, Ligands, Inhibitory Concentration 50, Structure-Activity Relationship, Alzheimer Disease, Drug Discovery, medicine, Humans, Molecular Targeted Therapy, 7-methoxytacrine, Biological evaluation, Pharmacology, Indole test, Amyloid beta-Peptides, Chemistry, DNA, In vitro, Molecular Docking Simulation, Neuroprotective Agents, Blood-Brain Barrier, Tacrine, Acetylcholinesterase, Molecular Medicine, Cholinesterase Inhibitors, Dimerization, Protein Binding, Research Article, medicine.drug
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6
المؤلفون: Vendula Hepnarova, Martina Hrabinova, Lubica Muckova, Tomas Kucera, Monika Schmidt, Rafael Dolezal, Lukas Gorecki, Veronika Hrabcova, Jan Korabecny, Eva Mezeiova, Daniel Jun, Jaroslav Pejchal
المصدر: Toxicology in Vitro. 85:105463
مصطلحات موضوعية: Insecticides, Mosquito Vectors, General Medicine, Toxicology, Organophosphates, Carbofuran, Butyrylcholinesterase, Anopheles, Acetylcholinesterase, Tacrine, Animals, Humans, Cholinesterase Inhibitors, Carbamates
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7
المؤلفون: Jaroslav Pejchal, Jiří Kassa, Filip Caisberger, Vendula Hepnarova, Jana Žďárová Karasová, Jana Hatlapatková
المصدر: Acta Medica, Vol 64, Iss 3, Pp 145-152 (2021)
مصطلحات موضوعية: Cholinesterase Reactivators, Pralidoxime, Antidotes, Pyridinium Compounds, Brain damage, Pharmacology, Neuroprotection, Poisons, chemistry.chemical_compound, Oximes, medicine, Animals, Chemical Warfare Agents, Rats, Wistar, Tabun, Pralidoxime Compounds, Neurotoxicity, General Medicine, medicine.disease, Oxime, Acetylcholinesterase, Organophosphates, Rats, Atropine, chemistry, Medicine, Cholinesterase Inhibitors, medicine.symptom, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::30ea4d69a081acbcc9bf865775ec9d0a
https://pubmed.ncbi.nlm.nih.gov/34779379 -
8
المؤلفون: Daniel Jun, Eva Mezeiova, Rudolf Andrys, Jan Korabecny, Lukas Gorecki, Kamil Musilek, David Malinak, Miroslava Hozova, Veronika Racakova, Petr Bzonek, Kamil Kuca, Miroslav Psotka, Vendula Hepnarova, Rafael Dolezal
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry
Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 478-488 (2020)مصطلحات موضوعية: Cholinesterase Reactivators, Stereochemistry, organophosphate, RM1-950, 01 natural sciences, oxime, chemistry.chemical_compound, Drug Discovery, Humans, Butyrylcholinesterase, Cholinesterase, Pharmacology, biology, 010405 organic chemistry, Organophosphate, General Medicine, Oxime, Isoquinolines, Acetylcholinesterase, In vitro, 0104 chemical sciences, reactivator, Molecular Docking Simulation, 010404 medicinal & biomolecular chemistry, chemistry, biology.protein, Therapeutics. Pharmacology, Cholinesterase Inhibitors, Research Paper
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9
المؤلفون: Ondrej Soukup, Martina Kaniakova, Tomas Kucera, Vendula Hepnarova, Martin Horak, Jan Korabecny, Karel Vales, Tereza Kobrlova, Eugenie Nepovimova, Kristina Holubova, Kristyna Skrenkova, Lenka Kleteckova, Zofia Chrienova
المصدر: Current Alzheimer Research. 16:821-833
مصطلحات موضوعية: Male, 0301 basic medicine, Cell Survival, Excitotoxicity, Glutamic Acid, Context (language use), CHO Cells, Pharmacology, Ligands, medicine.disease_cause, Receptors, N-Methyl-D-Aspartate, Neuroprotection, Capillary Permeability, Tissue Culture Techniques, 03 medical and health sciences, chemistry.chemical_compound, Cricetulus, 0302 clinical medicine, Alzheimer Disease, Memantine, medicine, Animals, Humans, Rats, Wistar, Cognitive decline, Glutamate receptor, Acetylcholinesterase, Molecular Docking Simulation, HEK293 Cells, Neuroprotective Agents, 030104 developmental biology, Neurology, chemistry, Blood-Brain Barrier, Tacrine, NMDA receptor, Cholinesterase Inhibitors, Neurology (clinical), 030217 neurology & neurosurgery, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::359004126134411738d964f70b5472cb
https://doi.org/10.2174/1567205016666190228122218 -
10
المؤلفون: Jana Zdarova Karasova, Jiri Kassa, Vendula Hepnarova, Jaroslav Pejchal, Lucie Junova, Rudolf Andrys, David Malinak, Petr Bzonek, Zuzana Kohoutova, Kamil Musilek
المصدر: Food and chemical toxicology : an international journal published for the British Industrial Biological Research Association. 167
مصطلحات موضوعية: Cholinesterase Reactivators, Mice, Antidotes, Oximes, Acetylcholinesterase, Animals, Pyridinium Compounds, General Medicine, Cholinesterase Inhibitors, Toxicology, Organophosphates, Food Science, Rats