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1
المؤلفون: Christian Tyrchan, Anna-Pia Palmgren, Hui-Fang Amy Chang, Yunhua Chen, Victoria Ullah, Karin Björhall, Annika Westin Eriksson, Rebecca Fransson, Mickael Mogemark, Tiiu Wennberg, Shuchun Zhao, Bold Peter, Linda Fredlund, Matthew Thomas, Eva Lamm Bergström, Nils Pemberton, Ulf Börjesson, Reed W. Smith, Mikael Brűlls, Johan Carlsson, Britt-Marie Fihn, Linda Öster, Mio Rodrigo Blomqvist, Hongbin Ge, Antonios Nikitidis, Wenzhen Yang, Anders Eriksson, Haijuan Huang, Sarah Lever, Perry Matthew, Kostas Karabelas, Helena Lindmark, Jens Petersen
المصدر: Journal of medicinal chemistry. 64(12)
مصطلحات موضوعية: Male, Class I Phosphatidylinositol 3-Kinases, Ovalbumin, High selectivity, Pharmacology, Crystallography, X-Ray, 01 natural sciences, 03 medical and health sciences, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, Rats, Inbred BN, Drug Discovery, medicine, Asthmatic patient, Potency, Structure–activity relationship, Animals, Class Ib Phosphatidylinositol 3-Kinase, Humans, Short duration, Protein Kinase Inhibitors, 030304 developmental biology, Asthma, 0303 health sciences, Sulfonamides, biology, Inhalation, Molecular Structure, Chemistry, medicine.disease, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Thiazoles, biology.protein, Leukocytes, Mononuclear, Molecular Medicine, Protein Binding
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2
المؤلفون: Eva Lamm Bergström, Fredrik Wågberg, Christian Tyrchan, Anders Lundqvist, Ulf Andersson, Xiao-Hong Zhou, Robert Ronn, Linda Swedin, Grigorios Nikitidis, Fanyi Jiang, Victoria Ullah, Antonios Nikitidis, Petra Johannesson, Eva Björkstrand, Hui-Fang Chang, Theresa Andreasson, Lena Ripa, Magnus Munck af Rosenschöld, Pernilla Glader, Anna Pettersen, Britta Bonn, Margareta Ek, Andrew M. Davis, Euan Gordon, Helena Käck, Dave Chapman, Mattias Rohman, Anna Malmberg
المصدر: Journal of Medicinal Chemistry. 62:7769-7787
مصطلحات موضوعية: chemistry.chemical_classification, 0303 health sciences, Ligand efficiency, Leukotriene C4, Pharmacology, 01 natural sciences, Peripheral blood mononuclear cell, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Enzyme, chemistry, In vivo, Pharmacodynamics, Drug Discovery, Molecular Medicine, Potency, IC50, 030304 developmental biology
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المؤلفون: Ulla Karlsson, Anders Gunnarsson, Stefan Tångefjord, Christian Köhler, Karl Edman, Göran Carlström, Ulrich Weininger, Tineke Papavoine, Victoria Ullah, Mikael Akke, Matti Lepistö
المصدر: Science Advances
مصطلحات موضوعية: 0303 health sciences, Multidisciplinary, Ligand, Chemistry, Allosteric regulation, SciAdv r-articles, Nuclear magnetic resonance spectroscopy, 010402 general chemistry, Biochemistry, 01 natural sciences, 0104 chemical sciences, 03 medical and health sciences, Glucocorticoid receptor, Structural Biology, Helix, Biophysics, Transcriptional regulation, Surface plasmon resonance, Pharmacophore, hormones, hormone substitutes, and hormone antagonists, Research Articles, Research Article, 030304 developmental biology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::79b642aa4382500c6724c685c4beac53
https://doi.org/10.1126/sciadv.abb5277 -
4
المؤلفون: Magnus, Munck Af Rosenschöld, Petra, Johannesson, Antonios, Nikitidis, Christian, Tyrchan, Hui-Fang, Chang, Robert, Rönn, Dave, Chapman, Victoria, Ullah, Grigorios, Nikitidis, Pernilla, Glader, Helena, Käck, Britta, Bonn, Fredrik, Wågberg, Eva, Björkstrand, Ulf, Andersson, Linda, Swedin, Mattias, Rohman, Theresa, Andreasson, Eva Lamm, Bergström, Fanyi, Jiang, Xiao-Hong, Zhou, Anders J, Lundqvist, Anna, Malmberg, Margareta, Ek, Euan, Gordon, Anna, Pettersen, Lena, Ripa, Andrew M, Davis
المصدر: Journal of medicinal chemistry. 62(17)
مصطلحات موضوعية: Dose-Response Relationship, Drug, Molecular Structure, Administration, Oral, Asthma, Rats, Disease Models, Animal, Structure-Activity Relationship, Pyrazines, Drug Discovery, Animals, Humans, Anti-Asthmatic Agents, Enzyme Inhibitors, Glutathione Transferase
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5
المؤلفون: Dave Chapman, Victoria Ullah, Lisa Wissler, James Bird, Jesper Malmberg, Petter Svanberg, Christian Köhler, Antonios Nikitidis, Matti Lepistö, Stefan Geschwindner, Karl Edman, Tomas Drmota, Lena Ripa, Richard P. Harrison, Hui-Fang Chang, Goran Edenro, Tove Hegelund-Myrbäck, Ramon Hendrickx, Roine I. Olsson, Matthew Dearman, Philip Thorne, Antoni Llinas, Karolina Lawitz, Markus Berger
المصدر: Journal of medicinal chemistry. 61(5)
مصطلحات موضوعية: 0301 basic medicine, Agonist, Indazoles, Side effect, medicine.drug_class, Pyridines, Anti-Inflammatory Agents, Administration, Oral, Pharmacology, Ligands, Partial agonist, Cell Line, 03 medical and health sciences, 0302 clinical medicine, Glucocorticoid receptor, Receptors, Glucocorticoid, In vivo, Drug Discovery, medicine, Glucose homeostasis, Animals, Humans, Receptor, Chemistry, Rats, 030104 developmental biology, 030220 oncology & carcinogenesis, Prednisolone, Molecular Medicine, medicine.drug
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6
المؤلفون: Antonio Llinas, Fredrik Thorstensson, Emma Lindhardt, Ågot Högberg, Kristina Nilsson, Anders Lindqvist, Annika Åstrand, Göran Duker, Victoria Ullah, Gavin O'Mahony, Qing-Dong Wang, Pernilla Ståhlberg, Nidhal Selmi, Laurent Knerr, Fabrizio Giordanetto
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:5557-5561
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Calcium Channels, T-Type, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Acetamides, Drug Discovery, Animals, Humans, Molecular Biology, Antihypertensive Agents, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Calcium channel, Organic Chemistry, T-type calcium channel, Stereoisomerism, Calcium Channel Inhibition, Ether-A-Go-Go Potassium Channels, High-Throughput Screening Assays, Rats, Chemical evolution, Molecular Medicine, Acetamide
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7
المؤلفون: Antonio Llinas, Göran Duker, Annika Åstrand, Victoria Ullah, Qing-Dong Wang, Fabrizio Giordanetto, Grigorios Nikitidis, Fredrik Thorstensson, Emma Lindhardt, Anders Lindqvist, Staffan Karlsson, Nidhal Selmi, Got Högberg, Andreas Wållberg, Laurent Knerr, Åsa Lindelöf
المصدر: Bioorganicmedicinal chemistry letters. 23(1)
مصطلحات موضوعية: Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Pharmacology, Biochemistry, chemistry.chemical_compound, Calcium Channels, T-Type, Structure-Activity Relationship, Dogs, Heart Rate, Drug Discovery, medicine, Animals, Humans, Hydroxymethyl, Benzamide, Molecular Biology, Ion channel, Mibefradil, Voltage-dependent calcium channel, Calcium channel, Organic Chemistry, T-type calcium channel, Calcium Channel Inhibition, Calcium Channel Blockers, chemistry, Benzamides, Molecular Medicine, medicine.drug, Half-Life
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المؤلفون: Nidhal Selmi, Anders Broo, Emma J. Williams, William McCoull, Peter Barton, Nathaniel G. Martin, Gareth Coope, Krister Österlund, Jane E. Moore, David S. Clarke, Alastair J. H. Brown, Stephen Stokes, Eleanor Rosevere, Tor Svensson, Robert D. M. Davies, Alexander G. Dossetter, Graeme R. Robb, Elizabeth E. Kelly, Jane L. Holmes, Claire Newton, Victoria Ullah, David G.A. Morgan, Philip A. MacFaul, Laurent Knerr
المصدر: MedChemComm. 4:456
مصطلحات موضوعية: Pharmacology, Food intake, biology, Chemistry, Organic Chemistry, hERG, Pharmaceutical Science, Biochemistry, Partial agonist, chemistry.chemical_compound, Pyrimidinones, Drug Discovery, Lipophilicity, biology.protein, Molecular Medicine, Inverse agonist, Piperidine, Quinazolinone, hormones, hormone substitutes, and hormone antagonists
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::0e338246543e6606730bbb19b24004e0
https://doi.org/10.1039/c2md20340e