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المؤلفون: Richard A. Hartz, Vijay T. Ahuja, Prasanna Sivaprakasam, Hong Xiao, Carol M. Krause, Wendy J. Clarke, Kevin Kish, Hal Lewis, Nicolas Szapiel, Ramu Ravirala, Sayali Mutalik, Deepa Nakmode, Devang Shah, Catherine R. Burton, John E. Macor, Gene M. Dubowchik
المصدر: Journal of Medicinal Chemistry. 66:4231-4252
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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2
المؤلفون: Richard A. Hartz, Vijay T. Ahuja, Guanglin Luo, Ling Chen, Prasanna Sivaprakasam, Hong Xiao, Carol M. Krause, Wendy J. Clarke, Songmei Xu, John S. Tokarski, Kevin Kish, Hal Lewis, Nicolas Szapiel, Ramu Ravirala, Sayali Mutalik, Deepa Nakmode, Devang Shah, Catherine R. Burton, John E. Macor, Gene M. Dubowchik
المصدر: Journal of Medicinal Chemistry.
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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3
المؤلفون: Richard A. Hartz, Vijay T. Ahuja, Susheel J. Nara, C. M. Vijaya Kumar, Raju K. V. L. P. Manepalli, Sarat Kumar Sarvasiddhi, Swarnamba Honkhambe, Vidya Patankar, Bireshwar Dasgupta, Ramkumar Rajamani, Jodi K. Muckelbauer, Daniel M. Camac, Kaushik Ghosh, Matthew Pokross, Susan E. Kiefer, Jeffrey M. Brown, Lisa Hunihan, Michael Gulianello, Martin Lewis, Jonathan S. Lippy, Neha Surti, Brian D. Hamman, Jason Allen, Walter A. Kostich, Joanne J. Bronson, John E. Macor, Carolyn D. Dzierba
المصدر: Journal of Medicinal Chemistry. 65:4121-4155
مصطلحات موضوعية: Structure-Activity Relationship, Drug Discovery, Quinazolines, Quinolines, Animals, Neuralgia, Molecular Medicine, Amides, Protein Kinase Inhibitors
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4
المؤلفون: Ching Kim Tye, Chunhong Yan, Sarah C. Traeger, Wayne Vaccaro, Yingru Zhang, Gerry Everlof, Jianqing Li, Henry Yip, Peng Li, John T. Hunt, Michael A. Poss, Gregory D. Vite, Mussari Christopher P, Steven Sheriff, Asoka Ranasinghe, Haiying Zhang, Richard A. Westhouse, Dharmpal S. Dodd, Richard Rampulla, Zheng Yang, Frank Marsilio, Derek J. Norris, Wen-Ching Han, Tram N. Huynh, Yufen Zhao, Patrice Gill, Nirmala Raghavan, Lalgudi S. Harikrishnan, Ashvinikumar V. Gavai, Susan Wee, John S. Tokarski, Dauh-Rurng Wu, Arvind Mathur, Mei-Li Wen, Huiping Zhang, David R. Tortolani, George V. Delucca, Krista Menard, Francis Y. Lee, Claude A. Quesnelle, Dawn Sun, Vijay T. Ahuja, Daniel O'malley, Christine Huang, Muthoni G. Kamau
المصدر: Journal of Medicinal Chemistry. 64:14247-14265
مصطلحات موضوعية: Drug, Proline, Phenylalanine, media_common.quotation_subject, Carbazoles, Administration, Oral, Antineoplastic Agents, Cell Cycle Proteins, Computational biology, BET inhibitor, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Transcriptional regulation, Humans, Potency, media_common, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Tryptophan, Signal transducing adaptor protein, Bromodomain, Molecular Medicine, Transcription Factors
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المؤلفون: Ashvinikumar V. Gavai, Brian E. Fink, Dianlin Xie, Susan Wee, David A Critton, Jesse Swanson, Carolyn Cao, John S. Tokarski, Vijay T. Ahuja, Daniel O'malley, Nicolas Szapiel, Benjamin M. Johnson, Cindy Wang, Anthony A. Paiva
المصدر: ACS Medicinal Chemistry Letters. 10:1486-1491
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, T cell, Organic Chemistry, Inhibitory postsynaptic potential, 01 natural sciences, Biochemistry, 0104 chemical sciences, Negative regulator, Cell biology, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, medicine.anatomical_structure, C-terminal Src kinase, Drug Discovery, Pyridine, medicine, Phosphorylation, Proto-oncogene tyrosine-protein kinase Src
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6
المؤلفون: Jodi K. Muckelbauer, Ramkumar Rajamani, Jeffrey M. Brown, C M Vijaya Kumar, Kumaran Dandapani, Jonathan Lippy, Saravanan Elavazhagan, Vijay T. Ahuja, John E. Macor, Carolyn Diane Dzierba, Brian D. Hamman, Walter Kostich, Michael Gulianello, Manoj Dokania, Susan E. Kiefer, Susheel J. Nara, Joanne J. Bronson, Amy Easton, Richard A. Hartz, Linda J. Bristow, Martin A. Lewis, Jason Allen, Sreenivasulu N Pattipati, Neha Surti, Lisa Hunihan, Daniel M. Camac
المصدر: Journal of medicinal chemistry. 64(15)
مصطلحات موضوعية: Male, Phenotypic screening, Pharmacology, Protein Serine-Threonine Kinases, chemistry.chemical_compound, Mice, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Humans, Dose-Response Relationship, Drug, Molecular Structure, Kinase, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Chronic pain, AAK1, Signal transducing adaptor protein, Brain, medicine.disease, Amides, Mice, Inbred C57BL, HEK293 Cells, Neuropathic pain, Microsomes, Liver, Molecular Medicine, Neuralgia, Caco-2 Cells, Penetrant (biochemical), Protein Kinases
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7
المؤلفون: Joanne J. Bronson, Nicholas J. Lodge, John E. Macor, James E. Grace, Richard A. Hartz, Vivekananda M. Vrudhula, Vijay T. Ahuja
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:1360-1363
مصطلحات موضوعية: 010405 organic chemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Crf1 receptor, Antagonist, Pharmaceutical Science, Prodrug, Pharmacology, 030226 pharmacology & pharmacy, 01 natural sciences, Biochemistry, 0104 chemical sciences, Bioavailability, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, Drug Discovery, Aqueous solubility, Alkoxy group, Molecular Medicine, Molecular Biology, Linker
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المؤلفون: Kimberley A. Lentz, Gail K. Mattson, James E. Grace, Nicholas J. Lodge, John E. Macor, Richard A. Hartz, Thaddeus F. Molski, Vijay T. Ahuja, Joanne J. Bronson
المصدر: Bioorganic & Medicinal Chemistry Letters. 26:2184-2187
مصطلحات موضوعية: Carbamate, Stereochemistry, Chemistry, Aryl, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Ether, 030226 pharmacology & pharmacy, Biochemistry, In vitro, Corticotropin-releasing hormone receptor 1, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Drug Discovery, medicine, Molecular Medicine, Structure–activity relationship, Receptor, Molecular Biology, IC50, 030217 neurology & neurosurgery
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9
المؤلفون: Zhi Liang, Alan Wilson, Li Dong, Neil T. Burford, David S. Kimball, Kenneth G. Carson, Yingzhi Bi, Yulian Zhang, Bireshwar Dasgupta, Carolyn Diane Dzierba, Richard A. Hartz, James E. Grace, G. Greg Zipp, Soojin Kwon, Martin A. Lewis, Joanne J. Bronson, Cynthia Anne Fink, Amr Nouraldeen, Saadat Aleem, Giovanni Cianchetta, Jiancheng Wang, Ying Liu, Vijay T. Ahuja, Robert L. Bertekap, Jianxin Han, Michael Alan Green, Angela Cacace, Godwin Kumi, Yudith Garcia, Ying Qiao, Meredith Ferrante, John E. Macor, Ryan Westphal
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:1448-1452
مصطلحات موضوعية: Agonist, Dose-Response Relationship, Drug, Molecular Structure, medicine.drug_class, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Small molecule, Receptors, G-Protein-Coupled, Structure-Activity Relationship, HEK293 Cells, Pharmacokinetics, Design synthesis, Ethanolamines, Drug Design, Drug Discovery, medicine, Humans, Molecular Medicine, Amines, Molecular Biology
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10
المؤلفون: Richard A, Hartz, Vivekananda M, Vrudhula, Vijay T, Ahuja, James E, Grace, Nicholas J, Lodge, Joanne J, Bronson, John E, Macor
المصدر: Bioorganicmedicinal chemistry letters. 27(6)
مصطلحات موضوعية: Pyrazines, Animals, Biological Availability, Prodrugs, Receptors, Corticotropin-Releasing Hormone, Rats