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1
المؤلفون: Geoffrey D. Clarke, Silvano Ronzoni, Carlo Farina, Paola Petrillo, Marco Artico, Drake S. Eggleston, Giulio Dondio, Giuseppe Petrone, Luciano Visentin, Vittorio Vecchietti
المصدر: Journal of Medicinal Chemistry. 40:3192-3198
مصطلحات موضوعية: Male, Models, Molecular, Agonist, Indoles, medicine.drug_class, Stereochemistry, Narcotic Antagonists, Carboxamide, Ligands, Chemical synthesis, Piperazines, Mice, Vas Deferens, Naltrindole, Receptors, Opioid, delta, Drug Discovery, medicine, Animals, Moiety, Computer Simulation, Pyrroles, Binding selectivity, Dose-Response Relationship, Drug, Chemistry, Brain, Nociceptors, Stereoisomerism, Enkephalin, Leucine-2-Alanine, Isoquinolines, Naltrexone, Drug Design, Benzamides, Quinolines, Molecular Medicine, SNC-80, Enantiomer, Signal Transduction, medicine.drug
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2
المؤلفون: Douglas W. P. Hay, Vittorio Vecchietti, Carlo Farina, Mark A. Luttmann, Henry M. Sarau, Roberto Rigolio, Andrew D. Medhurst, Luca F. Raveglia, Dulcie B. Schmidt, Giuseppe Giardina, Mario Grugni
المصدر: Journal of Medicinal Chemistry. 40:1794-1807
مصطلحات موضوعية: animal structures, Chemical Phenomena, Stereochemistry, CHO Cells, Substance P, Binding, Competitive, Chemical synthesis, Structure-Activity Relationship, Cricetinae, Drug Discovery, Animals, Humans, Receptor, Molecular Structure, Bicyclic molecule, Chemistry, Physical, Chemistry, Chinese hamster ovary cell, Antagonist, Hydrogen Bonding, Receptors, Neurokinin-3, Stereoisomerism, Peptide Fragments, Recombinant Proteins, In vitro, Biochemistry, embryonic structures, Quinolines, Molecular Medicine, Rabbits, Selectivity, Neurokinin 3 receptor, Muscle Contraction
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3
المؤلفون: Dulcie B. Schmidt, Andrew D. Medhurst, Marco Vassallo, Mario Grugni, Douglas W. P. Hay, Giuseppe Giardina, Carlo Farina, Henry M. Sarau, Vittorio Vecchietti, Roberto Rigolio, James J. Foley, Luca F. Raveglia
المصدر: Journal of Medicinal Chemistry. 39:2281-2284
مصطلحات موضوعية: Agonist, medicine.drug_class, Recombinant Fusion Proteins, Guinea Pigs, CHO Cells, Substance P, Binding, Competitive, Structure-Activity Relationship, chemistry.chemical_compound, Cricetulus, Piperidines, Cricetinae, Drug Discovery, medicine, Animals, Humans, Selective receptor modulator, Receptor, Ciliary Body, Receptors, Neurokinin-3, Receptor antagonist, Peptide Fragments, HYDIA, chemistry, Biochemistry, Drug Design, Quinolines, Molecular Medicine, Rabbits, Neurokinin A, Neurokinin B, Tachykinin receptor, Muscle Contraction
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4
المؤلفون: Giulio Dondio, Luciano Visentin, Giardina Giuseppe Arnaldo Mari, Silvano Ronzoni, Geoffrey D. Clarke, Paola Petrillo, Giuseppe Petrone, Vittorio Vecchietti
المصدر: Analgesia. 1:394-399
مصطلحات موضوعية: Stereochemistry, Chemistry, Delta opioid agonist, Geriatrics and Gerontology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::570ea79192d4a4adb5d5f7d9c6679ccd
https://doi.org/10.3727/107156995819563573 -
5
المؤلفون: Giuseppe Giardina, Geoffrey D. Clarke, Vittorio Vecchietti, Giulio Dondio, Giuseppe Petrone, M. Sbacchi
المصدر: Journal of Medicinal Chemistry. 37:3482-3491
مصطلحات موضوعية: Male, Pyrrolidines, Tetrahydronaphthalenes, Tertiary amine, Stereochemistry, Motor Activity, Pharmacology, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, medicine, Animals, Potency, Computer Simulation, ED50, Tetralones, Analgesics, Molecular Structure, Chemistry, Receptors, Opioid, kappa, Spiradoline, Biological activity, Diuresis, Rats, Opioid, Molecular Medicine, Piperidine, Analgesia, medicine.drug
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6
المؤلفون: R. Colle, Vittorio Vecchietti, G. D. Clarke, M. Sbacchi, Giuseppe Petrone, Giardina Giuseppe Arnaldo Mari
المصدر: ChemInform. 23
مصطلحات موضوعية: chemistry.chemical_compound, Class (set theory), chemistry, Tetrahydroisoquinoline, Stereochemistry, General Medicine, Opioid analgesics
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7
المؤلفون: G. D. Clarke, Giuseppe Petrone, R. Colle, Vittorio Vecchietti, Giulio Dondio, M. Sbacchi, Giardina Giuseppe Arnaldo Mari
المصدر: ChemInform. 23
مصطلحات موضوعية: Opioid, Stereochemistry, Chemistry, Antinociceptive Agents, medicine, General Medicine, Receptor, Selectivity, medicine.drug
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8
المؤلفون: Geoffrey D. Clarke, Giulio Dondio, Giuseppe Petrone, Vittorio Vecchietti, M. Sbacchi, Roberto Colle, Giuseppe Giardina
المصدر: Chirality. 4:8-15
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Receptors, Opioid, mu, Tartrate, Catalysis, Analytical Chemistry, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Antinociceptive Agents, Animals, Potency, Spectroscopy, Pipecolic acid, Pharmacology, Analgesics, Receptors, Opioid, kappa, Organic Chemistry, Diastereomer, Stereoisomerism, Kinetics, chemistry, Receptors, Opioid, μ-opioid receptor, Enantiomer
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9
المؤلفون: Roberto Colle, Geoffrey D. Clarke, Antonio Giordani, Vittorio Vecchietti, Giuseppe Giardina
المصدر: Journal of Medicinal Chemistry. 34:397-403
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Stereochemistry, medicine.drug_class, Hydrochloride, Guinea Pigs, Molecular Conformation, Substituent, Carboxamide, Structure-Activity Relationship, chemistry.chemical_compound, Piperidines, Drug Discovery, medicine, Animals, Moiety, Analgesics, Trifluoromethyl, Molecular Structure, Receptors, Opioid, kappa, Brain, Kinetics, chemistry, Receptors, Opioid, Molecular Medicine, Indicators and Reagents, Piperidine, Pharmacophore, Kappa
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10
المؤلفون: James J. Foley, Giuseppe Giardina, Carlo Farina, Douglas W. P. Hay, Henry M. Sarau, Luca F. Raveglia, Mark A. Luttmann, Andrew D. Medhurst, Roberto Rigolio, Mario Grugni, Vittorio Vecchietti, Stefano Cavagnera, Dulcie B. Schmidt, Davide Graziani
المصدر: Journal of medicinal chemistry. 42(6)
مصطلحات موضوعية: animal structures, medicine.drug_class, Stereochemistry, Iris, Carboxamide, CHO Cells, In Vitro Techniques, Motor Activity, Substance P, Cell Line, Mice, Radioligand Assay, Structure-Activity Relationship, In vivo, Cricetinae, Drug Discovery, Talnetant, medicine, Structure–activity relationship, Animals, Humans, Cloning, Molecular, Receptor, Chemistry, Antagonist, Muscle, Smooth, Receptors, Neurokinin-3, Miosis, Receptor antagonist, Peptide Fragments, embryonic structures, Quinolines, Molecular Medicine, Calcium, Rabbits, medicine.drug, Muscle Contraction