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1دورية أكاديمية
المؤلفون: Sharon McGonigle, Utpal Majumder, Donna Kolber-Simonds, Jiayi Wu, Andrew Hart, Thomas Noland, Karen TenDyke, Daniel Custar, Danyang Li, Hong Du, Maarten H. D. Postema, W. George Lai, Natalie C. Twine, Mary Woodall-Jappe, Kenichi Nomoto
المصدر: Cell Communication and Signaling, Vol 17, Iss 1, Pp 1-14 (2019)
مصطلحات موضوعية: Chlorotoxin, Neuropilin-1, Tumor, Uptake, Peptide-drug-conjugate, Medicine, Cytology, QH573-671
وصف الملف: electronic resource
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المؤلفون: Anshul Gupta, Jennifer L. Liras, Stephen Fowler, W. George Lai, Jane R. Kenny, Jonathan A. Phillips, Jinping Gan, Niresh Hariparsad, David B. Duignan, Wen Li Kelly Chen
المصدر: Lab on a chip. 20(3)
مصطلحات موضوعية: Drug Industry, Computer science, Biomedical Engineering, Drug Evaluation, Preclinical, Bioengineering, Context (language use), 030226 pharmacology & pharmacy, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Drug Development, Lab-On-A-Chip Devices, Animals, Humans, 030304 developmental biology, Pharmaceutical industry, ADME, 0303 health sciences, System development, business.industry, Drug discovery, General Chemistry, Human physiology, Microfluidic Analytical Techniques, Drug development, Risk analysis (engineering), Pharmaceutical Preparations, Proof of concept, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d7999b04fd17f88b03091a6f0d36dc64
https://pubmed.ncbi.nlm.nih.gov/31932816 -
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المؤلفون: Sherri Smith, Darrell Nix, Nathalie Rioux, Pete Smith, Joanne Schindler, Amy Kim, Federico Colombo, Y Amy Siu, W. George Lai
مصطلحات موضوعية: Pyridines, Health, Toxicology and Mutagenesis, Biological Availability, Antineoplastic Agents, Tumor cells, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Piperazines, Rats, Sprague-Dawley, Feces, 03 medical and health sciences, 0302 clinical medicine, Animals, Bile, Humans, Rats, Long-Evans, Tissue Distribution, Pharmacology, Chemistry, Haplorhini, General Medicine, Disposition, Small molecule, Rats, Cell biology, 030220 oncology & carcinogenesis, RNA splicing
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::086ad5cf1dd1b6387552a1d946c35242
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4
المؤلفون: W. George Lai, Min-Kun Chang, Cynthia A. Zamora, Maiko Nomoto, Y. Amy Siu, Peter Boyd, Edgar Schuck, Jagadeesh Aluri, Bhaskar Rege, Sanae Yasuda, Jim Ferry
المصدر: British Journal of Clinical Pharmacology. 84:952-960
مصطلحات موضوعية: Pharmacology, Drug, Agonist, business.industry, medicine.drug_class, CYP3A, Itraconazole, media_common.quotation_subject, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, 030220 oncology & carcinogenesis, Pharmacodynamics, Medicine, Pharmacology (medical), business, CYP2C9, Fluconazole, medicine.drug, media_common
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5
المؤلفون: Markus Warmuth, Manav Korpal, Deepti Banka, Peter Fekkes, Pavan Kumar, Andrew Hart, Lihua Yu, Ping Zhu, Lorna Helen Mitchell, Joyce Yang, W. George Lai, Amy Kim, Craig Karr, Pete Smith, Tarek Sahmoud, Xiaoling Puyang, Sherri Smith, Mike Thomas, Benjamin Caleb, O'shea Morgan Welzel, Victoria Rimkunas, Huilan Yao, Sean Eckley, Allison Davis, Silvia Buonamici, Crystal MacKenzie, V. Subramanian, Jeremy Wu, Zheng Guo Zhu, Christopher Rowbottom, Reynolds Dominic, Nicholas A. Larsen, Nathalie Rioux, Sean Irwin, Craig Furman
المصدر: Cancer Research. 77:DDT01-04
مصطلحات موضوعية: Cancer Research, Fulvestrant, business.industry, 010401 analytical chemistry, Cancer, Estrogen receptor, Pharmacology, medicine.disease, 01 natural sciences, 0104 chemical sciences, 03 medical and health sciences, 0302 clinical medicine, Breast cancer, Oncology, Nuclear receptor, Selective estrogen receptor modulator, 030220 oncology & carcinogenesis, Medicine, business, Estrogen receptor beta, Tamoxifen, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::71b5b0fa7e9d8e6795b2dcf66171548d
https://doi.org/10.1158/1538-7445.am2017-ddt01-04 -
6
المؤلفون: Kazutomi Kusano, Edgar Schuck, Michiko Sugawara, W. George Lai, Krista Condon, Christopher DesJardins, Earvin Liang
المصدر: Cancer Chemotherapy and Pharmacology
مصطلحات موضوعية: Male, 0301 basic medicine, Cancer Research, Pharmacology, Toxicology, Rats, Sprague-Dawley, Mice, chemistry.chemical_compound, 0302 clinical medicine, Tandem Mass Spectrometry, Tissue Distribution, Pharmacology (medical), Melanoma, Tumor xenograft, High concentration, Mice, Inbred BALB C, Tumor, Brain, Ketones, Oncology, 030220 oncology & carcinogenesis, Female, Original Article, medicine.symptom, Perfusion, Half-Life, Eribulin, Halichondrin B, Antineoplastic Agents, Vascular Remodeling, 03 medical and health sciences, Dogs, Species Specificity, Pharmacokinetics, medicine, Animals, Humans, Distribution (pharmacology), Furans, Dose-Response Relationship, Drug, Xenograft, Xenograft Model Antitumor Assays, Rats, 030104 developmental biology, Mechanism of action, chemistry, Chromatography, Liquid
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7
المؤلفون: Y. Amy Siu, W. George Lai
المصدر: Drug Metabolism and Disposition. 45:183-189
مصطلحات موضوعية: Metabolic Clearance Rate, Pharmaceutical Science, In Vitro Techniques, Models, Biological, 030226 pharmacology & pharmacy, Substrate Specificity, 03 medical and health sciences, 0302 clinical medicine, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, CYP2C9, Cytochrome P-450 CYP2C9, Pharmacology, Cross-Over Studies, CYP3A4, biology, Chemistry, Cytochrome P450, Substrate (chemistry), Metabolism, Meloxicam, Losartan, Pharmaceutical Preparations, Biochemistry, 030220 oncology & carcinogenesis, Microsomes, Liver, biology.protein, Microsome, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2be46ff02067829ce430655c877d84ec
https://doi.org/10.1124/dmd.116.073510 -
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المؤلفون: Kristian Jensen, Wayne Tang, Mary Grimes, David Calkins, W. George Lai, Sayan Mondal, Victoria A. Feher, Jeff Bell, Wu Yin, Fiona M. McRobb, Shulu Feng, Michael Trzoss, Goran Krilov, Hamish Wright, Andrew Placzek, Robert Pelletier, Morgan Lawrenz, Nie Zhe, Aleksey Gerasyuto, Karen Akinsanya
المصدر: Blood. 136:30-30
مصطلحات موضوعية: biology, Venetoclax, Chronic lymphocytic leukemia, Immunology, Cell Biology, Hematology, medicine.disease, Biochemistry, Jurkat cells, BCL10, chemistry.chemical_compound, medicine.anatomical_structure, chemistry, Ibrutinib, medicine, biology.protein, Cancer research, Bruton's tyrosine kinase, Diffuse large B-cell lymphoma, B cell
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::eb01c8f81a6d5bd57cabeffa46499596
https://doi.org/10.1182/blood-2020-141146 -
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المؤلفون: James J. Vornov, Ying Wu, Kenichi Nomoto, Larisa Reyderman, Nancy Wong, Christopher DesJardins, Yanke Yu, Bruce A. Littlefield, Krystyna M. Wozniak, W. George Lai, Barbara S. Slusher
المصدر: Cancer Research. 76:3332-3339
مصطلحات موضوعية: 0301 basic medicine, Eribulin Mesylate, Cancer Research, Time Factors, Paclitaxel, Blotting, Western, Apoptosis, Pharmacology, Microtubules, Article, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Ganglia, Spinal, medicine, Animals, Tissue Distribution, Furans, Cell Proliferation, Mice, Inbred BALB C, Dose-Response Relationship, Drug, business.industry, Neurotoxicity, Peripheral Nervous System Diseases, Ketones, medicine.disease, Sciatic Nerve, Tubulin Modulators, Electrophysiology, 030104 developmental biology, medicine.anatomical_structure, Peripheral neuropathy, Oncology, chemistry, Epothilones, Peripheral nervous system, Female, Sciatic nerve, business, 030217 neurology & neurosurgery, Eribulin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2354bf4cbf0c4beb2e17561324defff3
https://doi.org/10.1158/0008-5472.can-15-2525 -
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المؤلفون: Heidi J. Einolf, Susanna Tse, Tonika Bohnert, Sirimas Sudsakorn, Ying-Hong Wang, David Moore, Jim Keirns, Ling He, Robert L. Walsky, Rangaraj Narayanan, Wanping Geng, Aarti Patel, Louis Leung, W. George Lai, Xiaoqing Yang, Ralph Stearns, Dieter Lang, Michael Sinz, Yuan Chen, Chuang Lu, Jan Wahlstrom, Ian Templeton
المصدر: Drug Metabolism and Disposition. 44:1399-1423
مصطلحات موضوعية: Drug, Drug Industry, Computer science, media_common.quotation_subject, Population, Decision tree, Pharmaceutical Science, Pharmacology, Risk Assessment, 030226 pharmacology & pharmacy, Substrate Specificity, 03 medical and health sciences, 0302 clinical medicine, Species Specificity, New chemical entity, Drug Discovery, Animals, Humans, Computer Simulation, Drug Interactions, education, Biotransformation, media_common, education.field_of_study, Decision Trees, Perspective (graphical), Models, Theoretical, Enzymes, Kinetics, Identification (information), Drug metabolizing enzymes, Pharmaceutical Preparations, Risk analysis (engineering), 030220 oncology & carcinogenesis, Risk assessment
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::57ff752216b7095cfbd939b67f0dd8ae
https://doi.org/10.1124/dmd.115.069096