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1
المؤلفون: Helen T. Lee, Brian R. Krause, Bruce D. Roth, R. L. Stanfield, W. H. Roark, Joseph Armand Picard, Drago Robert Sliskovic, R. F. Bousley, K. L. Hamelehle
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:289-294
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Sterol O-acyltransferase, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Organophosphorus Compounds, Microsomes, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, Sulfonamides, biology, Cholesterol, Anticholesteremic Agents, Organic Chemistry, Phosphoramidate, Enzyme, chemistry, Acyltransferases, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Sterol O-Acyltransferase
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2
المؤلفون: Drago Sliskovic, Essenburg Ad, Joseph Armand Picard, J. F. Reindel, L. L. Minton, B.R. Krause, R. L. Stanfield, W. H. Roark
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:713-718
مصطلحات موضوعية: chemistry.chemical_classification, Cholesterol, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biological activity, Pharmacology, Biochemistry, Acyl transferase, chemistry.chemical_compound, Acyl-CoA, Enzyme, chemistry, Amide, Drug Discovery, Molecular Medicine, Bioassay, Molecular Biology, Ex vivo
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3
المؤلفون: T. L. Stoeber, R. L. Stanfield, W. H. Roark, Brian R. Krause, C. J. Blankley, Bharat K. Trivedi, J. A. Picard, Ann Holmes, Essenburg Ad, M. K. Shaw
المصدر: Journal of Medicinal Chemistry. 36:3300-3307
مصطلحات موضوعية: chemistry.chemical_classification, biology, Cholesterol, Anticholesteremic Agents, Sterol O-acyltransferase, In vitro, Structure-Activity Relationship, chemistry.chemical_compound, Enzyme, Biochemistry, chemistry, In vivo, Enzyme inhibitor, Drug Discovery, biology.protein, Urea, Molecular Medicine, Structure–activity relationship, Moiety, Carbanilides, Sterol O-Acyltransferase
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4
المؤلفون: E. Ferguson, Roger S. Newton, J. A. Picard, C. S. Sekerke, D. R. Sliskovic, Bruce D. Roth, M. K. Shaw, W. H. Roark, Brian R. Krause
المصدر: ChemInform. 22
مصطلحات موضوعية: chemistry.chemical_compound, biology, Chemistry, Pyran, Stereochemistry, HMG-CoA reductase, biology.protein, General Medicine, Cholesterol biosynthesis
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5
المؤلفون: A. D. Essenburg, Brian R. Krause, Bharat K. Trivedi, R. L. Stanfield, M. K. Shaw, T. L. Stoeber, W. H. Roark, Joseph Armand Picard, C. J. Blankley, Ann Holmes
المصدر: ChemInform. 25
مصطلحات موضوعية: chemistry.chemical_compound, Biochemistry, Chemistry, Sterol O-acyltransferase, Urea, General Medicine
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6
المؤلفون: Brian R. Krause, W. H. Roark, Bruce D. Roth, R. L. Stanfield, Reynold Homan, J. A. Picard, K. L. Hamelehle, Maureen K. Anderson, R. F. Bousley
المصدر: ChemInform. 27
مصطلحات موضوعية: Biochemistry, Chemistry, In vivo, medicine.drug_class, Sterol O-acyltransferase, medicine, General Medicine, Sulfonylurea
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7
المؤلفون: Brian R. Krause, Bruce D. Roth, R. L. Stanfield, R. F. Bousley, K. L. Hamelehle, Helen T. Lee, W. H. Roark, Joseph Armand Picard, Drago Robert Sliskovic
المصدر: ChemInform. 29
مصطلحات موضوعية: Chemistry, Stereochemistry, Phosphoramidate, General Medicine, Acyl CoA cholesterol O acyltransferase
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8
المؤلفون: Ann Holmes, Bruce D. Roth, C. J. Blankley, Essenburg Ad, K.A. Kieft, W. H. Roark, R. L. Stanfield, Bharat K. Trivedi, Brian R. Krause, Milton L. Hoefle
المصدر: Journal of Medicinal Chemistry. 35:1609-1617
مصطلحات موضوعية: Male, medicine.drug_class, Sterol O-acyltransferase, Alpha (ethology), Carboxamide, Cholesterol, Dietary, Structure-Activity Relationship, In vivo, Drug Discovery, medicine, Animals, Potency, IC50, Hypolipidemic Agents, chemistry.chemical_classification, Fatty acid, Rats, Inbred Strains, Rats, Cholesterol, Enzyme, chemistry, Biochemistry, Molecular Medicine, lipids (amino acids, peptides, and proteins), Rabbits, Sterol O-Acyltransferase
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9
المؤلفون: J. A. Picard, M. K. Shaw, W. H. Roark, R. L. Stanfield, Roger S. Newton, Bruce David Roth, Drago Robert Sliskovic, B.R. Krause, C. J. Blankley, Catherine Sekerke
المصدر: Journal of Medicinal Chemistry. 35:2095-2103
مصطلحات موضوعية: Male, Chemical Phenomena, Pyridines, Stereochemistry, Reductase, chemistry.chemical_compound, Dogs, In vivo, Drug Discovery, polycyclic compounds, medicine, Animals, Lovastatin, Pravastatin, Molecular Structure, biology, Chemistry, Physical, Chemistry, Anticholesteremic Agents, nutritional and metabolic diseases, Biological activity, Hydroxymethylglutaryl-CoA reductase, Cholesterol, Enzyme inhibitor, Pyran, Pyrazines, biology.protein, Pyrazoles, Molecular Medicine, Female, lipids (amino acids, peptides, and proteins), Hydroxymethylglutaryl-CoA Reductase Inhibitors, medicine.drug
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10
المؤلفون: A M, Doherty, J S, Kaltenbronn, J P, Hudspeth, J T, Repine, W H, Roark, I, Sircar, F J, Tinney, C J, Connolly, J C, Hodges, M D, Taylor
المصدر: Journal of Medicinal Chemistry. 34:1258-1271
مصطلحات موضوعية: Male, Models, Molecular, Molecular Conformation, Cathepsin D, Structure-Activity Relationship, chemistry.chemical_compound, Renin, Drug Discovery, Renin–angiotensin system, Side chain, Animals, Potency, Enzyme Inhibitors, Binding site, Antihypertensive Agents, Binding Sites, Dipeptide, Molecular Structure, biology, Lysine, In vitro, Kinetics, Macaca fascicularis, Biochemistry, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine