-
1
المؤلفون: Marco M. Gottardis, Robert Kramer, Gregory Vite, Shen-Jue Chen, Joseph Dinchuk, William R. Foster, Mark E. Salvati, Weifang Shan, Mary Obermeier, J. Suso Platero, Thomas E. Spires, Liang Schweizer, Cheryl A. Rizzo, Janet Dell-John, Mary Ellen Cvijic, Aaron Balog, Maria Jure-Kunkel, Ricardo M. Attar
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8ea96b450993c30817e08b09d67ecd09
https://doi.org/10.1158/0008-5472.22377966 -
2
المؤلفون: Marco M. Gottardis, Robert Kramer, Gregory Vite, Shen-Jue Chen, Joseph Dinchuk, William R. Foster, Mark E. Salvati, Weifang Shan, Mary Obermeier, J. Suso Platero, Thomas E. Spires, Liang Schweizer, Cheryl A. Rizzo, Janet Dell-John, Mary Ellen Cvijic, Aaron Balog, Maria Jure-Kunkel, Ricardo M. Attar
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::77108c0dff54d0d9d17df83470660395
https://doi.org/10.1158/0008-5472.22377963.v1 -
3
المؤلفون: Marco M. Gottardis, Robert Kramer, Gregory Vite, Shen-Jue Chen, Joseph Dinchuk, William R. Foster, Mark E. Salvati, Weifang Shan, Mary Obermeier, J. Suso Platero, Thomas E. Spires, Liang Schweizer, Cheryl A. Rizzo, Janet Dell-John, Mary Ellen Cvijic, Aaron Balog, Maria Jure-Kunkel, Ricardo M. Attar
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::71c30c0ceeb3ee6de838292a026446d0
https://doi.org/10.1158/0008-5472.22377969 -
4
المؤلفون: Lisa M. Kopcho, Johnni Gullo-Brown, Shweta Padmanabhan, Pattasseri Shabeerali, Arvind Mathur, Prabhakar Rajanna, Lorell Discenza, Liping Zhang, Zhenqiu Hong, Sarah C. Traeger, Zheng Yang, Cherney Emily Charlotte, Richard Rampulla, David K. Williams, Gopal Dhar, Kimberly A. Foster, James Kempson, Derrick Maley, Mary F. Grubb, Xiao Zhu, Xin Li, Weifang Shan, Robert M. Borzilleri, Diane Delpy, Kevin Stefanski, T. Thanga Mariappan, Gregory D. Vite, Kathy A. Johnston, Audris Huang, Asoka Ranasinghe, Mark Fereshteh, Aravind Anandam, Steven P. Seitz, John T. Hunt, Aaron Balog, Celia D’Arienzo, Anuradha Gupta, Tai-An Lin, Roshan Y. Nimje, Weiwei Guo, Christine Huang, Venkata Murali, Sandeep Mahankali
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: chemistry.chemical_compound, Oxidative metabolism, chemistry, Metastatic melanoma, Mouse xenograft, Organic Chemistry, Drug Discovery, Pyridine, Quinoline, Biochemistry, Combinatorial chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f0f0d7f8a891846e7ad07844b139d549
https://europepmc.org/articles/PMC8274105/ -
5
المؤلفون: M. Jure-Kunkel, Jay A. Markwalder, Weifang Shan, Bin Chen, Steven P. Seitz, Andrew Nation, John T. Hunt, Lauren Haque, Gregory D. Vite, Jennifer Donnell, David K. Williams, Kelly L. Covello, Aaron Balog, Hart Amy C, Sunil Kumar Mandal, Libing Chen
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:732-736
مصطلحات موضوعية: 0301 basic medicine, Clinical Biochemistry, Pharmaceutical Science, Phenylenediamines, Biochemistry, HeLa, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Immune system, o-Phenylenediamine, Drug Discovery, Humans, Indoleamine-Pyrrole 2,3,-Dioxygenase, Potency, Enzyme Inhibitors, Indoleamine 2,3-dioxygenase, Molecular Biology, chemistry.chemical_classification, Tumor microenvironment, biology, Organic Chemistry, biology.organism_classification, 030104 developmental biology, Enzyme, chemistry, 030220 oncology & carcinogenesis, Microsomes, Liver, Cancer research, Molecular Medicine, Kynurenine, HeLa Cells
-
6
المؤلفون: Janet Dell-John, John D. Dimarco, Cheryl A. Rizzo, Mark E. Salvati, Steven H. Spergel, Gregory Scott Martin, Weifang Shan, Aaron Balog, Georgia Cornelius, Richard Rampulla, Marco M. Gottardis, Andrew Nation, Christian L. Holst, Liang Schweizer, Gregory D. Vite, Lana M. Rossiter, Ricardo M. Attar, David J. Fairfax, Thomas E. Spires, Stanley R. Krystek, George L. Trainor, Jack Z. Gougoutas
المصدر: ACS Medicinal Chemistry Letters. 6:908-912
مصطلحات موضوعية: Nonsteroidal, Bicalutamide, business.industry, digestive, oral, and skin physiology, Organic Chemistry, Antagonist, Cancer, Pharmacology, medicine.disease, Biochemistry, In vitro, Androgen receptor, stomatognathic diseases, Prostate cancer, chemistry.chemical_compound, chemistry, Drug Discovery, Medicine, Androgen receptor antagonist, business, medicine.drug
-
7
المؤلفون: George L. Trainor, Jun Dai, Arvind Mathur, Francis Y. Lee, Sunilkumar Mandal, Yingru Zhang, Richard Rampulla, Kiran Babu Gona, Patrice Gill, Raja Thiruvenkadam, Victor R. Guarino, Wen-Ching Han, Ding Ren Shen, Aaron Balog, Mary Ellen Cvijic, Dauh-Rurng Wu, Gregory D. Vite, Krista Menard, Anne Rose, Sathiah Kandula, Ashvinikumar V. Gavai, Weifang Shan, John T. Hunt, Asoka Ranasinghe, Kelly McGlinchey, Richard A. Westhouse, Claude A. Quesnelle, Derek J. Norris, Mei-Li Wen, Ronald E. White, Kamalraj Thiyagarajan
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:1905-1909
مصطلحات موضوعية: Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Antineoplastic Agents, Pharmacology, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Receptor, Solid tumor, Molecular Biology, Cell Proliferation, Benzodiazepinones, Dose-Response Relationship, Drug, Molecular Structure, Receptors, Notch, Chemistry, Organic Chemistry, Biological activity, Neoplasms, Experimental, medicine.disease, Leukemia, Orally active, Microsomes, Liver, Molecular Medicine, Drug Screening Assays, Antitumor
-
8
المؤلفون: Claude A. Quesnelle, Patrice Gill, Richard Rampulla, Ching Su, Gerry Everlof, George L. Trainor, Ke Chen, Vinod Arora, Richard A. Westhouse, Celia D’Arienzo, Andrew J. Tebben, Weifang Shan, John T. Hunt, Derek J. Norris, Louis J. Lombardo, Zheng Yang, Arvind Mathur, Mei-Li Wen, Yingru Zhang, Dauh-Rurng Wu, Wen-Ching Han, Krista Menard, Victor R. Guarino, Asoka Ranasinghe, Richard E. Olson, Ashvinikumar V. Gavai, Bruce S. Fischer, Phil S. Baran, Anne Rose, Lan Xiao, Ronald E. White, Mary Ellen Cvijic, Gregory D. Vite, Ding Ren Shen, Jere E. Meredith, Haiqing Wang, Francis Y. Lee, Aaron Balog
المصدر: ACS Medicinal Chemistry Letters. 6:523-527
مصطلحات موضوعية: business.industry, Organic Chemistry, Pharmacology, medicine.disease, Biochemistry, T Acute Lymphoblastic Leukemia, Leukemia, In vivo, Drug Discovery, medicine, Receptor, business, Solid tumor, Clinical evaluation, Triple-negative breast cancer
-
9
المؤلفون: Kelly J. Fitzgerald, David Spiegel, Aaron Balog, Weifang Shan, Andrew Zhang, Eugene F. Douglass, Mariya D. Kolesnikova, Patrick J. McEnaney
المصدر: Journal of the American Chemical Society
مصطلحات موضوعية: Glutamate Carboxypeptidase II, Protein Conformation, Chemistry Techniques, Synthetic, 01 natural sciences, Biochemistry, Article, Antibodies, Catalysis, 03 medical and health sciences, Prostate cancer, Colloid and Surface Chemistry, Phagocytosis, Antigen, Biomimetic Materials, Cell Line, Tumor, Glutamate carboxypeptidase II, medicine, Humans, 030304 developmental biology, 0303 health sciences, biology, 010405 organic chemistry, Chemistry, Receptors, IgG, Cancer, General Chemistry, medicine.disease, 3. Good health, 0104 chemical sciences, Synthetic antibody, Cell biology, Molecular Docking Simulation, Molecular Weight, Drug Design, Antigens, Surface, Cancer cell, biology.protein, Fc-Gamma Receptor, Antibody
-
10
المؤلفون: George L. Trainor, Andrew Nation, Ricardo M. Attar, Jun Dai, Xiao Zhu, Jing Chen, Mary T. Obermeier, Weifang Shan, Mary Ellen Cvijic, Gregory D. Vite, Cheryl A. Rizzo, Sarah C. Traeger, Michael Galella, Ashvinikumar V. Gavai, Thomas E. Spires, Aaron Balog, Yingru Zhang, Jieping Geng
المصدر: Bioorganicmedicinal chemistry letters. 26(23)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Pharmacology, Biochemistry, 03 medical and health sciences, Bridged Bicyclo Compounds, Structure-Activity Relationship, 0302 clinical medicine, Pharmacokinetics, Naphthalenesulfonates, Cell Line, Tumor, Drug Discovery, Androgen Receptor Antagonists, Structure–activity relationship, Androgen receptor antagonist, Animals, Humans, Molecular Biology, Bicyclic molecule, Chemistry, Organic Chemistry, Biological activity, Rats, Androgen receptor, 030104 developmental biology, Nuclear receptor, Receptors, Androgen, 030220 oncology & carcinogenesis, Molecular Medicine