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1
المؤلفون: Candace Crogan-Grundy, Nilantha Sudath Sirisoma, Shailaja Kasibhatla, Sui Xiong Cai, William Kemnitzer, Songchun Jiang, John Drewe, Ben Tseng
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1288-1292
مصطلحات موضوعية: Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Carboxamide, Ring (chemistry), Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Structure–activity relationship, Cytotoxicity, Molecular Biology, Fluorenes, Aryl, Organic Chemistry, HCT116 Cells, Amides, High-Throughput Screening Assays, Mechanism of action, chemistry, Caspases, Molecular Medicine, medicine.symptom, Lead compound
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2
المؤلفون: John Drewe, Ben Tseng, William Kemnitzer, Shailaja Kasibhatla, Sui Xiong Cai, Han-Zhong Zhang, Jared Kuemmerle
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4410-4415
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Primary alcohol, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Cell Line, Tumor, Furan, Drug Discovery, Animals, Combinatorial Chemistry Techniques, Humans, Hydroxymethyl, Infusions, Intravenous, Cytotoxicity, Molecular Biology, Oxadiazoles, Molecular Structure, Aryl, Organic Chemistry, Water, In vitro, Models, Chemical, Solubility, chemistry, Drug Design, Molecular Medicine, Neoplasm Transplantation
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3
المؤلفون: Sui Xiong Cai, Chris May, Ben Tseng, John Drewe, Nilantha Sudath Sirisoma, William Kemnitzer
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:3536-3540
مصطلحات موضوعية: Stereochemistry, High-throughput screening, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Biochemistry, Chemical synthesis, Structure-Activity Relationship, In vivo, Cell Line, Tumor, Drug Discovery, Humans, Structure–activity relationship, Inducer, Molecular Biology, Aniline Compounds, Chemistry, Organic Chemistry, Pyrimidines, Cell culture, Caspases, Cancer cell, Molecular Medicine, Drug Screening Assays, Antitumor
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4
المؤلفون: William, Kemnitzer, Jared, Kuemmerle, Songchun, Jiang, Nilantha, Sirisoma, Shailaja, Kasibhatla, Candace, Crogan-Grundy, Ben, Tseng, John, Drewe, Sui Xiong, Cai
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:3481-3484
مصطلحات موضوعية: Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Biochemistry, Structure-Activity Relationship, Caspases, Cell Line, Tumor, Drug Discovery, Quinolines, Humans, Molecular Medicine, Drug Screening Assays, Antitumor, Molecular Biology
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5
المؤلفون: William, Kemnitzer, Nilantha, Sirisoma, Bao, Nguyen, Songchun, Jiang, Shailaja, Kasibhatla, Candace, Crogan-Grundy, Ben, Tseng, John, Drewe, Sui Xiong, Cai
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:3045-3049
مصطلحات موضوعية: Fluorenes, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, HCT116 Cells, Biochemistry, Structure-Activity Relationship, Caspases, Cell Line, Tumor, Drug Design, Drug Discovery, Humans, Pyrazoles, Molecular Medicine, Drug Screening Assays, Antitumor, Molecular Biology
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6
المؤلفون: Nilantha Sudath Sirisoma, Songchun Jiang, Han-Zhong Zhang, John Drewe, Sui Xiong Cai, William Kemnitzer, Ben Tseng, Candace Crogan-Grundy, Shailaja Kasibhatla, Jared Kuemmerle
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:6259-6264
مصطلحات موضوعية: Clinical Biochemistry, Cell, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Biochemistry, Structure-Activity Relationship, Drug Discovery, medicine, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Cytotoxicity, Molecular Biology, Caspase, Molecular Structure, biology, Cell growth, Chemistry, Tubulin Modulators, Organic Chemistry, HCT116 Cells, medicine.anatomical_structure, Cell culture, Caspases, Cancer cell, Quinolines, biology.protein, Molecular Medicine, Female, Drug Screening Assays, Antitumor
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7
المؤلفون: Shailaja Kasibhatla, Ben Tseng, Real Denis, Candace Crogan-Grundy, Serge Lamothe, Henriette Gourdeau, Songchun Jiang, Charles Blais, Giorgio Attardo, Hong Zhang, John Drewe, William Kemnitzer, Sui Xiong Cai
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:5571-5575
مصطلحات موضوعية: Stereochemistry, Chemistry, Pharmaceutical, High-throughput screening, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Humans, Structure–activity relationship, Pyrroles, Cytotoxicity, Molecular Biology, Cell Proliferation, Pyrrole, chemistry.chemical_classification, Bicyclic molecule, Aryl, Organic Chemistry, Enzyme Activation, Models, Chemical, chemistry, Chromones, Caspases, Drug Design, Molecular Medicine, Drug Screening Assays, Antitumor, Lactone
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8
المؤلفون: Sui Xiong Cai, Serge Lamothe, Candace Crogan-Grundy, Shailaja Kasibhatla, Monica Bubenik, William Kemnitzer, John Drewe, Henriette Gourdeau, Giorgio Attardo, Yan Wang, Songchun Jiang, Real Denis, Denis Labrecque, Ben Tseng
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:603-607
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Apoptosis, Ether, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Amide, Drug Discovery, Humans, Structure–activity relationship, Benzopyrans, Cytotoxicity, Molecular Biology, Caspase, chemistry.chemical_classification, biology, Chemistry, Aryl, Organic Chemistry, Enzyme, Caspases, biology.protein, Molecular Medicine, Cell Division
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9
المؤلفون: Lifen Xu, Shailaja Kasibhatla, Nancy Barriault, Denis Labrecque, Jennifer Dodd, Louis Vaillancourt, Shaojuan Jia, Henriette Gourdeau, Serge Lamothe, Ben Tseng, Songchun Jiang, Sui Xiong Cai, Candace Crogan-Grundy, John Drewe, Giorgio Attardo, William Kemnitzer, Real Denis, Sylvie Charron, Hong Zhang, Jianghong Zhao
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:4745-4751
مصطلحات موضوعية: Stereochemistry, High-throughput screening, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, medicine, Humans, Structure–activity relationship, Benzopyrans, Cytotoxicity, Molecular Biology, Caspase, Cell Proliferation, biology, Cell growth, Organic Chemistry, Enzyme Activation, Mechanism of action, chemistry, Cell culture, Caspases, biology.protein, Molecular Medicine, medicine.symptom, Hydrophobic and Hydrophilic Interactions, Lead compound
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10
المؤلفون: Real Denis, Serge Lamothe, Sui Xiong Cai, Ben Tseng, Shailaja Kasibhatla, William Kemnitzer, Denis Labreque, Monica Bubenick, Candace Crogan-Grundy, Giorgio Attardo, Hong Zhang, John Drewe, Henriette Gourdeau, Songchun Jiang
المصدر: Journal of medicinal chemistry. 51(3)
مصطلحات موضوعية: Indoles, Stereochemistry, Antineoplastic Agents, Apoptosis, Chemical synthesis, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, medicine, Structure–activity relationship, Humans, Benzopyrans, Pyrroles, Alkyl, Pyrrole, Cell Proliferation, chemistry.chemical_classification, Cell growth, Chemistry, Aryl, Tubulin Modulators, Enzyme Activation, Mechanism of action, Cell culture, Caspases, Molecular Medicine, medicine.symptom, Drug Screening Assays, Antitumor