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1
المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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2
المؤلفون: Renato T. Skerlj, Jason B. Crawford, Gary Bridger, Wilson Trevor R, Jenny Ji, Bryon Carpenter, Gang Chen
المصدر: Organic Process Research & Development. 16:109-116
مصطلحات موضوعية: Stereochemistry, Longest linear sequence, Chemistry, Organic Chemistry, CCR5 receptor antagonist, Physical and Theoretical Chemistry, Laboratory scale, Combinatorial chemistry
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3
المؤلفون: Curtis Harwig, Rossana Wauthy, Renato Skerlj, Fluri Maria Di, Yongbao Zhu, Duane Veale, Dominique Schols, Gary Bridger, Helen Yee, Wen Yang, Wilson Trevor R, David Bogucki, Christopher Ronald Smith, Erik De Clercq, Krystyna A. Skupinska, Jonathon Langille, Jason M. Crawford, Dana Huskens, Ernie Mceachern
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:262-266
مصطلحات موضوعية: Receptors, CXCR4, Anti-HIV Agents, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Butylamines, Virus Replication, Biochemistry, Chemical synthesis, CXCR4, Heterocyclic Compounds, 1-Ring, Structure-Activity Relationship, Chemokine receptor, Dogs, Pharmacokinetics, Drug Discovery, Animals, Humans, Structure–activity relationship, Calcium Signaling, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Virology, Rats, Viral replication, Aminoquinolines, HIV-1, Molecular Medicine, Benzimidazoles
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4
المؤلفون: Wilson Trevor R, Yuanxi Zhou, Zhongren Wang, David Bogucki, Susan Nan, Katrien Princen, Pedro E. Hernandez-Abad, Renato Skerlj, Jason B. Crawford, Dominique Schols, Eva Maria Boehringer, Sigrid Hatse, Gary Bridger, Markus Metz, Erik De Clercq
المصدر: Journal of Medicinal Chemistry. 53:1250-1260
مصطلحات موضوعية: Receptors, CXCR4, Anti-HIV Agents, Pyridines, Stereochemistry, T-Lymphocytes, T cell, HIV Infections, Virus Replication, Chemical synthesis, Virus, Structure-Activity Relationship, Chemokine receptor, Heterocyclic Compounds, Drug Discovery, medicine, Humans, Structure–activity relationship, Receptor, Molecular Structure, Chemistry, In vitro, medicine.anatomical_structure, Models, Chemical, Biochemistry, Viral replication, HIV-1, Molecular Medicine
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5
المؤلفون: Jason B. Crawford, Gang Chen, Ernie Mceachern, Gary Bridger, Curtis Harwig, Atsma Bern, Alan Kaller, Renato Skerlj, Ian Baird, Wilson Trevor R, Bryon Carpenter, David Gauthier
المصدر: Organic Process Research & Development. 12:823-830
مصطلحات موضوعية: Organic Chemistry, Imine, chemistry.chemical_element, Zinc, Borohydride, CXCR4, Reductive amination, Chemokine Receptor Antagonist, chemistry.chemical_compound, Sodium borohydride, chemistry, Reagent, Organic chemistry, Physical and Theoretical Chemistry
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6
المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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7
المؤلفون: Gary J. Bridger, Wilson Trevor R, Yuanxi Zhou, Renato Skerlj
المصدر: ChemInform. 33
مصطلحات موضوعية: chemistry.chemical_classification, Iodide, chemistry.chemical_element, General Medicine, Ring (chemistry), Combinatorial chemistry, Catalysis, Coupling (electronics), chemistry.chemical_compound, chemistry, Intramolecular force, Reagent, Pyridine, Palladium
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8
المؤلفون: Duane Veale, Jason B. Crawford, Gary Bridger, Erik De Clercq, Dominique Schols, Ernest J. McEachern, Bem Atsma, Katrien Princen, Jonathon Langille, Renato Skerlj, Yuanxi Zhou, Al Kaller, Curtis Harwig, Sigrid Hatse, Susan Nan, Wilson Trevor R
المصدر: Journal of medicinal chemistry. 53(8)
مصطلحات موضوعية: Receptors, CXCR4, Cell Membrane Permeability, Anti-HIV Agents, Administration, Oral, Biological Availability, CCR5 receptor antagonist, Pharmacology, Butylamines, Virus Replication, Cell Line, Chemokine receptor, Heterocyclic Compounds, 1-Ring, Radioligand Assay, Structure-Activity Relationship, Dogs, Drug Discovery, Structure–activity relationship, Animals, Humans, Receptor, CXCR4 antagonist, Chemistry, Stereoisomerism, Small molecule, Rats, Viral replication, Cell culture, Aminoquinolines, HIV-1, Leukocytes, Mononuclear, Molecular Medicine, Benzimidazoles, Calcium
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9
المؤلفون: Yuanxi Zhou, Renato Skerlj, Gary J. Bridger, Wilson Trevor R
المصدر: The Journal of organic chemistry. 67(4)
مصطلحات موضوعية: chemistry.chemical_classification, Intramolecular reaction, Organic Chemistry, Iodide, chemistry.chemical_element, Alkylation, Combinatorial chemistry, Chemical synthesis, chemistry.chemical_compound, chemistry, Intramolecular force, Pyridine, Organic chemistry, Cyclophane, Palladium