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1دورية أكاديمية
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2دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
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3دورية أكاديمية
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4دورية أكاديمية
المؤلفون: Dussault, Patrick H., Woller, Kevin R.
المصدر: The Chemical Educator. March 1996 1(1):1-6
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المؤلفون: Nirupama B. Soni, Anil Vasudevan, Jun Guo, Marina A. Pliushchev, Julie L. Wilsbacher, H. Robin Heyman, Michael R. Michaelides, Kathy Sarris, Bryan K. Sorensen, Richard F. Clark, Noah Tu, Min Cheng, George Doherty, Alla Korepanova, Anurupa Shrestha, Michael L. Curtin, Mikkel Algire, Badagnani Ilaria, Kenton L. Longenecker, Chris Tse, Diana Raich, Woller Kevin R, Robin R. Frey, Violeta L. Marin, Gary G. Chiang, T. Matthew Hansen, Ana L. Aguirre, F. Greg Buchanan, Peter Kovar, David Maag, Dong Cheng, Paul L. Richardson, Ramzi F. Sweis
المصدر: Bioorganicmedicinal chemistry letters. 27(15)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Clinical Biochemistry, Nicotinamide phosphoribosyltransferase, Pharmaceutical Science, Antineoplastic Agents, Isoindoles, Crystallography, X-Ray, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Cell Line, Tumor, Neoplasms, Drug Discovery, Structure–activity relationship, Animals, Humans, Urea, Enzyme Inhibitors, Nicotinamide Phosphoribosyltransferase, Molecular Biology, Cell Proliferation, Antitumor activity, Drug discovery, Cell growth, Organic Chemistry, Substrate (chemistry), Isoindoline, 030104 developmental biology, chemistry, Molecular Medicine, Cytokines
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6دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
7
المؤلفون: Jose-Andres Salmeron, Kevin P. Cusack, Dawn M. George, Thomas D. Gordon, Michael Friedman, Bernd Janssen, Agnieszka Bischoff, Claude Barberis, Woller Kevin R, Yong Jia, Neil Wishart, Shannon R. Fix-Stenzel, Richard W. Dixon, Christopher Quinn, Maria A. Argiriadi, Zhengtian Yu, Anca Clabbers, Hamish Allen, Maria D Moskey
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:4952-4955
مصطلحات موضوعية: Models, Molecular, Molecular model, Pyridines, Stereochemistry, High-throughput screening, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Thiophenes, Crystallography, X-Ray, Biochemistry, MAP3K8, Chemical synthesis, Structure-Activity Relationship, Proto-Oncogene Proteins, Drug Discovery, Combinatorial Chemistry Techniques, Humans, Molecular Biology, chemistry.chemical_classification, Molecular Structure, Bicyclic molecule, biology, Kinase, Organic Chemistry, MAP Kinase Kinase Kinases, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
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المؤلفون: Valerie L. Pivorunas, Douglas Marcotte, Andrew Burchat, Maria A. Argiriadi, Eric R. Goedken, David Banach, Woller Kevin R, Ramkrishna Sadhukhan, Lu Wang, Neil Wishart, Gary Overmeyer, Robert V. Talanian, Dixon Richard W, Medha J. Tomlinson, Jeffrey W. Voss, David W. Borhani, Silvino Sousa, Moore Nigel St John
المصدر: BMC Structural Biology, Vol 12, Iss 1, p 22 (2012)
BMC Structural Biologyمصطلحات موضوعية: Drug, Indazoles, Jak kinase, media_common.quotation_subject, Molecular Sequence Data, Crystal structure, Crystallography, X-Ray, Protein Structure, Secondary, law.invention, Mice, Structure-Activity Relationship, Structural Biology, law, Enzyme Stability, Protein purification, Animals, Humans, Structure–activity relationship, Amino Acid Sequence, Crystallization, Protein Kinase Inhibitors, lcsh:QH301-705.5, Janus Kinases, media_common, TYK2 Kinase, Chemistry, Combinatorial chemistry, Tyk2, Crystallography, lcsh:Biology (General), Drug Design, Proteolysis, Structure based, Research Article
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المؤلفون: Nathan S. Josephsohn, John W. Maull, Moore Nigel St John, Brian Bettencourt, Morytko Michael J, Lu Wang, Edit Tarcsa, Jonathan George, Biqin Li, Paul Rafferty, Diana L. Donnelly-Roberts, Marian T. Namovic, Patrick Betschmann, Michael Friedman, Jose-Andres Salmeron-Garcia, Gavin C. Hirst, Donald Konopacki, Woller Kevin R
المصدر: Bioorganicmedicinal chemistry letters. 18(14)
مصطلحات موضوعية: Chemistry, Pharmaceutical, Clinical Biochemistry, Interleukin-1beta, Pharmaceutical Science, Pharmacology, Biochemistry, Chemical synthesis, Guanidines, Piperazines, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, In vivo, Drug Discovery, Purinergic P2 Receptor Antagonists, Structure–activity relationship, Animals, Humans, Receptor, Molecular Biology, Piperazine, Whole blood, Molecular Structure, Chemistry, Receptors, Purinergic P2, Organic Chemistry, Biological activity, In vitro, Rats, Models, Chemical, Drug Design, Molecular Medicine, Receptors, Purinergic P2X7
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المؤلفون: Haipeng Chen, Morytko Michael J, Anna M. Ericsson, Patrick Betschmann, Diana L. Donnelly-Roberts, Michael F. Jarvis, Marian T. Namovic, William A. Carroll, Paul Rafferty, Woller Kevin R
المصدر: Bioorganicmedicinal chemistry letters. 18(6)
مصطلحات موضوعية: Nitrile, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, In Vitro Techniques, Biochemistry, Chemical synthesis, Piperazines, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Purinergic P2 Receptor Antagonists, Structure–activity relationship, Moiety, Animals, Humans, Receptor, Molecular Biology, Molecular Structure, Chemistry, Receptors, Purinergic P2, Organic Chemistry, Antagonist, In vitro, Recombinant Proteins, Rats, Piperazine, Molecular Medicine, Receptors, Purinergic P2X7