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1
المؤلفون: Shulin Han, Jeremy S. Caldwell, Xiaoqi Gao, Vicki Zhou, Achim Brinker, Xiang-ju Gu
المصدر: Analytical Biochemistry. 385:300-308
مصطلحات موضوعية: chemistry.chemical_classification, Conformational change, ABL, Protein Conformation, Kinase, Allosteric regulation, Mutation, Missense, Biophysics, Cell Biology, Biology, Biochemistry, Small molecule, Cell Line, Enzyme, chemistry, Animals, Humans, Luciferase, Enzyme Inhibitors, Luciferases, Oncogene Proteins v-abl, Molecular Biology, Intracellular
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2
المؤلفون: Ha-Soon, Choi, Zhicheng, Wang, Wendy, Richmond, Xiaohui, He, Kunyong, Yang, Tao, Jiang, Donald, Karanewsky, Xiang-ju, Gu, Vicki, Zhou, Yi, Liu, Jianwei, Che, Christian C, Lee, Jeremy, Caldwell, Takanori, Kanazawa, Ichiro, Umemura, Naoko, Matsuura, Osamu, Ohmori, Toshiyuki, Honda, Nathanael, Gray, Yun, He
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:2689-2692
مصطلحات موضوعية: Pyrimidines, Molecular Structure, Focal Adhesion Protein-Tyrosine Kinases, Organic Chemistry, Clinical Biochemistry, Drug Discovery, Pharmaceutical Science, Molecular Medicine, Enzyme Inhibitors, Molecular Biology, Biochemistry
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3
المؤلفون: Hayk Asatryan, Drew Gunderson, Frederick J. King, Sungjoon Kim, Jason T. Matzen, Daniel G. Sipes, Gang Xia, S. Frank Yan, Andrew I. Su, Jeremy S. Caldwell, Alham Saadat, Markus Warmuth, Peter G. Schultz, Tami Hood, Xiang-ju Gu, Ronak Beigi, Laura Jarnes, Jeff Janes, Michael Garcia, Jonathan S. Melnick, Richard A. Harig, Jim Yuchen Chang, Vicki Zhou, Christopher M. Shaw, Yingyao Zhou, Nathanael S. Gray, Robert T. Downs
المصدر: Proceedings of the National Academy of Sciences. 103:3153-3158
مصطلحات موضوعية: Time Factors, Multidisciplinary, ABL, Databases, Factual, Kinase, Phosphotransferases, Drug Evaluation, Preclinical, Reproducibility of Results, Robotics, Molecular Pharmacology, Computational biology, Biological Sciences, Biology, Small molecule, Molecular biology, Cell Line, Automation, Mice, Structure-Activity Relationship, Drug development, Growth factor receptor, Animals, Structure–activity relationship, Protein Kinase Inhibitors, Proto-oncogene tyrosine-protein kinase Src
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d85ea39d8267429bf0bd1743f5ae5680
https://doi.org/10.1073/pnas.0511292103 -
4
المؤلفون: Xiang-ju Gu, Vicki Zhou, Justin Haugen, Scott A. Lesley, Heath E. Klock, Yi Liu, Shifeng Pan, Nathanael S. Gray, Shulin Han, Michael Hornsby, Daniel McMullan, Jeremy S. Caldwell
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:5467-5473
مصطلحات موضوعية: Models, Molecular, Phosphopeptides, MAPK/ERK pathway, Protein Conformation, Stereochemistry, Clinical Biochemistry, Allosteric regulation, MAP Kinase Kinase 1, Pharmaceutical Science, Biochemistry, chemistry.chemical_compound, Allosteric Regulation, Coumarins, Drug Discovery, Humans, Enzyme Inhibitors, Phosphorylation, Extracellular Signal-Regulated MAP Kinases, Protein kinase A, Molecular Biology, chemistry.chemical_classification, Binding Sites, biology, Organic Chemistry, Coumarin, In vitro, Kinetics, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Signal transduction
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5
المؤلفون: Jeremy S. Caldwell, Heath E. Klock, Achim Brinker, Shulin Han, Xiang-ju Gu, Vicki Zhou
المصدر: Analytical Biochemistry. 331:349-357
مصطلحات موضوعية: Base Sequence, biology, Ligand binding assay, Biophysics, Biotin, Cell Biology, Surface Plasmon Resonance, Geldanamycin, Biochemistry, Hsp90, Radicicol, chemistry.chemical_compound, Scintillation proximity assay, Förster resonance energy transfer, chemistry, Heat shock protein, Fluorescence Resonance Energy Transfer, polycyclic compounds, biology.protein, HSP90 Heat-Shock Proteins, Surface plasmon resonance, Molecular Biology, DNA Primers
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6
المؤلفون: Xueshi Hao, Linyi Wei, Xiang-ju Gu, Warne Robert L, Yi Liu, Dirksen E. Bussiere, Xiaoqi Gao, Tetsuo Uno
المصدر: Bioorganicmedicinal chemistry letters. 20(13)
مصطلحات موضوعية: Models, Molecular, animal structures, Molecular model, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Protein Serine-Threonine Kinases, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, Humans, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Kinase, Organic Chemistry, Pyruvate Dehydrogenase Acetyl-Transferring Kinase, Stereoisomerism, Azepines, In vitro, Enzyme Activation, Enzyme, Drug Design, Molecular Medicine, Signal transduction, Linker
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7
المؤلفون: Gang Xia, Francisco Adrian, Xiang-ju Gu, Markus Warmuth, Sungjoon Kim
المصدر: Current opinion in oncology. 19(1)
مصطلحات موضوعية: Cancer Research, Antineoplastic Agents, Computational biology, Biology, Pharmacology, Cell Line, Mice, Epidermal growth factor, medicine, Animals, Kinome, Protein Kinase Inhibitors, Epidermal Growth Factor, Drug discovery, Kinase, Cancer, medicine.disease, ErbB Receptors, Cell Transformation, Neoplastic, Oncology, Cell culture, Drug Resistance, Neoplasm, Drug Design, Signal transduction, Function (biology), Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::11021e952cc3107741b9b02ff7f786a0
https://pubmed.ncbi.nlm.nih.gov/17133113 -
8
المؤلفون: Osamu Ohmori, Zhicheng Wang, Ha-Soon Choi, Yi Liu, Toshiyuki Honda, Jeremy S. Caldwell, Xiang-ju Gu, Wendy Richmond, Vicki Zhou, Takanori Kanazawa, Nathanael S. Gray, Kunyong Yang, Ichiro Umemura, Naoko Matsuura, Yun He, Donald S. Karanewsky, Tao Jiang, Christian C. Lee, Jianwei Che, Xiaohui He
المصدر: Bioorganicmedicinal chemistry letters. 16(8)
مصطلحات موضوعية: Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Biochemistry, Chemical synthesis, Focal adhesion, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Humans, Pyrroles, Enzyme Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Kinase, Organic Chemistry, In vitro, Enzyme, Pyrimidines, chemistry, Enzyme inhibitor, Focal Adhesion Protein-Tyrosine Kinases, biology.protein, Molecular Medicine, Signal transduction, Drug Screening Assays, Antitumor
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9
المؤلفون: Achim Brinker, Yun He, Vicki Zhou, Jeremy S. Caldwell, Shulin Han, Andreas Kreusch, Scott A. Lesley, Xiang-ju Gu, Ha-Soon Choi
المصدر: Bioorganicmedicinal chemistry letters. 15(5)
مصطلحات موضوعية: Models, Molecular, Time Factors, Molecular model, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Crystal structure, Pyrazole, Crystallography, X-Ray, Biochemistry, Cell Line, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Side chain, Molecule, Humans, HSP90 Heat-Shock Proteins, Molecular Biology, Adenine binding, Molecular Structure, Hydrogen bond, Chemistry, Organic Chemistry, Hydrogen Bonding, Protein Structure, Tertiary, Molecular Medicine, Pyrazoles, Binding domain
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10دورية أكاديمية
المؤلفون: Melnick, Jonathan S., Janes, Jeff, Sungjoon Kim, Chang, Jim Y., Sipes, Daniel G., Gunderson, Drew, James, Laura, Matzen, Jason T., Garcia, Michael E., Hood, Tami L., Ronak Beigi, Gang Xia, Harig, Richard A., Asatryan, Hayk, Yan, S. Frank, Yingyao Zhou, Xiang-Ju Gu, Saadat, Alham, Zhou, Vicki, King, Frederick J.
المصدر: Proceedings of the National Academy of Sciences of the United States of America; 2/28/2006, Vol. 103 Issue 9, p3153-3158, 6p, 1 Color Photograph, 2 Diagrams, 1 Graph
مصطلحات موضوعية: CYTOLOGY, MOLECULAR pharmacology, DRUG development, MOLECULES, PEPTIDES, RNA, FIRE assay, PROTEIN-tyrosine kinases, QUANTITATIVE research