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المؤلفون: John T. Randolph, Matthew J. O’Connor, Fei Han, Charles W. Hutchins, Y. Amy Siu, Min Cho, Yunan Zheng, Jonathan A. Hickson, Jana L. Markley, Vlasios Manaves, Mikkel Algire, Kenton A. Baker, Alex M. Chapman, Sujatha M. Gopalakrishnan, Sanjay C. Panchal, Kelly Foster-Duke, DeAnne F. Stolarik, Anita Kempf-Grote, Darby Dammeier, Stacey Fossey, Qi Sun, Chaohong Sun, Yu Shen, Michael J. Dart, Warren M. Kati, Albert Lai, Ari J. Firestone, Michael E. Kort
المصدر: Journal of Medicinal Chemistry. 66:3852-3865
مصطلحات موضوعية: Drug Discovery, Molecular Medicine
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المؤلفون: Heidi J. Einolf, Barry Jones, Phillip D. Yates, Theunis C. Goosen, Diane Ramsden, Conrad Fung, Y. Amy Siu, Niresh Hariparsad, Simon Wong, Liangfu Chen, Jairam Palamanda, George Zhang, Donald J. Tweedie, Shannon Dallas
المصدر: Drug Metabolism and Disposition. 49:94-110
مصطلحات موضوعية: CYP2B6, Pharmaceutical Science, Guidelines as Topic, Pharmacology, Models, Biological, Risk Assessment, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Drug Development, Cytochrome P-450 CYP1A2, Cytochrome P-450 CYP3A, Humans, Medicine, Drug Interactions, Pharmacokinetics, EC50, ADME, CYP3A4, business.industry, CYP1A2, Reproducibility of Results, Drug interaction, Confidence interval, Cytochrome P-450 CYP2B6, Enzyme Induction, 030220 oncology & carcinogenesis, Hepatocytes, Drug and Narcotic Control, business, Risk assessment
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fa020936133a247e86ba65e02dc01b76
https://doi.org/10.1124/dmd.120.000055 -
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المؤلفون: Sherri Smith, Darrell Nix, Nathalie Rioux, Pete Smith, Joanne Schindler, Amy Kim, Federico Colombo, Y Amy Siu, W. George Lai
مصطلحات موضوعية: Pyridines, Health, Toxicology and Mutagenesis, Biological Availability, Antineoplastic Agents, Tumor cells, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, Piperazines, Rats, Sprague-Dawley, Feces, 03 medical and health sciences, 0302 clinical medicine, Animals, Bile, Humans, Rats, Long-Evans, Tissue Distribution, Pharmacology, Chemistry, Haplorhini, General Medicine, Disposition, Small molecule, Rats, Cell biology, 030220 oncology & carcinogenesis, RNA splicing
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::086ad5cf1dd1b6387552a1d946c35242
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المؤلفون: W. George Lai, Min-Kun Chang, Cynthia A. Zamora, Maiko Nomoto, Y. Amy Siu, Peter Boyd, Edgar Schuck, Jagadeesh Aluri, Bhaskar Rege, Sanae Yasuda, Jim Ferry
المصدر: British Journal of Clinical Pharmacology. 84:952-960
مصطلحات موضوعية: Pharmacology, Drug, Agonist, business.industry, medicine.drug_class, CYP3A, Itraconazole, media_common.quotation_subject, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Pharmacokinetics, 030220 oncology & carcinogenesis, Pharmacodynamics, Medicine, Pharmacology (medical), business, CYP2C9, Fluconazole, medicine.drug, media_common
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المؤلفون: Y. Amy Siu, W. George Lai
المصدر: Drug Metabolism and Disposition. 45:183-189
مصطلحات موضوعية: Metabolic Clearance Rate, Pharmaceutical Science, In Vitro Techniques, Models, Biological, 030226 pharmacology & pharmacy, Substrate Specificity, 03 medical and health sciences, 0302 clinical medicine, medicine, Cytochrome P-450 CYP3A, Humans, Drug Interactions, CYP2C9, Cytochrome P-450 CYP2C9, Pharmacology, Cross-Over Studies, CYP3A4, biology, Chemistry, Cytochrome P450, Substrate (chemistry), Metabolism, Meloxicam, Losartan, Pharmaceutical Preparations, Biochemistry, 030220 oncology & carcinogenesis, Microsomes, Liver, biology.protein, Microsome, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2be46ff02067829ce430655c877d84ec
https://doi.org/10.1124/dmd.116.073510 -
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المؤلفون: Donald J. Tweedie, Robert L. Walsky, Diane Ramsden, Conrad Fung, Liangfu Chen, Michael A. Mohutsky, David B. Buckley, Theunis C. Goosen, Y. Amy Siu, Maria Fitzgerald, Shannon Dallas, George Zhang, Jane R. Kenny, Niresh Hariparsad, Heidi J. Einolf, Joshua G. Dekeyser
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(9)
مصطلحات موضوعية: Flumazenil, Quality Control, CYP3A, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Inventions, False positive paradox, Medicine, Cytochrome P-450 CYP3A, Humans, Clinical significance, Inducer, Drug Interactions, RNA, Messenger, EC50, Messenger RNA, CYP3A4, business.industry, Cytochrome P-450 CYP3A Inducers, In vitro, 030220 oncology & carcinogenesis, Hepatocytes, Drug and Narcotic Control, Rifampin, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1a363861f9fd5379ff3cfeccdf0985ed
https://pubmed.ncbi.nlm.nih.gov/29959133 -
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المؤلفون: Hao Ming-Hong, Y. Amy Siu, W. George Lai, Vaishali Dixit
المصدر: Drug metabolism and pharmacokinetics. 33(5)
مصطلحات موضوعية: 0301 basic medicine, Quinidine, Models, Molecular, CYP2D6, Pharmaceutical Science, Pharmacology, digestive system, Substrate Specificity, Hydroxylation, 03 medical and health sciences, chemistry.chemical_compound, Structure-Activity Relationship, medicine, Humans, heterocyclic compounds, Pharmacology (medical), Enzyme Inhibitors, skin and connective tissue diseases, CYP2C9, Cytochrome P-450 CYP2C9, CYP3A4, Dose-Response Relationship, Drug, Molecular Structure, organic chemicals, Genetic Variation, Dextromethorphan, Recombinant Proteins, Kinetics, 030104 developmental biology, chemistry, Cytochrome P-450 CYP2D6, Celecoxib, Microsome, medicine.drug
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المؤلفون: Y. Amy Siu, Jairam Palamanda, Robert L. Walsky, George Zhang, David B. Buckley, Michael A. Mohutsky, Donald J. Tweedie, Liangfu Chen, Magalie Pardon, Shannon Dallas, Suresh K. Balani, Diane Ramsden, Barry Jones, Heidi J. Einolf, Jane R. Kenny, Odette A. Fahmi, Michael Sinz, Niresh Hariparsad, Joshua G. Dekeyser
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 45(10)
مصطلحات موضوعية: Pharmacology, Medical education, Drug Industry, United States Food and Drug Administration, Drug-drug interaction, MEDLINE, Pharmaceutical Science, Induction time, Positive control, Down-Regulation, 030226 pharmacology & pharmacy, United States, Interaction studies, Food and drug administration, 03 medical and health sciences, Cytochrome P-450 CYP2B6, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, Agency (sociology), Humans, Drug Interactions, Duration (project management), Psychology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::daa706cdb57f6dcbd095aafbcf456d8b
https://pubmed.ncbi.nlm.nih.gov/28646080 -
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المؤلفون: Maiko, Nomoto, Cynthia A, Zamora, Edgar, Schuck, Peter, Boyd, Min-Kun, Chang, Jagadeesh, Aluri, Y Amy, Siu, W George, Lai, Sanae, Yasuda, Jim, Ferry, Bhaskar, Rege
المصدر: British journal of clinical pharmacology. 84(5)
مصطلحات موضوعية: Adult, Male, Adolescent, Cytochrome P-450 CYP2C9 Inhibitors, Platelet Count, Cytochrome P-450 CYP3A Inducers, Thiophenes, Middle Aged, Healthy Volunteers, Thiazoles, Young Adult, Cytochrome P-450 CYP3A Inhibitors, Humans, Drug Interactions, Female, Itraconazole, Rifampin, Fluconazole, Receptors, Thrombopoietin, Cytochrome P-450 CYP2C9 Inducers
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المؤلفون: Maria Fitzgerald, Diane Ramsden, Jane R. Kenny, Josh Dekeyser, Y. Amy Siu, Donald J. Tweedie, Michael A. Mohutsky, Liangfu Chen, George Zhang, Niresh Hariparsad, Shannon Dallas, Theunis C. Goosen, David B. Buckley, Heidi J. Einolf, Robert L. Walsky, Conrad Fung
المصدر: Drug Metabolism and Pharmacokinetics. 34:S44
مصطلحات موضوعية: Pharmacology, Messenger RNA, CYP3A4, business.industry, Drug-drug interaction, Pharmaceutical Science, Medicine, Pharmacology (medical), business, Risk assessment, In vitro