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1دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
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2
المؤلفون: Mason Helen J, Karen D. Brown, Valeria Chu, Guyan Liang, Daniel M. Green, Alfred P. Spada, Henry W. Pauls, Ross Bentley, Cuong Ly, Roderick S. Davis, Dennis J. Colussi, Daniel L. Cheney, Michael R. Becker, Y.M. Choi-Sledeski, Christopher T. Dunwiddie, Robert J. Leadley, Ewing William R, John H. Barton
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2539-2544
مصطلحات موضوعية: Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Isostere, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Benzamidine, Amidine, Serine, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Structure–activity relationship, Molecular Biology, Binding Sites, Organic Chemistry, Isoquinolines, Benzamidines, chemistry, Molecular Medicine, Factor Xa Inhibitors
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3
المؤلفون: Alfred P. Spada, Robert J. Leadley, Jonathan S. Mason, Dennis J. Colussi, Ewing William R, Mark H. Perrone, Karen D. Brown, Michael R. Becker, Don D. Cha, Daniel M. Green, Ross Bentley, Henry W. Pauls, Christopher T. Dunwiddie, Jean-Pierre Guilloteau, Y.M. Choi-Sledeski, Sebastien Maignan, Mason Helen J, Vincent E. Manetta, Charles Kasiewski, Valeria Chu, Roderick S. Davis, Suzanne Morgan, Daniel L. Cheney, Jeff Bostwick
المصدر: Journal of Medicinal Chemistry. 42:3557-3571
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, medicine.drug_class, Factor Xa Inhibitor, Thiophenes, Crystallography, X-Ray, Amidine, Structure-Activity Relationship, chemistry.chemical_compound, Thrombin, In vivo, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Sulfonamides, Molecular Structure, biology, Chemistry, Anticoagulant, Anticoagulants, Stereoisomerism, Thrombosis, Trypsin, Pyrrolidinones, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Rabbits, Factor Xa Inhibitors, medicine.drug
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4
المؤلفون: Y.M. Choi-Sledeski, Daniel M. Green, Joseph G. Bruno, Francis A. Volz, Michael N. Chang, John R. Regan, Mcgarry Daniel G
المصدر: The Journal of Organic Chemistry. 62:5174-5190
مصطلحات موضوعية: chemistry.chemical_classification, Organic Chemistry, Iodide, chemistry.chemical_element, Diphenylmethane, Alkylation, chemistry.chemical_compound, Elastase inhibitor, chemistry, Reagent, Functional group, Organic chemistry, Phenol, Palladium
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5
المؤلفون: Salvino Joseph M, Michael R. Becker, Yong Gong, Y.M. Choi-Sledeski, Roderick S. Davis, Henry W. Pauls, Karen D. Brown, Valeria Chu
المصدر: Bioorganicmedicinal chemistry letters. 10(10)
مصطلحات موضوعية: medicine.drug_mechanism_of_action, Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Anticoagulants, Biochemistry, Combinatorial chemistry, Pyrrolidinones, chemistry.chemical_compound, Structure-Activity Relationship, Sulfonate, Phase (matter), Drug Discovery, medicine, Molecular Medicine, Combinatorial Chemistry Techniques, Molecular Biology, Polymer supported, Factor Xa Inhibitors
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6
المؤلفون: Charles Kasiewski, Suzanne Morgan, Roderick S. Davis, Robert J. Leadley, Jeff Bostwick, Valeria Chu, Henry W. Pauls, Ewing William R, Karen D. Brown, Cuong Ly, Michael R. Becker, Mason Helen J, Ross Bentley, Y.M. Choi-Sledeski, Dennis J. Colussi, Alfred P. Spada, Aiwen Li
المصدر: Bioorganicmedicinal chemistry letters. 9(18)
مصطلحات موضوعية: Thienopyridine, medicine.drug_mechanism_of_action, Stereochemistry, Clinical Biochemistry, Factor Xa Inhibitor, Pharmaceutical Science, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, medicine, Structure–activity relationship, Animals, Pyrrolidinones, Molecular Biology, chemistry.chemical_classification, biology, Organic Chemistry, Thrombosis, Sulfonamide, Rats, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Factor Xa Inhibitors
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7
المؤلفون: Sébastien Maignan, Davis Roderick S, Dunwiddie Christopher T, Michael R. Becker, William P. Dankulich, Karen Brown, Jean-Pierre Guilloteau, Mcgarry Daniel G, Daniel M. Green, Christopher L. Heran, Robert L. Morris, Robert J. Leadley, Spada Alfred P, Ross G. Bentley, William R. Ewing, Helen J. Mason, Valeria Chu, Y.M. Choi-Sledeski, Suzanne R Morgan, Daniel L. Cheney, Pauls Henry W, Dennis Colussi, Vincent E. Manetta
المصدر: Journal of medicinal chemistry. 42(18)
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, medicine.drug_mechanism_of_action, Stereochemistry, Factor Xa Inhibitor, Amidines, Rats, Sprague-Dawley, In vivo, Drug Discovery, medicine, Animals, Humans, Sulfones, Binding site, chemistry.chemical_classification, Sulfonamides, Binding Sites, biology, Chemistry, Active site, Anticoagulants, Thrombosis, Trypsin, In vitro, Pyrrolidinones, Rats, Enzyme, Enzyme inhibitor, biology.protein, Molecular Medicine, medicine.drug, Factor Xa Inhibitors, Protein Binding
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8دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
9دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل. -
10دورية أكاديمية
لا يتم عرض هذه النتيجة على الضيوف.
تسجيل الدخول للوصول الكامل.