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المؤلفون: Yann Dudit, Zehong Wan, Don O. Somers, Yingxia Sang, Vipulkumar Kantibhai Patel, Pascal Grondin, Joseph E. Coyle, Veronique Beneton, Rachel McMenamin, Lee William Page, Philip J. Day, Alison Jo-Anne Woolford, Lionel Trottet, Valerio Berdini, Florent Potvain, Sharna J. Rich, Christopher William Murray, Pascal Huet, Lydia Y. W. Lee, Xiaomin Zhang, Eric S. Manas
المصدر: Journal of Medicinal Chemistry. 59:10738-10749
مصطلحات موضوعية: 0301 basic medicine, Virtual screening, biology, Lipoprotein-associated phospholipase A2, Active site, Pharmacology, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, Fragment (logic), 030220 oncology & carcinogenesis, Drug Discovery, Lipophilicity, Lactam, biology.protein, Molecular Medicine, Bioassay, lipids (amino acids, peptides, and proteins), IC50
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المؤلفون: Alison J-A, Woolford, Philip J, Day, Véronique, Bénéton, Valerio, Berdini, Joseph E, Coyle, Yann, Dudit, Pascal, Grondin, Pascal, Huet, Lydia Y W, Lee, Eric S, Manas, Rachel L, McMenamin, Christopher W, Murray, Lee W, Page, Vipulkumar K, Patel, Florent, Potvain, Sharna J, Rich, Yingxia, Sang, Don O, Somers, Lionel, Trottet, Zehong, Wan, Xiaomin, Zhang
المصدر: Journal of medicinal chemistry. 59(23)
مصطلحات موضوعية: Models, Molecular, Dose-Response Relationship, Drug, Lactams, Molecular Structure, Administration, Oral, Biological Availability, Crystallography, X-Ray, Rats, Structure-Activity Relationship, Dogs, 1-Alkyl-2-acetylglycerophosphocholine Esterase, Animals, Humans, Tissue Distribution, Enzyme Inhibitors
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المؤلفون: Delphine Delannée, Pascal Huet, Chun-wa Chung, Anne Marie Jeanne Bouillot, Françoise Gellibert, Antonia J. Lewis, Yann Lamotte, Yann Dudit, Lionel Trottet, Jason Witherington, Olivier Mirguet, Edwige Nicodeme, Paul Bamborough, Gael Krysa
المصدر: ChemMedChem. 9(3)
مصطلحات موضوعية: Models, Molecular, Chromosomal Proteins, Non-Histone, Protein domain, Biology, Protein Serine-Threonine Kinases, Crystallography, X-Ray, Biochemistry, Histones, Mice, Structure-Activity Relationship, Transcription (biology), Histone tails, Drug Discovery, Animals, Acetylated histone, General Pharmacology, Toxicology and Pharmaceutics, Naphthyridines, Gene, Protein Kinase Inhibitors, Pharmacology, Messenger RNA, Mice, Inbred BALB C, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Anti-Inflammatory Agents, Non-Steroidal, Nuclear Proteins, Chromatin, Bromodomain, Protein Structure, Tertiary, Molecular Medicine, Transcription Factors
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المؤلفون: Jean-Marie Brusq, Pascal Grondin, Benjamin Beaufils, Frédéric Donche, Stéphane Sautet, Celine Marques, Edwige Nicodeme, Yann Dudit, Catherine-Anne Clément, Pascal Huet, Yannick Saintillan, Eric Boursier, Jérôme Toum, Mathieu Pizzonero, Emilie Rondet, Lionel Trottet, Olivier Mirguet
مصطلحات موضوعية: chemistry.chemical_classification, medicine.medical_specialty, business.industry, Organic Chemistry, AMPK, Type 2 diabetes, medicine.disease, Biochemistry, Proinflammatory cytokine, Endocrinology, Enzyme, Pharmacokinetics, chemistry, Internal medicine, Drug Discovery, Hyperlipidemia, medicine, business, Protein kinase A, Beta oxidation
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8260bf96114fc481fec9048186ad6416
https://europepmc.org/articles/PMC4027520/ -
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المؤلفون: Delphine Delannée, Agnès Costaz, Jonathan Thomas Seal, Lionel Trottet, Rémi Tellier, Jean-Marie Brusq, Olivier Mirguet, Anne Marie Jeanne Bouillot, Sandrine Martin, Gael Krysa, Anne-Benedicte Boullay, Jorge Kirilovsky, Eric Boursier, Jérôme Toum, Yann Dudit, Van-Loc Nguyen, Edwige Nicodeme, Françoise Gellibert, Alizon M. Riou, Pascal Huet, Romain Luc Marie Gosmini, Yann Lamotte, Florence Blandel, Frédéric Donche
المصدر: Bioorganicmedicinal chemistry letters. 22(8)
مصطلحات موضوعية: Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Nerve Tissue Proteins, Biochemistry, Chemical synthesis, Heterocyclic Compounds, 4 or More Rings, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Downregulation and upregulation, Drug Discovery, Structure–activity relationship, Animals, Humans, Histone Chaperones, Molecular Biology, Biological evaluation, Histone Acetyltransferases, Mice, Inbred BALB C, Apolipoprotein A-I, Chemistry, Drug discovery, Organic Chemistry, Nuclear Proteins, Hep G2 Cells, In vitro, Bromodomain, Cell biology, Rats, Up-Regulation, Immunology, Hepatic stellate cell, Quinolines, Molecular Medicine