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1
المؤلفون: Tomohiro Ohashi, Tomoteru Yamasaki, Yasuyuki Debori, Tatsuki Koike, Tomokazu Kusumoto, Ryouta Maeda, Masayuki Fujinaga, Akito Hata, Takeshi Wakabayashi, Yasushi Hattori, Ming-Rong Zhang, Miyanohana Yuhei, Ryo Yamashita, Maki Miyamoto, Yiding Zhang, Hidekatsu Wakizaka
المصدر: Journal of Medicinal Chemistry. 64:11990-12002
مصطلحات موضوعية: Indole test, chemistry.chemical_classification, medicine.diagnostic_test, Chemistry, Diacylglycerol kinase gamma, Phosphatidic acid, Imaging agent, chemistry.chemical_compound, Enzyme, Positron emission tomography, Drug Discovery, medicine, Biophysics, Molecular Medicine, IC50, Diacylglycerol kinase
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2
المؤلفون: Toshiki Kurosawa, Daiki Sako, Yuma Tega, Yasuyuki Debori, Yumi Tomihara, Kazunobu Aoyama, Yoshiyuki Kubo, Nobuyuki Amano, Yoshiharu Deguchi
المصدر: Pharmaceutical research. 39(7)
مصطلحات موضوعية: Pharmacology, Tight Junction Proteins, Organic Chemistry, Induced Pluripotent Stem Cells, Pharmaceutical Science, Brain, Endothelial Cells, Membrane Transport Proteins, Blood-Brain Barrier, Molecular Medicine, Humans, Pharmacology (medical), RNA, Messenger, Cells, Cultured, Biotechnology
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3
المؤلفون: Yasushi, Hattori, Tomoteru, Yamasaki, Tomohiro, Ohashi, Yuhei, Miyanohana, Tomokazu, Kusumoto, Ryouta, Maeda, Maki, Miyamoto, Yasuyuki, Debori, Akito, Hata, Yiding, Zhang, Hidekatsu, Wakizaka, Takeshi, Wakabayashi, Masayuki, Fujinaga, Ryo, Yamashita, Ming-Rong, Zhang, Tatsuki, Koike
المصدر: Journal of medicinal chemistry. 64(16)
مصطلحات موضوعية: Male, Mice, Inbred C57BL, Rats, Sprague-Dawley, Diacylglycerol Kinase, Indoles, Drug Design, Positron-Emission Tomography, Animals, Brain, Humans, Carbon Radioisotopes, Radiopharmaceuticals
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4
المؤلفون: Osamu Kurasawa, Yasutomi Asano, Ke Li, Hiroshi Banno, Jun Fujimoto, Georgia Kefala, Gyorgy Snell, Irena Levin, Takuto Kojima, Ryo Mizojiri, Bi-Ching Sang, Richard Tjhen, Michael G. Klein, Scott Weston Lane, Isaac Hoffman, Tsuyoshi Ishii, Douglas R. Cary, Xin Liu, Akito Hata, Tadahiro Nambu, Yasuyuki Debori, Tomoya Sameshima, Terufumi Takagi, Steve C. Ding, Akito Nakamura, Maki Miyamoto
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: chemistry.chemical_classification, Tumor microenvironment, Asparaginase, 010405 organic chemistry, Kinase, Organic Chemistry, Allosteric regulation, Pharmacology, 01 natural sciences, Biochemistry, 0104 chemical sciences, Amino acid, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, chemistry, Amino acid homeostasis, Cell culture, Drug Discovery, Potency
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5
المؤلفون: Toshiki Kurosawa, Daiki Sako, Yuma Tega, Yasuyuki Debori, Yumi Tomihara, Kazunobu Aoyama, Yoshiyuki Kubo, Nobuyuki Amano, Yoshiharu Deguchi
المصدر: Pharmaceutical Research. 39:1661-1661
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Pharmaceutical Science, Molecular Medicine, Pharmacology (medical), Biotechnology
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6
المؤلفون: Takao Watanabe, Yasuyuki Debori, Kazuya Maeda, Hiroyuki Kusuhara, Shigeru Horita, Hideki Nakayama, Brian W. Ogilvie, Zhuohan Hu, Tsunenori Kondo, Yuichi Sugiyama, Andrew Parkinson, Tomoko Watanabe
المصدر: Drug Metabolism and Disposition. 39:1031-1038
مصطلحات موضوعية: Anions, medicine.medical_specialty, Organic anion transporter 1, Metabolic Clearance Rate, Metabolite, Pharmaceutical Science, In Vitro Techniques, Organic Anion Transporters, Sodium-Independent, Substrate Specificity, chemistry.chemical_compound, Pharmacokinetics, Predictive Value of Tests, Internal medicine, medicine, Humans, Gemfibrozil, Drug Interactions, Cells, Cultured, Pharmacology, Kidney, biology, Drug interaction, Kidney Tubules, Endocrinology, medicine.anatomical_structure, Liver, Pharmaceutical Preparations, chemistry, Hepatocytes, biology.protein, Glucuronide, Pravastatin, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::11172aa043291caac1d8927c37624a3d
https://doi.org/10.1124/dmd.110.036129 -
7
المؤلفون: Yuichi Sugiyama, Hiroyuki Kusuhara, Yasuyuki Debori, Hisamitsu Hayashi, Alfred H. Schinkel, Kazuya Maeda, Soichiro Matsushima, John D. Schuetz
المصدر: Molecular Pharmacology. 73:1474-1483
مصطلحات موضوعية: Male, medicine.medical_specialty, ATP-binding cassette transporter, Pharmacology, Cell Line, Bile Acids and Salts, Mice, chemistry.chemical_compound, Adenosine Triphosphate, Dogs, Pharmacokinetics, Internal medicine, medicine, Animals, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 11, biology, Membrane transport protein, Multidrug resistance-associated protein 2, Membrane Transport Proteins, Biological Transport, Transporter, Glutathione, Multidrug Resistance-Associated Protein 2, Recombinant Proteins, Mice, Inbred C57BL, Organic anion-transporting polypeptide, Endocrinology, Gene Expression Regulation, Liver, chemistry, Quinolines, biology.protein, Molecular Medicine, ATP-Binding Cassette Transporters, Terfenadine, Efflux, Multidrug Resistance-Associated Proteins
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::af3fad81676c24322084d17ad37ac1eb
https://doi.org/10.1124/mol.107.041459 -
8
المؤلفون: Yasuyuki Debori, Hisamichi Yamabayashi, Hiroyuki Kuroiwa, Norihiro Takeuchi, Noriko Higashi, Yuichi Sato, Akiyo Shigematsu, Naoshi Kawai, Awazu Shoji, Joji Yui, Yuko Hamai, Akiko Hatori, Takeo Yamamoto
المصدر: Regulatory Toxicology and Pharmacology. 40:207-218
مصطلحات موضوعية: Pathology, medicine.medical_specialty, Tissue Fixation, Mice, Nude, Mitosis, Bone Neoplasms, Spleen, Biology, Toxicology, Mice, Bone Marrow, In vivo, Cell Line, Tumor, medicine, Animals, Humans, Tissue Distribution, Yttrium Radioisotopes, Amitosis, Lobules of liver, Radionuclide Imaging, Induced pluripotent stem cell, Cell Nucleus, Mice, Inbred BALB C, Osteosarcoma, Stem Cells, General Medicine, medicine.disease, Molecular biology, Jejunum, medicine.anatomical_structure, Area Under Curve, Isotope Labeling, Autoradiography, Plasmacytoma, Stem cell, Epiphyses, Half-Life, Thymidine
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9
المؤلفون: Gyorgy Snell, Mie Yoshimatsu, Hiroyuki Sumi, Yasuyuki Debori, Masato Yabuki, Tomoyasu Ishikawa, Nao Morishita, Bunnai Saito, Sei Yoshida, Zenyu Shiokawa, Yuya Oguro, Douglas R. Dougan, Kentaro Hashimoto, Yohei Kosugi
المصدر: Bioorganicmedicinal chemistry. 21(24)
مصطلحات موضوعية: Models, Molecular, ATP Binding Cassette Transporter, Subfamily B, Cell Membrane Permeability, Indoles, Membrane permeability, Apoptosis Inhibitor, Stereochemistry, Cell Survival, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Apoptosis, Crystallography, X-Ray, Biochemistry, Inhibitor of Apoptosis Proteins, chemistry.chemical_compound, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, HATU, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, Molecular Biology, Cell Proliferation, Indole test, Dose-Response Relationship, Drug, Molecular Structure, Cell growth, Organic Chemistry, XIAP, chemistry, Drug Design, Pyrazines, Lipophilicity, Molecular Medicine, Drug Screening Assays, Antitumor
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10
المؤلفون: Sandrine Camus, Naoki Kotani, Christophe Chesne, Yuichi Sugiyama, Kazuya Maeda, Yasuyuki Debori, Ruoya Li
المصدر: Molecular pharmaceutics. 9(12)
مصطلحات موضوعية: Taurocholic Acid, Organic anion transporter 1, Blotting, Western, Detergents, Pharmaceutical Science, Organic Anion Transporters, Organic Anion Transporters, Sodium-Dependent, Organic Anion Transporters, Sodium-Independent, Flow cytometry, Solute Carrier Organic Anion Transporter Family Member 1B3, Drug Discovery, medicine, Humans, Drug Interactions, Cells, Cultured, Messenger RNA, medicine.diagnostic_test, biology, Symporters, Chemistry, Liver-Specific Organic Anion Transporter 1, HEK 293 cells, Transporter, Biological Transport, Cell Differentiation, Flow Cytometry, Blot, HEK293 Cells, Biochemistry, Cell culture, biology.protein, Hepatocytes, Molecular Medicine, Function (biology)