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1
المؤلفون: Keng-Chang Tsai, Yih-Shyun E. Cheng, Jim-Min Fang, Ting-Jen Cheng, Jia-Tsrong Jan, Peng-Hao Hsu, Kuan-Lin Wu, Din-Chi Chiu, Pei-Shan Lee
المصدر: European Journal of Medicinal Chemistry. 154:314-323
مصطلحات موضوعية: Oseltamivir, Stereochemistry, Carboxylic acid, Administration, Oral, Microbial Sensitivity Tests, 010402 general chemistry, Antiviral Agents, 01 natural sciences, Structure-Activity Relationship, chemistry.chemical_compound, Zanamivir, Oral administration, Drug Discovery, medicine, Moiety, Prodrugs, Guanidine, Pharmacology, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, biology, 010405 organic chemistry, Organic Chemistry, General Medicine, Prodrug, Orthomyxoviridae, 0104 chemical sciences, Molecular Docking Simulation, chemistry, biology.protein, Hydrophobic and Hydrophilic Interactions, Neuraminidase, medicine.drug
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2
المؤلفون: Ting-Jen Cheng, Yih-Shyun E. Cheng, Jim-Min Fang, Bei-Tao Hong
المصدر: European journal of medicinal chemistry. 163
مصطلحات موضوعية: Carboxylic acid, Carboxylic Acids, Neuraminidase, Sulfonic acid, Sulfinic acid, 01 natural sciences, Medicinal chemistry, Antiviral Agents, Sulfone, 03 medical and health sciences, Hydrolysis, chemistry.chemical_compound, Structure-Activity Relationship, Influenza A Virus, H1N1 Subtype, Oseltamivir, Drug Discovery, Influenza, Human, Humans, Sulfones, Enzyme Inhibitors, 030304 developmental biology, Pharmacology, chemistry.chemical_classification, 0303 health sciences, biology, Sulfur Compounds, 010405 organic chemistry, Organic Chemistry, Active site, General Medicine, Boronic Acids, 0104 chemical sciences, Sulfonate, chemistry, biology.protein, Sulfonic Acids, Boronic acid
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3
المؤلفون: Chung-Ming Sun, Ting Jen Cheng, Yih Shyun E. Cheng, Olivia A. Lin, Suz Ting Wang, Yufeng J. Tseng, Wen I. Huang, Shi Yun Wang, Meng I. Lin, Chia Hsin Lee, Prasad S. Dangate, Bo-Han Su, Wen Chun Wu
المصدر: European Journal of Medicinal Chemistry. 102:477-486
مصطلحات موضوعية: viruses, RNA-dependent RNA polymerase, Microbial Sensitivity Tests, medicine.disease_cause, Antiviral Agents, Virus, Structure-Activity Relationship, Viral Proteins, chemistry.chemical_compound, Influenza A Virus, H1N1 Subtype, Quinoxalines, RNA polymerase, Drug Discovery, Influenza A virus, medicine, Pyrroles, Binding site, Nuclear export signal, Ribonucleoprotein, Pharmacology, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, virus diseases, General Medicine, Virology, Nucleoprotein, Nucleoproteins, Pyrimidines, chemistry
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4
المؤلفون: Wen-I Huang, Bei-Tao Hong, Yih-Shyun E. Cheng, Chi-Huey Wong, Keng-Chang Tsai, Chun-Lin Chen, Shi-Yun Wang, Jim-Min Fang
المصدر: Bioorganic & Medicinal Chemistry. 22:6647-6654
مصطلحات موضوعية: Models, Molecular, Oseltamivir, Stereochemistry, medicine.drug_class, Carboxylic acid, Clinical Biochemistry, Substituent, Neuraminidase, Pharmaceutical Science, Microbial Sensitivity Tests, medicine.disease_cause, Antiviral Agents, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Influenza A Virus, H1N1 Subtype, Drug Discovery, Influenza A virus, medicine, Enzyme Inhibitors, Molecular Biology, IC50, chemistry.chemical_classification, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, Neuraminidase inhibitor, biology, Chemistry, Organic Chemistry, Sulfonamide, biology.protein, Molecular Medicine
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5
المؤلفون: Jim-Min Fang, Shi-Yun Wang, Jiun-Jie Shie, Tzu-Chen Lin, Yih-Shyun E. Cheng, Chun-Jung Lin, Jia-Tsrong Jan, Chun-Lin Chen, Keng-Chang Tsai, Chi-Huey Wong
المصدر: European Journal of Medicinal Chemistry. 81:106-118
مصطلحات موضوعية: Male, Models, Molecular, Oseltamivir, Phosphorous Acids, medicine.drug_class, Stereochemistry, viruses, Molecular Conformation, Biological Availability, Neuraminidase, Microbial Sensitivity Tests, Antiviral Agents, Intestinal absorption, Cell Line, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Drug Discovery, medicine, Animals, Humans, Enzyme Inhibitors, Pharmacology, Mice, Inbred BALB C, Mice, Inbred ICR, Dose-Response Relationship, Drug, biology, Influenza treatment, Neuraminidase inhibitor, Organic Chemistry, Lethal dose, virus diseases, Esters, General Medicine, Orthomyxoviridae, Phosphonate, chemistry, Biochemistry, biology.protein, Female, Nasal administration, Caco-2 Cells, Chickens
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6
المؤلفون: Charng-Sheng Tsai, Hsin-Yung Yen, Meng-I Lin, Tsung-I Tsai, Shi-Yun Wang, Wen-I Huang, Tsui-Ling Hsu, Yih-Shyun E. Cheng, Jim-Min Fang, Chi-Huey Wong
المصدر: Proceedings of the National Academy of Sciences. 110:2466-2471
مصطلحات موضوعية: Proteomics, Streptavidin, Molecular Probe Techniques, Neuraminidase, Conjugated system, Sialidase, DNA Adducts, chemistry.chemical_compound, Biotin, Tandem Mass Spectrometry, Influenza, Human, Humans, Moiety, Multidisciplinary, Molecular Structure, biology, Biochemistry, chemistry, Alkynes, Molecular Probes, Physical Sciences, Click chemistry, biology.protein, Click Chemistry, Molecular probe, Chromatography, Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4fd10f19e998cc2c3a085dad826cd43d
https://doi.org/10.1073/pnas.1222183110 -
7
المؤلفون: Jim-Min Fang, Wen-I Huang, Ting-Jen R. Cheng, Chi-Huey Wong, Nung-Sen Wang, Chung-Kai Cheng, Yih-Shyun E. Cheng, Chung-Yi Wu, Ho-Sheng Wu, Wen-Hsien Wen, Ching-Yao Su, Chun-Lin Chen, Shi-Yun Wang, Mengi Lin, Ming-Tsan Liu, Chien-Tai Ren
المصدر: Angewandte Chemie. 125:384-388
مصطلحات موضوعية: Oseltamivir, viruses, Drug resistance, Pharmacology, medicine.disease_cause, Antiviral Agents, Binding, Competitive, Catalysis, chemistry.chemical_compound, Zanamivir, Influenza A Virus, H1N2 Subtype, Drug Resistance, Viral, Influenza A virus, medicine, Humans, biology, virus diseases, General Chemistry, General Medicine, biochemical phenomena, metabolism, and nutrition, Virology, respiratory tract diseases, chemistry, biology.protein, Neuraminidase, medicine.drug
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8
المؤلفون: Chih An Chen, Shi Yun Wang, Oliver Yoa Pu Hu, Wei-Che Hsieh, Yih Shyun E. Cheng, Pei Wei Huang, Wen Hao Lin, E. Bart Tarbet, Jim-Min Fang, Steven Weinheimer, Jia Tsrong Jan, Chun-Lin Chen, Ting Jen R Cheng, Chi-Huey Wong, Jiun-Jie Shie
المصدر: Journal of Medicinal Chemistry. 55:8657-8670
مصطلحات موضوعية: Influenzavirus A, Male, Oseltamivir, Influenzavirus B, Phosphorous Acids, Administration, Oral, Biological Availability, Neuraminidase, Pharmacology, medicine.disease_cause, Antiviral Agents, Article, Madin Darby Canine Kidney Cells, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Influenza A Virus, H1N1 Subtype, Cytopathogenic Effect, Viral, Drug Stability, Orthomyxoviridae Infections, Pharmacokinetics, Oral administration, Acetamides, Cyclohexenes, Drug Resistance, Viral, Drug Discovery, Influenza A virus, medicine, Animals, Humans, Mice, Inbred BALB C, Influenza A Virus, H5N1 Subtype, biology, Chemistry, Blood Proteins, Blood proteins, Rats, Bioavailability, Mutation, Microsomes, Liver, biology.protein, Molecular Medicine, Female, Protein Binding
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9
المؤلفون: Shi-Yun Wang, Chi-Huey Wong, Wen-I Huang, Jim-Min Fang, Ting-Jen R. Cheng, Peng-Cheng Wang, Keng-Chang Tsai, Yin-Chen Tseng, Yih-Shyun E. Cheng
المصدر: Journal of medicinal chemistry. 59(11)
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Epoxide, Acids, Carbocyclic, Neuraminidase, Cyclopentanes, Microbial Sensitivity Tests, 010402 general chemistry, 01 natural sciences, Antiviral Agents, Guanidines, chemistry.chemical_compound, Structure-Activity Relationship, Drug Discovery, Influenza, Human, medicine, Cyclopentene, Structure–activity relationship, Animals, Humans, Carboxylate, Enzyme Inhibitors, biology, Dose-Response Relationship, Drug, Molecular Structure, 010405 organic chemistry, Active site, Phosphonate, 0104 chemical sciences, chemistry, biology.protein, Molecular Medicine, Peramivir, Rabbits, medicine.drug
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10
المؤلفون: Kung-Cheng Liu, Jim-Min Fang, Jia-Tsrong Jan, Ting-Jen R. Cheng, Shi-Yun Wang, Shi-Ting Yang, Yih-Shyun E. Cheng, Chi-Huey Wong
المصدر: Journal of Medicinal Chemistry. 55:8493-8501
مصطلحات موضوعية: Lipopolysaccharides, medicine.drug_class, Neuraminidase, Pharmacology, medicine.disease_cause, Antiviral Agents, Anti-inflammatory, Virus, Cell Line, Proinflammatory cytokine, Rats, Sprague-Dawley, Interferon-gamma, Mice, Structure-Activity Relationship, Caffeic Acids, Dogs, Influenza A Virus, H1N1 Subtype, Zanamivir, Orthomyxoviridae Infections, Drug Discovery, medicine, Influenza A virus, Animals, Mice, Inbred BALB C, Influenza A Virus, H5N1 Subtype, biology, Interleukin-6, Tumor Necrosis Factor-alpha, Chemistry, Anti-Inflammatory Agents, Non-Steroidal, virus diseases, Virology, Influenza A virus subtype H5N1, Rats, biology.protein, Molecular Medicine, Female, medicine.drug, Conjugate