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1
المؤلفون: Shu Fu Lin, Li-Wei Teng, Ya-Chi Huang, Shyh-Fong Chen, Guan-Ru Huang, Chih-Lin Chang, Pi-Chen Hsu, Min-Sian Huang, Yu-Sheng Gao, Ya-Wen Chan, Jiann-Jyh Huang, Sheng-Chuan Yang, Bo-Han Jian, Yann-Yu Lu, Yu-Fen Chen, Tzu-Hao Lo, Shih-Hsien Chuang, Wen-Yun Hsueh, Po-Hsun Huang, Hsin-Yi Huang, Lien-Hsiang Chang, Win-Yin Wei, Ying-Chou Chen, Her-Sheng Lin, Shan-Yen Chou, Ta-Tung Yuan, Yu-Ting Chao, Ying-Shuan E. Lee, Yi-Feng Kao, Yu-Hsiang Lin, Jo-Chu Lin, Hung-Huang Liu, Shao-Yun Wang, Chin-Hung Lai, Shin-Yi Huang
المصدر: Journal of Medicinal Chemistry. 64:1435-1453
مصطلحات موضوعية: 0303 health sciences, biology, Nitrile, Stereochemistry, Topoisomerase, Substrate (chemistry), 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Cascade reaction, chemistry, Mechanism of action, Docking (molecular), Drug Discovery, biology.protein, medicine, Molecular Medicine, Structure–activity relationship, Dimethylformamide, medicine.symptom, 030304 developmental biology
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2
المؤلفون: Wen-Yun, Hsueh, Ying-Shuan E, Lee, Min-Sian, Huang, Chin-Hung, Lai, Yu-Sheng, Gao, Jo-Chu, Lin, Yu-Fen, Chen, Chih-Lin, Chang, Shan-Yen, Chou, Shyh-Fong, Chen, Yann-Yu, Lu, Lien-Hsiang, Chang, Shu Fu, Lin, Yu-Hsiang, Lin, Pi-Chen, Hsu, Win-Yin, Wei, Ya-Chi, Huang, Yi-Feng, Kao, Li-Wei, Teng, Hung-Huang, Liu, Ying-Chou, Chen, Ta-Tung, Yuan, Ya-Wen, Chan, Po-Hsun, Huang, Yu-Ting, Chao, Shin-Yi, Huang, Bo-Han, Jian, Hsin-Yi, Huang, Sheng-Chuan, Yang, Tzu-Hao, Lo, Guan-Ru, Huang, Shao-Yun, Wang, Her-Sheng, Lin, Shih-Hsien, Chuang, Jiann-Jyh, Huang
المصدر: Journal of medicinal chemistry. 64(3)
مصطلحات موضوعية: Male, Models, Molecular, Mice, Nude, Antineoplastic Agents, Quinolones, Xenograft Model Antitumor Assays, Catalysis, Rats, Molecular Docking Simulation, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, DNA Topoisomerases, Type I, Drug Design, Nitriles, Animals, Humans, Female, Drug Screening Assays, Antitumor, Topoisomerase I Inhibitors, Copper
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3
المؤلفون: Win Yin Wei, Chia Wei Liu, Mann-Yan Kuo, Pei-Yi Tsai, Ying-Shuan E. Lee
المصدر: Molecular Cancer Therapeutics. 18:C046-C046
مصطلحات موضوعية: Patched, Medulloblastoma, Cancer Research, biology, Cell growth, Chemistry, medicine.disease, Hedgehog signaling pathway, Oncology, GLI1, medicine, biology.protein, Cancer research, Stem cell, Smoothened, Hedgehog
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6542575ebac34504676c8b1d6d7bf126
https://doi.org/10.1158/1535-7163.targ-19-c046 -
4
المؤلفون: Sheng-Chuan Yang, Ying-Shuan E. Lee, Chia-Wei Liu, Johnson Y.N. Lau, Shih-Hsien Chuang, Jun-Yu Lai, Her-Sheng Lin, Jia-Ming Chang, Ju-Ying Yang, Pei-Shiou Jian, Chun-Liang Lai, Yu-Hsiang Lin, Chia-chi Chang, Lynn Y L Huang, King Lam, Jiann-Jyh Huang
المصدر: Journal of Medicinal Chemistry. 57:4098-4110
مصطلحات موضوعية: Male, hERG, Antineoplastic Agents, Protein Serine-Threonine Kinases, Pharmacology, Compound 32, Rats, Sprague-Dawley, Mice, In vivo, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, NIMA-Related Kinases, IC50, Mice, Inbred BALB C, biology, Chemistry, Nuclear Proteins, Xenograft Model Antitumor Assays, In vitro, Rats, Cytoskeletal Proteins, Thiazoles, Astemizole, Cell culture, Cancer cell, biology.protein, Molecular Medicine, Female, medicine.drug
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5
المؤلفون: Li-Wei Teng, Mei-Hui Lee, Yu-Chuan Wang, Yu-Hsiang Lin, Ying-Shuan E. Lee, Sheng-Chuan Yang, Chao-Cheng Chiang, Shu Fu Lin, Shih-Hsien Chuang, Chia-Wei Liu, Jiann-Jyh Huang, Hung-Jyun Huang, Chun-Liang Lai, Ru-Wen Wang, Jia-Ming Chang, Win-Yin Wei, Ju-Ying Yang
المصدر: RSC Adv.. 4:58990-58998
مصطلحات موضوعية: MAPK/ERK pathway, biology, Stereochemistry, Chemistry, Kinase, General Chemical Engineering, Autophosphorylation, Assay, General Chemistry, chemistry.chemical_compound, Biochemistry, biology.protein, STAT3, Protein kinase B, IC50, Pyrrole
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::1a338f8d3cc7061761706b64db95da6f
https://doi.org/10.1039/c4ra08720h -
6
المؤلفون: Jiann-Jyh Huang, Win-Yin Wei, Ying-Shuan E. Lee, Tsai-Yuan Chang, Chin-Kang Sha, Chih-Shang Chen, Hsiang Yu Chen, Yun-Peng Tu
المصدر: ACS Medicinal Chemistry Letters. 3:1075-1080
مصطلحات موضوعية: chemistry.chemical_classification, Double bond, Stereochemistry, Organic Chemistry, Substituent, Biology, Biochemistry, In vitro, chemistry.chemical_compound, Tubulin, chemistry, Microtubule, Drug Discovery, Cancer cell, biology.protein, Potency, Methylene
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7
المؤلفون: Tzan-Wu Tsai, Shu-Rung Lin, Shu-Wha Lin, Pei-Hsing Huang, I.-Shing Yu, Huei-Jane Chen, Ying-Shuan E. Lee
المصدر: Thrombosis and Haemostasis. 84:865-870
مصطلحات موضوعية: Serine protease, biology, Cell growth, Hepsin, Hematology, Liver regeneration, Cell biology, medicine.anatomical_structure, Biochemistry, Cell culture, Hepatocyte, biology.protein, medicine, Alkaline phosphatase, Northern blot
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::abdfb7466e16c4f27fd75eba227eac2e
https://doi.org/10.1055/s-0037-1614129 -
8
المؤلفون: Ying-Shuan E. Lee, Pan-Chyr Yang, Yen His Liu, Y.-Y. Lu, Chih-Hsin Yang, Shian-Yi Chiou, Yu-Wen Tseng, Yu Jie Lin, Li Jung Chen, Mann-Yan Kuo, Yi-Ting Huang
المصدر: Molecular Cancer Therapeutics. 12:C270-C270
مصطلحات موضوعية: Cancer Research, Chemistry, Cell growth, Cancer, Pharmacology, medicine.disease, mTORC2, Oncology, In vivo, LNCaP, medicine, Lung cancer, Tyrosine kinase, PI3K/AKT/mTOR pathway
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::1554b39e540b1717a93fa4d1f1ee39ae
https://doi.org/10.1158/1535-7163.targ-13-c270