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1
المؤلفون: Amol Magdum, Anil Panmand, Ravi K. Bhamidipati, Amol A. Raje, Vamsi Madgula, Ganesh Bhat, Meena Patel, Sreekanth R. Rouduri, Siddhartha De, Yogesh D. Shejul, Rajesh Bonagiri, Vandna Prasad, Anita Chugh, Ashwinkumar V. Meru, Vidya Ramdas, Sujay Basu, Dinesh A. Barawkar, Venkata P. Palle, Azfar Quraishi, Narayanan Hariharan, Sumit Chaudhary, Kasim A. Mookhtiar, Indraneel Ghosh, Minakshi Naykodi, K. Kashinath, Sachin Thorat
المصدر: ACS Medicinal Chemistry Letters. 8:835-840
مصطلحات موضوعية: Parkinson's disease, Organic Chemistry, Adenosine A2A receptor, Pharmacology, Catalepsy, Biology, medicine.disease, 01 natural sciences, Biochemistry, In vitro, 0104 chemical sciences, Functional antagonism, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, medicine, Antagonism, Receptor, 030217 neurology & neurosurgery, Depression (differential diagnoses)
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2
المؤلفون: Dinesh A. Barawkar, Siddhartha De, Yogesh Waman, Ashwinkumar V. Meru, Vidya Ramdas, Kasim A. Mookhtiar, Srinivasa B. Reddy, Sumit Chaudhary, Sujay Basu, Santosh Kumar Madadi, Rhishikesh Thakare, Venkata P. Palle, Anita Chugh, Gaurav Bedse, Summon Koul, Srinivas Rao Chennamaneni, Yogesh D. Shejul, Neela Prasad, Sandhya Chaturvedi, Rajesh Bonagiri, Suraj Menon, Jayasagar Gundu
المصدر: Bioorganic & Medicinal Chemistry. 25:1963-1975
مصطلحات موضوعية: 0301 basic medicine, Primary (chemistry), Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Diuresis, PK Parameters, 030204 cardiovascular system & hematology, Pharmacology, Biochemistry, 03 medical and health sciences, Adenosine A1 receptor, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, Pharmacokinetics, In vivo, Drug Discovery, Molecular Medicine, Molecular Biology, Hypoxanthine, Biological evaluation
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3
المؤلفون: Azfar Quraishi, Anita Chug, Suraj Menon, Vishal Unadkat, Sujay Basu, Madhav S. Seervi, Vandna Prasad, Sumit Chaudhary, Yogesh D. Shejul, Ganesh Bhat, Sachin Thorat, Ravi K. Bhamidipati, Shariq S. Ansari, Ashwinkumar V. Meru, Rhishikesh Thakare, Kasim A. Mookhtiar, Yogesh Salve, Venkata P. Palle, Minakshi Naykodi, Siddhartha De, Vaibhav Jain, Harish Patil, Indraneel Ghosh, Dinesh A. Barawkar, Meena Patel, Sreekanth R. Rouduri
المصدر: Journal of Medicinal Chemistry. 60:681-694
مصطلحات موضوعية: 0301 basic medicine, Chemistry, Antagonist, Pharmacology, 01 natural sciences, Adenosine receptor, In vitro, 0104 chemical sciences, Bioavailability, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Benzothiazole, Pharmacokinetics, Drug Discovery, Molecular Medicine, Solubility, ADME
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4
المؤلفون: Sujay, Basu, Dinesh A, Barawkar, Vidya, Ramdas, Minakshi, Naykodi, Yogesh D, Shejul, Meena, Patel, Sachin, Thorat, Anil, Panmand, K, Kashinath, Rajesh, Bonagiri, Vandna, Prasad, Ganesh, Bhat, Azfar, Quraishi, Sumit, Chaudhary, Amol, Magdum, Ashwinkumar V, Meru, Indraneel, Ghosh, Ravi K, Bhamidipati, Amol A, Raje, Vamsi L M, Madgula, Siddhartha, De, Sreekanth R, Rouduri, Venkata P, Palle, Anita, Chugh, Narayanan, Hariharan, Kasim A, Mookhtiar
المصدر: ACS medicinal chemistry letters. 8(8)
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5
المؤلفون: Sujay, Basu, Dinesh A, Barawkar, Sachin, Thorat, Yogesh D, Shejul, Meena, Patel, Minakshi, Naykodi, Vaibhav, Jain, Yogesh, Salve, Vandna, Prasad, Sumit, Chaudhary, Indraneel, Ghosh, Ganesh, Bhat, Azfar, Quraishi, Harish, Patil, Shariq, Ansari, Suraj, Menon, Vishal, Unadkat, Rhishikesh, Thakare, Madhav S, Seervi, Ashwinkumar V, Meru, Siddhartha, De, Ravi K, Bhamidipati, Sreekanth R, Rouduri, Venkata P, Palle, Anita, Chug, Kasim A, Mookhtiar
المصدر: Journal of medicinal chemistry. 60(2)
مصطلحات موضوعية: Male, Receptor, Adenosine A2A, Administration, Oral, Cyclohexanols, Adenosine A2 Receptor Antagonists, Antiparkinson Agents, Levodopa, Molecular Docking Simulation, Structure-Activity Relationship, HEK293 Cells, Drug Design, Microsomes, Liver, Animals, Humans, Benzothiazoles, Rats, Wistar
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6
المؤلفون: Summon, Koul, Vidya, Ramdas, Dinesh A, Barawkar, Yogesh B, Waman, Neela, Prasad, Santosh Kumar, Madadi, Yogesh D, Shejul, Rajesh, Bonagiri, Sujay, Basu, Suraj, Menon, Srinivasa B, Reddy, Sandhya, Chaturvedi, Srinivas Rao, Chennamaneni, Gaurav, Bedse, Rhishikesh, Thakare, Jayasagar, Gundu, Sumit, Chaudhary, Siddhartha, De, Ashwinkumar V, Meru, Venkata, Palle, Anita, Chugh, Kasim A, Mookhtiar
المصدر: Bioorganicmedicinal chemistry. 25(6)
مصطلحات موضوعية: Male, Proton Magnetic Resonance Spectroscopy, Adenosine A1 Receptor Antagonists, Mass Spectrometry, Rats, Radioligand Assay, HEK293 Cells, Drug Design, Hypoxanthines, Animals, Humans, Carbon-13 Magnetic Resonance Spectroscopy, Rats, Wistar, Chromatography, Liquid
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7
المؤلفون: Gagan Kukreja, Sophie Roy, Siddhartha De, Anita Chugh, Samuel D. Wright, Ravi P. Nargund, Suhas Tambe, Yogesh D. Shejul, Deepak B. Salunke, Michael P. Graziano, Jayasagar Gundu, Santosh Kurhade, Debnath Bhuniya, Kasim A. Mookhtiar, Sheo B. Singh, Joseph P. Vacca, Dhananjay N. Umrani, Bhavesh Dave, Minakshi Naykodi, Tian-Quan Cai, Sreemita Majumdar, Doris F. Cully, Prasun K. Chakravarty, Nadim S. Shaikh, Venkata P. Palle, Srinivasa B. Reddy, Prasad Shitole
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:3596-3602
مصطلحات موضوعية: Male, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Biochemistry, Receptors, G-Protein-Coupled, Small Molecule Libraries, Inhibitory Concentration 50, In vivo, Drug Discovery, Succinate receptor 1, Animals, Structure–activity relationship, Rats, Wistar, Receptor, Molecular Biology, G protein-coupled receptor, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Biological activity, Small molecule, Rats, Molecular Medicine