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1
المؤلفون: Kenji Yoshikawa, Toshiharu Yoshino, Makoto Takemura, Akiyoshi Mochizuki, Toshiharu Ohta, Tsutomu Nagata, Kouichi Uoto, Yoshihiro Yokomizo, Hiroyuki Naito, Katsuhiro Kawakami, Hideyuki Kanno, Makoto Suzuki
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2133-2140
مصطلحات موضوعية: Models, Molecular, Serine Proteinase Inhibitors, Molecular model, medicine.drug_mechanism_of_action, Stereochemistry, Carboxylic acid, Clinical Biochemistry, Factor Xa Inhibitor, Substituent, Pharmaceutical Science, Ethylenediamine, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Structure–activity relationship, Moiety, Molecular Biology, chemistry.chemical_classification, Organic Chemistry, chemistry, Drug Design, Molecular Medicine, Factor Xa Inhibitors
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2
المؤلفون: Kenji Namba, Masami Ohtsuka, Yoshihiro Yokomizo, Hironobu Nitanai, Kazuki Hoshino, Makoto Takemura, Ving J. Lee, Kiyoshi Nakayama, Jason Z. Zhang, Yoshida Kenichi, William J. Watkins, Hiroko Kanda
المصدر: Bioorganic & Medicinal Chemistry. 14:8506-8518
مصطلحات موضوعية: Ofloxacin, Pyrimidine, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Levofloxacin, Microbial Sensitivity Tests, medicine.disease_cause, Biochemistry, Rats, Sprague-Dawley, Aztreonam, chemistry.chemical_compound, Drug Discovery, medicine, Animals, Lung, Molecular Biology, Antibacterial agent, Chemistry, Pseudomonas aeruginosa, Aryl, Organic Chemistry, Membrane Transport Proteins, Biological activity, biochemical phenomena, metabolism, and nutrition, Anti-Bacterial Agents, Rats, Pyrimidines, Molecular Medicine, Efflux, Bacterial Outer Membrane Proteins, medicine.drug
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3
المؤلفون: Yoshida Kenichi, William J. Watkins, Monica Palme, Aesop Cho, Katsuya Akimoto, Kazuki Hoshino, Ving J. Lee, Atsunobu Sakamoto, Jason Z. Zhang, Haruko Kawato, Kiyoshi Nakayama, Hiroko Ishida, Masami Ohtsuka, Yoshihiro Yokomizo, Noriko Kuru, Toshiharu Ohta, Junko Itoh
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:2493-2497
مصطلحات موضوعية: Photoisomerization, Photochemistry, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Microbial Sensitivity Tests, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Drug Stability, Isomerism, Membrane Transport Modulators, Amide, Drug Resistance, Bacterial, Drug Discovery, Peptide bond, Moiety, Tetrazole, Molecular Biology, Antibacterial agent, Acrylic acid, Organic Chemistry, Membrane Transport Proteins, Pyrimidines, Acrylates, chemistry, Pseudomonas aeruginosa, Molecular Medicine, Efflux, Bacterial Outer Membrane Proteins
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4
المؤلفون: Aesop Cho, Yoshida Kenichi, Monica Palme, William J. Watkins, Atsunobu Sakamoto, Toshiharu Ohta, Noriko Kuru, Ving J. Lee, Masami Ohtsuka, Jun Watanabe, Haruko Kawato, Jason Z. Zhang, Hiroko Ishida, Kiyoshi Nakayama, Kazuki Hoshino, Yoshihiro Yokomizo, Kumi Yoshida
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:475-479
مصطلحات موضوعية: Chemistry, Pseudomonas aeruginosa, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Membrane Transport Proteins, Pharmaceutical Science, medicine.disease_cause, Biochemistry, Mexab oprm, Pyrimidines, Membrane Transport Modulators, Drug Discovery, medicine, Molecular Medicine, Potency, Moiety, Efflux, Pharmacophore, Carrier Proteins, Molecular Biology, Bacterial Outer Membrane Proteins, Protein Binding
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5
المؤلفون: Kumi Yoshida, Haruko Kawato, Yoshida Kenichi, William J. Watkins, Ving J. Lee, Yohei Ishida, Tsuyoshi Otani, Thomas E. Renau, Yoshihiro Yokomizo, Hiroko Ishida, Kazuki Hoshino, Masami Ohtsuka, Toshiharu Ohta, Yuichi Kurosaka, Kiyoshi Nakayama
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:4205-4208
مصطلحات موضوعية: Sitafloxacin, Ofloxacin, Neutropenia, Lactams, Clinical Biochemistry, Biological Transport, Active, Pharmaceutical Science, Diaphragm pump, Levofloxacin, Microbial Sensitivity Tests, Plasma protein binding, medicine.disease_cause, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Sepsis, Drug Discovery, medicine, Animals, Molecular Biology, Serum Albumin, Pseudomonas aeruginosa, Chemistry, Organic Chemistry, Membrane Transport Proteins, Drug Resistance, Microbial, Biological activity, Gene Expression Regulation, Bacterial, Anti-Bacterial Agents, Rats, Molecular Medicine, Efflux, Pharmacophore, Carrier Proteins, Bacterial Outer Membrane Proteins, Fluoroquinolones, Protein Binding, medicine.drug
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6
المؤلفون: Yoshida Kenichi, Shigeru Hosono, William J. Watkins, Haruko Kawato, Yoshihiro Yokomizo, Kiyoshi Nakayama, Kumi Yoshida, Toshiharu Ohta, Kazuki Hoshino, Roger Leger, Masami Ohtsuka, Ving J. Lee, Jason Z. Zhang, Yohei Ishida, Thomas E. Renau, Hiroko Ishida
المصدر: Bioorganic & Medicinal Chemistry Letters. 13:4201-4204
مصطلحات موضوعية: Neutropenia, Lactams, Clinical Biochemistry, Biological Transport, Active, Pharmaceutical Science, Diaphragm pump, Microbial Sensitivity Tests, medicine.disease_cause, Biochemistry, Mice, Structure-Activity Relationship, In vivo, Sepsis, Drug Discovery, medicine, Animals, Molecular Biology, Serum Albumin, Antibacterial agent, biology, Pseudomonas aeruginosa, Chemistry, Organic Chemistry, Membrane Transport Proteins, Drug Resistance, Microbial, Gene Expression Regulation, Bacterial, biology.organism_classification, In vitro, Anti-Bacterial Agents, Pseudomonadales, Molecular Medicine, Efflux, Carrier Proteins, Bacterial Outer Membrane Proteins, Protein Binding, Pseudomonadaceae
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7
المؤلفون: Yasuyuki TAKEDA, Keiichi KAWAGOE, Aki YOKOMIZO, Yoshihiro YOKOMIZO, Toru HOSOKAMI, Yoshimasa SHIMOTO, Yoshiaki TABUCHI, Yoshiyasu OGIHARA, Yuko HONDA, Keiko KAWARABAYASHI, Miki ISERI, Shuichi YOKOHAMA
المصدر: Chemical and Pharmaceutical Bulletin. 47:755-771
مصطلحات موضوعية: Male, Alkylation, Chemical Phenomena, Chemistry, Physical, Phenylurea Compounds, CHO Cells, General Chemistry, General Medicine, Acetates, Phenoxyacetates, Receptor, Cholecystokinin B, Rats, Rats, Sprague-Dawley, Structure-Activity Relationship, Gastric Mucosa, Cricetinae, Gastrins, Drug Discovery, Animals, Humans, Pentagastrin, Receptors, Cholecystokinin
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0f40ab67adeb5103712825d89a2a0cd8
https://doi.org/10.1248/cpb.47.755 -
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المصدر: ChemInform. 24
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Trimethylsilyl, chemistry.chemical_element, Stereoselectivity, General Medicine, Medicinal chemistry, Trifluoromethanesulfonate, Catalysis, Titanium
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9
المصدر: Chemistry Letters. 21:1401-1404
مصطلحات موضوعية: chemistry.chemical_classification, Reaction mechanism, Trimethylsilyl, Chemistry, Glycoside, chemistry.chemical_element, General Chemistry, Catalysis, chemistry.chemical_compound, Aldose, Organic chemistry, Stereoselectivity, Trifluoromethanesulfonate, Titanium
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b426d254d974f11cf024d905c00f824c
https://doi.org/10.1246/cl.1992.1401 -
10
المؤلفون: Kazuki Hoshino, Yoshida Kenichi, William J. Watkins, Atsunobu Sakamoto, Masami Ohtsuka, Kumi Yoshida, Yoshihiro Yokomizo, Yuichiro Imamura, Kiyoshi Nakayama, Hironobu Nitanai, Hiroko Kanda, Makoto Takemura, Ving J. Lee, Jason Z. Zhang, Noriko Kuru, Kenji Namba
المصدر: Bioorganicmedicinal chemistry. 15(22)
مصطلحات موضوعية: Male, Pyrimidine, Drug-Related Side Effects and Adverse Reactions, Stereochemistry, Clinical Biochemistry, Drug Evaluation, Preclinical, Pharmaceutical Science, Aztreonam, Microbial Sensitivity Tests, medicine.disease_cause, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Piperidines, In vivo, Drug Discovery, medicine, Animals, Ammonium, Pseudomonas Infections, Infusions, Intravenous, Molecular Biology, Antibacterial agent, biology, Molecular Structure, Pseudomonas aeruginosa, Organic Chemistry, Membrane Transport Proteins, Stereoisomerism, Haplorhini, biology.organism_classification, Anti-Bacterial Agents, Rats, Quaternary Ammonium Compounds, chemistry, Solubility, Pseudomonadales, Molecular Medicine, Female, Efflux, Bacterial Outer Membrane Proteins