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المؤلفون: Theresa L. Johnson, Steven Kazmirski, Simon Low, Cyrille Kuhn, Robert V. Stanton, Yuan-Hua Ding, Gayatri D. Deshmukh, Jessie M. English, Haile Tecle, Glen Rennie, Ping Ye, Hu Liu, Joseph Wu, Alan C. Cheng, Suzanne L. Jacques, Rocco Coli, Frederic Feru
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:4885-4891
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Amino Acid Motifs, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Pyrazole, Biochemistry, Chemical synthesis, Mitogen-Activated Protein Kinase 14, Structure-Activity Relationship, chemistry.chemical_compound, Microsomes, Drug Discovery, medicine, Humans, Structure–activity relationship, Amino Acid Sequence, Binding site, Protein Kinase Inhibitors, Molecular Biology, Binding Sites, Adenine binding, biology, Chemistry, Adenine, Phenylurea Compounds, Organic Chemistry, Enzyme inhibitor, biology.protein, Pyrazoles, Molecular Medicine, Selectivity
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المؤلفون: Darcy Kohls, Simon Low, Glen Rennie, Yuan-Hua Ding, Cyrille Kuhn, Frederic Feru, Michael Kothe, Rocco Coli
المصدر: Chemical Biology & Drug Design. 70:540-546
مصطلحات موضوعية: Pharmacology, Gene isoform, Kinase, Chemistry, Organic Chemistry, Regulator, Polo-like kinase, medicine.disease_cause, Biochemistry, PLK1, enzymes and coenzymes (carbohydrates), Drug Discovery, medicine, Molecular Medicine, Transferase, biological phenomena, cell phenomena, and immunity, Carcinogenesis, Selectivity
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المؤلفون: Simon Low, Rocco Coli, Yuan-Hua Ding, Alan C. Cheng, Alissa L. Sheils, Cyrille Kuhn, Thomas A. Wynn, Theresa L. Johnson, Jim Nonomiya, Suzanne L. Jacques, Darcy Kohls, Cristina Lewis, Michael Kothe, Kimberly A. Verdries, Christine Loh
المصدر: Biochemistry. 46:5960-5971
مصطلحات موضوعية: Protein Folding, Protein Conformation, Molecular Sequence Data, Cell Cycle Proteins, Protein Serine-Threonine Kinases, Mitogen-activated protein kinase kinase, Crystallography, X-Ray, MAP3K7, Biochemistry, MAP2K7, Catalytic Domain, Proto-Oncogene Proteins, Enzyme Stability, Humans, Amino Acid Sequence, c-Raf, Phosphorylation, Binding Sites, biology, Cyclin-dependent kinase 4, Cyclin-dependent kinase 2, Enzyme Activation, Kinetics, Protein kinase domain, biology.protein, Cyclin-dependent kinase 9
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المؤلفون: Qing Cao, Yuan-Hua Ding, Yan Zhang, Michael Kothe, Tom Ellenberger, Andre Iffland, Simon Low, Darcy Kohls, Ajith V. Kamath, Jing Luan
المصدر: Biochemistry. 44:8312-8325
مصطلحات موضوعية: Phosphodiesterase Inhibitors, Molecular Sequence Data, Plasma protein binding, Biology, Crystallography, X-Ray, Biochemistry, Substrate Specificity, chemistry.chemical_compound, 3',5'-Cyclic-GMP Phosphodiesterases, Catalytic Domain, Humans, Amino Acid Sequence, Binding site, Cyclic guanosine monophosphate, Triticum, Cyclic Nucleotide Phosphodiesterases, Type 5, Binding Sites, Cell-Free System, Drug discovery, Adenine, Active site, Phosphodiesterase, Smooth muscle contraction, Cyclic Nucleotide Phosphodiesterases, Type 2, Cyclic Nucleotide Phosphodiesterases, Type 3, Cyclic Nucleotide Phosphodiesterases, Type 4, chemistry, 3',5'-Cyclic-AMP Phosphodiesterases, Protein Biosynthesis, Mutagenesis, Site-Directed, biology.protein, Phosphodiesterase 2, Rolipram, Sequence Alignment, Protein Binding
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المؤلفون: Richard C. Mulligan, Daniel Kalman, Stephen D. Gillies, Kashi Javaherian, Calvin J. Kuo, Susan Park, Junne Kamihara, Rolf Christofferson, Guillermo García-Cardeña, Yuan-Hua Ding, Kin-Ming Lo, Kenneth R. LaMontagne, Brian D. Ackley, Judah Folkman
المصدر: The Journal of Cell Biology
مصطلحات موضوعية: rho GTP-Binding Proteins, endostatin, extracellular matrix, Recombinant Fusion Proteins, Bacterial Toxins, Blotting, Western, Morphogenesis, morphogenesis, Angiogenesis Inhibitors, CDC42, Biology, Extracellular matrix, Mice, 03 medical and health sciences, 0302 clinical medicine, Bacterial Proteins, Cell Movement, Collagen Type XVIII, Animals, Humans, cdc42 GTP-Binding Protein, Protein kinase A, Cells, Cultured, collagen XVIII, 030304 developmental biology, 0303 health sciences, Cytotoxins, Cell Biology, Peptide Fragments, Endostatins, Protein Structure, Tertiary, rac GTP-Binding Proteins, Cell biology, Rac GTP-Binding Proteins, motility, Cdc42 GTP-Binding Protein, 030220 oncology & carcinogenesis, Original Article, Collagen, Endothelium, Vascular, Mitogen-Activated Protein Kinases, Endostatin, Dimerization
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f470bc4ecc21f8bb4c6b3863a2de6c47
https://doi.org/10.1083/jcb.152.6.1233 -
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المؤلفون: Stefan Hausmann, William E. Biddison, Kathrine J. Smith, Yuan-Hua Ding, David N. Garboczi, Ursula Utz, Don C. Wiley, Kai W. Wucherpfennig
المصدر: The Journal of Immunology. 162:5389-5397
مصطلحات موضوعية: Immunology, Immunology and Allergy
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::7d77cd19f9e491febeee628f97dd3ea1
https://doi.org/10.4049/jimmunol.162.9.5389 -
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المؤلفون: Rupert Timpl, Robert Shapiro, Kashi Javaherian, Rajiv Chopra, Yuan-Hua Ding, Thomas Boehm, Don C. Wiley, B. A. Harris, Erhard Hohenester, Kin-Ming Lo, Judah Folkman, Julia Lanciotti, Yue Li
المصدر: Proceedings of the National Academy of Sciences. 95:10443-10448
مصطلحات موضوعية: Stereochemistry, Recombinant Fusion Proteins, chemistry.chemical_element, macromolecular substances, Crystal structure, Zinc, Crystallography, X-Ray, Residue (chemistry), Aspartic acid, Collagen Type XVIII, Humans, Binding site, DNA Primers, Binding Sites, Multidisciplinary, Base Sequence, Heparin, Chemistry, Biological Sciences, Peptide Fragments, Endostatins, N-terminus, Crystallography, cardiovascular system, Collagen, Endostatin, Dimerization
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c3695c4c25282415840a4d19e7672bb4
https://doi.org/10.1073/pnas.95.18.10443 -
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المؤلفون: John M. Rosenberg, Robert L. Duda, Roger W. Hendrix, Yuan-hua Ding
المصدر: Biochemistry. 34:14918-14931
مصطلحات موضوعية: Protein Denaturation, Protein Folding, Protein subunit, Molecular Sequence Data, macromolecular substances, Siphoviridae, medicine.disease_cause, Guanidines, Biochemistry, Chaperonin, Adenosine Triphosphate, Capsid, Chaperonin 10, medicine, Trypsin, Amino Acid Sequence, Escherichia coli, Guanidine, Electrophoresis, Agar Gel, Base Sequence, Chemistry, Capsomere, Chaperonin 60, GroES, Virology, GroEL, Binding constant, Molecular Weight, Mutagenesis, Insertional, enzymes and coenzymes (carbohydrates), biological sciences, Biophysics, bacteria, Electrophoresis, Polyacrylamide Gel, Peptides, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::312fe99998ab53ff8ae5f0434b8d07db
https://doi.org/10.1021/bi00045a037 -
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المؤلفون: Feng Yin, Jing Wang, Yanchao Wang, Jun Xu, Hui Zhang, Xiaoming Zhang, Jianxian Gong, Guimiao Lin, Rongfeng Lan, Fei Lu, Zhen Yang, Yuan-Hua Ding
المصدر: Laboratory investigation; a journal of technical methods and pathology. 92(10)
مصطلحات موضوعية: Glycine, Mice, Nude, Cell Cycle Proteins, Biology, Protein Serine-Threonine Kinases, PLK1, Pathology and Forensic Medicine, Inhibitory Concentration 50, Mice, Aurora Kinases, Cell Line, Tumor, Neoplasms, Proto-Oncogene Proteins, Nitriles, Animals, Humans, Sulfones, Cyclin B1, Molecular Biology, Protein Kinase Inhibitors, Aurora Kinase A, Cell Proliferation, Mice, Inbred BALB C, Kinase, Cyclin-dependent kinase 2, Cyclin-dependent kinase 3, Geminin, Cell Biology, Phenotype, Amides, Cell biology, Thiazoles, Cell culture, Cancer cell, Cancer research, biology.protein, Benzimidazoles, Female, Cell Division
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المؤلفون: Yuan-Hua Ding, Brendan Connolly, Alissa L. Sheils, Michael Kothe, Alan C. Cheng, Ajith V. Kamath, Darcy Kohls, Maura E. Charlton, Laura Weibley, Lily Yang, Qing Cao, Brian J. Stockman
المصدر: Chemical biologydrug design. 73(2)
مصطلحات موضوعية: animal structures, Magnetic Resonance Spectroscopy, Nitrogen, Protein Conformation, Allosteric regulation, Fluorine-19 NMR, Protein Serine-Threonine Kinases, Ligands, Biochemistry, 3-Phosphoinositide-Dependent Protein Kinases, Catalytic Domain, Drug Discovery, Humans, Computer Simulation, PI3K/AKT/mTOR pathway, Pharmacology, Kinase, Chemistry, Organic Chemistry, Nuclear magnetic resonance spectroscopy, Protein Structure, Tertiary, Docking (molecular), Molecular Medicine, Phosphorylation, Signalling cascades, Allosteric Site, Hydrogen