نتائج البحث - "hA3AR"

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دورية أكاديمية

Design, Synthesis and Evaluation of New Indolylpyrimidylpiperazines for Gastrointestinal Cancer Therapy

المؤلفون: Aaron Tan, Maria V. Babak, Gopalakrishnan Venkatesan, Clarissa Lim, Karl-Norbert Klotz, Deron Raymond Herr, Siew Lee Cheong, Stephanie Federico, Giampiero Spalluto, Wei-Yi Ong, Yu Zong Chen, Jason Siau Ee Loo, Giorgia Pastorin

المصدر: Molecules, Vol 24, Iss 20, p 3661 (2019)

مصطلحات موضوعية: gastrointestinal cancer, ha3ar, partial agonists, indolylpyrimidylpiperazines, Organic chemistry, QD241-441

وصف الملف: electronic resource

Relation: https://www.mdpi.com/1420-3049/24/20/3661; https://doaj.org/toc/1420-3049

URL الوصول: https://doaj.org/article/21a6812bfdcc407e937785beaa8ff631

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Design, synthesis and evaluation of new indolylpyrimidylpiperazines for gastrointestinal cancer therapy

المؤلفون: Maria V. Babak, Giampiero Spalluto, Wei-Yi Ong, Aaron Tan, Siew Lee Cheong, Giorgia Pastorin, Clarissa Lim, Yu Zong Chen, Karl-Norbert Klotz, Deron R. Herr, Jason S. E. Loo, Stephanie Federico, Gopalakrishnan Venkatesan

المساهمون: Tan, A., Babak, M. V., Venkatesan, G., Lim, C., Klotz, K. -N., Herr, D. R., Cheong, S. L., Federico, S., Spalluto, G., Ong, W. -Y., Chen, Y. Z., Loo, J. S. E., Pastori, G.

المصدر: Molecules
Molecules, Vol 24, Iss 20, p 3661 (2019)

مصطلحات موضوعية: Models, Molecular, Indoles, Tertiary amine, HA, Pharmaceutical Science, Pharmacology, Analytical Chemistry, 0302 clinical medicine, Cricetinae, Drug Discovery, Receptor, Cytotoxicity, Gastrointestinal Neoplasms, Indolylpyrimidylpiperazine, 0303 health sciences, Chemistry, Communication, Ligand (biochemistry), Adenosine A2 Receptor Antagonists, Chemistry (miscellaneous), 030220 oncology & carcinogenesis, Molecular Medicine, ha3ar, Receptor, Adenosine A2A, hA3AR, Indolylpyrimidylpiperazines, CHO Cells, Pyrimidinones, Partial agonists, Partial agonist, lcsh:QD241-441, 03 medical and health sciences, Structure-Activity Relationship, Gastrointestinal cancer, Cricetulus, lcsh:Organic chemistry, Structure–activity relationship, Animals, Humans, ddc:610, Physical and Theoretical Chemistry, Piperazine, Binding selectivity, 030304 developmental biology, Cell Proliferation, Organic Chemistry, Receptor, Adenosine A3, Adenosine receptor, 3, AR

وصف الملف: application/pdf; ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::43f14bceec5f55b21302d334a3c747c2
http://hdl.handle.net/11368/2954606

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دورية أكاديمية

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N8-Isopentyl and N8-Phenylethyl Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidine Derivatives as Adenosine Receptor Antagonists

المؤلفون: FEDERICO, STEPHANIE, REDENTI, SARA, SPALLUTO, GIAMPIERO, Klotz, Karl Norbert, Moro, Stefano

المساهمون: Società chimica italiana. Divisione di chimica farmaceutica, Federico, Stephanie, Redenti, Sara, Klotz, Karl Norbert, Moro, Stefano, Spalluto, Giampiero

مصطلحات موضوعية: antagonists, 5-c]pyrimidine, GPCR, hA3AR, pyrazolo[4, 3-e]1, 4-triazolo[1, adenosine receptors, hA3AR, antagonists, GPCR, pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine, adenosine receptors

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::fb2d6cbdc49c9c1e26298490579355b7
http://hdl.handle.net/11368/2835197

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[1,2,4]Triazolo[1,5-a][1,3,5]Triazine Derivatives as Antagonists for the Adenosine Receptors: a Preliminary Study on Affinity at the A3 Subtype

المؤلفون: FEDERICO, STEPHANIE, MORO, STEFANO, SPALLUTO, GIAMPIERO, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl Norbert

المساهمون: Divisione di Chimica Farmaceutica della Società Chimica Italiana, Federico, Stephanie, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl Norbert, Moro, Stefano, Spalluto, Giampiero

مصطلحات موضوعية: antagonists, GPCR, 5]triazines, hA3AR, 4]triazolo[1, [1, [1,2,4]triazolo[1,5-a][1,3,5]triazines, adenosine receptors, GPCR, hA3AR, antagonists, 5-a][1, adenosine receptors

وصف الملف: CD-ROM

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::6d2e21d6030e1e6bfc4167a7daf98337
http://hdl.handle.net/11368/2834216

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1,2,4]Triazolo[1,5-c]pyrimidines as New Potent Human A3 Adenosine Receptor Antagonists

المؤلفون: SPALLUTO, GIAMPIERO, FEDERICO, STEPHANIE, MORO, STEFANO, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl Norbert

المساهمون: Comitato organizzatore NPCF7, Spalluto, Giampiero, Federico, Stephanie, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl Norbert, Moro, Stefano

مصطلحات موضوعية: 5-c]pyrimidine, GPCR, 4]Triazolo[1, adenosine receptors, [1,2,4]Triazolo[1,5-c]pyrimidine, hA3AR, GPCR, hA3AR, [1, adenosine receptors

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::964a4b9e0acaa2502491eee71147edaa
http://hdl.handle.net/11368/2834211

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Novel fluorescent hA3 adenosine receptor antagonists

المؤلفون: Federico, Stephanie, Kozma, Eszter, Kumar, T. Santhosh, Jacobson, Kenneth A., Moro, Stefano, Spalluto, Giampiero

المساهمون: Comitato organizzatore del NPCF 7, Federico, Stephanie, Kozma, Eszter, Kumar, T. Santhosh, Jacobson, Kenneth A., Moro, Stefano, Spalluto, Giampiero

مصطلحات موضوعية: antagonists, GPCR, fluorescent probes, hA3AR, adenosine receptors, fluorescent probes, GPCR, adenosine receptors, antagonists, hA3AR

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::dc929c1d44b112f31398a54561186c89
https://hdl.handle.net/11368/2834209

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[1,2,4]Triazolo[1,5-c]pyrimidine Nucleus as Adenosine Receptor Antagonists: Shift in Selectivity from A2A to A3 Adenosine Receptors

المؤلفون: FEDERICO, STEPHANIE, MORO, STEFANO, SPALLUTO, GIAMPIERO, Ciancetta, Antonella, Paoletta, Silvia, Cacciari, Barbara, Klotz, Karl Norbert

المساهمون: Purine club, Federico, Stephanie, Ciancetta, Antonella, Paoletta, Silvia, Cacciari, Barbara, Klotz, Karl Norbert, Moro, Stefano, Spalluto, Giampiero

مصطلحات موضوعية: 5-c]pyrimidine, GPCR, 4]Triazolo[1, hA3AR, hA2AAR, [1,2,4]Triazolo[1,5-c]pyrimidine, adenosine receptors, GPCR, hA2AAR, hA3AR, [1, adenosine receptors

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::3017cea16cd2fa6d42f7b4f0dded87f1
http://hdl.handle.net/11368/2834207

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Exploring Directionality of 5-Substitutions in a New Series of 5-Alkyamino-pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidine as a Strategy to Design Novel Human A3 Adenosine Receptors Antagonists

المؤلفون: FEDERICO, STEPHANIE, MORO, STEFANO, SPALLUTO, GIAMPIERO, Ciancetta, Antonella, Paoletta, Silvia, Pastorin, Giorgia, Cacciari, Barbara, Klotz, Karl Norbert

المساهمون: Purine club, Federico, Stephanie, Ciancetta, Antonella, Paoletta, Silvia, Pastorin, Giorgia, Cacciari, Barbara, Klotz, Karl Norbert, Moro, Stefano, Spalluto, Giampiero

مصطلحات موضوعية: GPCR, adenosine receptor antagonists, pyrazolo[4, 3-e]1, 4-triazolo[1, hA3AR, pyrazolo[4,3-e]1,2,4-triazolo[1,5-c]pyrimidines, GPCR, adenosine receptors, hA3AR, adenosine receptor antagonists, 5-c]pyrimidines, adenosine receptors

وصف الملف: ELETTRONICO

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::4678b07dcb07e9e685d07f30e1ef670b
http://hdl.handle.net/11368/2834206

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[1,2,4]triazolo[1,5-c]pyrimidines as A(3) adenosine receptor antagonists

المؤلفون: Federico, Stephanie, Redenti, Sara, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl-Norbert, Stefano Moro, Spalluto, Giampiero

المساهمون: SPRINGER, VAN GODEWIJCKSTRAAT 30, 3311 GZ DORDRECHT, NETHERLANDS, Federico, Stephanie, Redenti, Sara, Ciancetta, Antonella, Cacciari, Barbara, Klotz, Karl Norbert, Moro, Stefano, Spalluto, Giampiero

المصدر: ResearcherID
Web of Science

مصطلحات موضوعية: 5-c]pyrimidine, GPCR, 4]Triazolo[1, hA3AR, hA2AAR, [1,2,4]Triazolo[1,5-c]pyrimidine, adenosine receptors, GPCR, hA2AAR, hA3AR, [1, adenosine receptors

وصف الملف: STAMPA

URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::071eb170860f64696f34aa5048b42bd7
http://gateway.webofknowledge.com/gateway/Gateway.cgi?GWVersion=2&SrcAuth=ORCID&SrcApp=OrcidOrg&DestLinkType=FullRecord&DestApp=WOS_CPL&KeyUT=WOS:000348578700289&KeyUID=WOS:000348578700289

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