المؤلفون: Abbass EM; Chemistry Department, Faculty of Science, Ain Shams University, Cairo, Egypt. eslammorad@sci.asu.edu.eg., El-Rayyes A; Chemistry Department, College of Science, Northern Border University, 1321, Arar, Saudi Arabia., Khalil Ali A; Chemistry Department, Faculty of Science, Ain Shams University, Cairo, Egypt., El-Farargy AF; Chemistry Department, Faculty of Science, Zagazig University, Zagazig, Egypt., Kozakiewicz-Piekarz A; Department of Biomedical Chemistry and Polymers, Faculty of Chemistry, Nicolaus Copernicus University in Toruń, Toruń, Poland., Ramadan RM; Chemistry Department, Faculty of Science, Ain Shams University, Cairo, Egypt. rmramadan@sci.asu.edu.eg.

المصدر: Scientific reports [Sci Rep] 2024 Aug 13; Vol. 14 (1), pp. 18773. Date of Electronic Publication: 2024 Aug 13.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-2322 (Electronic) Linking ISSN: 20452322 NLM ISO Abbreviation: Sci Rep Subsets: MEDLINE

مواضيع طبية MeSH: Molecular Docking Simulation* , Thiazolidines*/chemistry , Thiazolidines*/chemical synthesis , Thiazolidines*/pharmacology, Catalysis ; Spiro Compounds/chemistry ; Spiro Compounds/chemical synthesis ; Spiro Compounds/pharmacology ; Crystallography, X-Ray/methods ; Anti-Bacterial Agents/pharmacology ; Anti-Bacterial Agents/chemistry ; Anti-Bacterial Agents/chemical synthesis ; Density Functional Theory ; Microbial Sensitivity Tests ; Ferric Compounds/chemistry ; Hydrogen Bonding

المؤلفون: Szlachcikowska D; Department of Biotechnology and Cell Biology, Medical College, University of Information Technology and Management in Rzeszow, Sucharskiego 2, 35-225 Rzeszow, Poland., Tabęcka-Łonczyńska A; Department of Biotechnology and Cell Biology, Medical College, University of Information Technology and Management in Rzeszow, Sucharskiego 2, 35-225 Rzeszow, Poland., Holota S; Department of Pharmaceutical, Organic and Bioorganic Chemistry, Danylo Halytsky Lviv National Medical University, Pekarska 69, 79010 Lviv, Ukraine.; Department of Organic Chemistry and Pharmacy, Lesya Ukrainka Volyn National University, Volya Avenue 13, 43025 Lutsk, Ukraine., Roman O; Department of Pharmaceutical, Organic and Bioorganic Chemistry, Danylo Halytsky Lviv National Medical University, Pekarska 69, 79010 Lviv, Ukraine., Shepeta Y; Department of Pharmaceutical Chemistry, National Pirogov Memorial Medical University, Pirogov 56, 21018 Vinnytsia, Ukraine., Lesyk R; Department of Biotechnology and Cell Biology, Medical College, University of Information Technology and Management in Rzeszow, Sucharskiego 2, 35-225 Rzeszow, Poland.; Department of Pharmaceutical, Organic and Bioorganic Chemistry, Danylo Halytsky Lviv National Medical University, Pekarska 69, 79010 Lviv, Ukraine., Szychowski KA; Department of Biotechnology and Cell Biology, Medical College, University of Information Technology and Management in Rzeszow, Sucharskiego 2, 35-225 Rzeszow, Poland.

المصدر: International journal of molecular sciences [Int J Mol Sci] 2024 Jul 03; Vol. 25 (13). Date of Electronic Publication: 2024 Jul 03.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

مواضيع طبية MeSH: Thiazolidines*/pharmacology , Thiazolidines*/chemistry , NF-kappa B*/metabolism , Signal Transduction*/drug effects, Humans ; A549 Cells ; Fibroblasts/metabolism ; Fibroblasts/drug effects ; Antioxidants/pharmacology ; Antioxidants/chemistry

المؤلفون: Saeed A; Department of Chemistry, Faculty of Science, Mansoura University, 35516, Mansoura, Egypt., Soliman AM; Department of Chemistry, Faculty of Science, Omar Al-Mukhtar University, 919, El-Bayda, Libya., Abdullah MMS; Department of Chemistry, College of Science, King Saud University, P.O. Box 2455, 11451, Riyadh, Saudi Arabia., Abdel-Latif E; Department of Chemistry, Faculty of Science, Mansoura University, 35516, Mansoura, Egypt., El-Demerdash A; Metabolic Biology & Biological Chemistry Department, John Innes Centre, Norwich Research Park, NR4 7UH, Norwich, UK.

المصدر: Chemistry & biodiversity [Chem Biodivers] 2024 Jul; Vol. 21 (7), pp. e202301870. Date of Electronic Publication: 2024 Jun 25.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Verlag Helvetica Chimica Acta Country of Publication: Switzerland NLM ID: 101197449 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1612-1880 (Electronic) Linking ISSN: 16121872 NLM ISO Abbreviation: Chem Biodivers Subsets: MEDLINE

مواضيع طبية MeSH: Molecular Docking Simulation* , Antineoplastic Agents*/pharmacology , Antineoplastic Agents*/chemistry , Antineoplastic Agents*/chemical synthesis , Thiadiazoles*/chemistry , Thiadiazoles*/pharmacology , Thiadiazoles*/chemical synthesis , Thiazolidines*/chemistry , Thiazolidines*/pharmacology , Thiazolidines*/chemical synthesis , Drug Screening Assays, Antitumor*, Humans ; Structure-Activity Relationship ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Molecular Structure ; Dose-Response Relationship, Drug

المؤلفون: Wan XC; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Zhu WJ; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Chen Y; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Cui ZH; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Zhang H; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Zheng FH; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Zhang YN; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China., Fang GM; School of Life Science, Institutes of Physical Science and Information Technology, Anhui University, Hefei, 230601, P. R. China.

المصدر: Organic letters [Org Lett] 2024 Jun 14; Vol. 26 (23), pp. 5021-5026. Date of Electronic Publication: 2024 Jun 06.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 100890393 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1523-7052 (Electronic) Linking ISSN: 15237052 NLM ISO Abbreviation: Org Lett Subsets: MEDLINE

مواضيع طبية MeSH: Oxidation-Reduction* , Thiazolidines*/chemistry , Thiazolidines*/chemical synthesis , Peptides*/chemistry , Peptides*/chemical synthesis, Molecular Structure ; Hydrazines/chemistry ; Proline/chemistry ; Esters/chemistry ; Sulfhydryl Compounds/chemistry

المؤلفون: Isogawa M; Institute for Clinical and Translational Science, Nara Medical University Hospital, 840 Shijo-Cho, Kashihara, Nara, 634-8522, Japan., Makino H; Division of Diabetes and Lipid Metabolism, National Cerebral and Cardiovascular Center, 6-1 Kishibe-Shimmachi, Suita, Osaka, 564-8565, Japan. makinoh@ncvc.go.jp., Son C; Department of Diabetes and Endocrinology, Kobe City Nishi-Kobe Medical Center, 5-7-1 Koji-Dai Nishi-Ku, Kobe, Hyogo, 651-2273, Japan., Nishimura K; Department of Preventive Medicine, National Cerebral and Cardiovascular Center, 6-1 Kishibe-Shimmachi, Suita, Osaka, 564-8565, Japan., Hirata T; Human Care Research Team, Tokyo Metropolitan Institute for Geriatrics and Gerontology, 35-2 Sakae-Cho, Itabashi-Ku, Tokyo, 173-0015, Japan., Kasama S; Center for Clinical Research and Advanced Medicine, Shiga University of Medical Science, Seta Tsukinowa-Cho, Otsu, Shiga, 520-2192, Japan., Miyamoto Y; Open Innovation Center (OIC), National Cerebral and Cardiovascular Center, 6-1 Kishibe-Shimmachi, Suita, Osaka, 564-8565, Japan., Noguchi M; Division of Diabetes and Lipid Metabolism, National Cerebral and Cardiovascular Center, 6-1 Kishibe-Shimmachi, Suita, Osaka, 564-8565, Japan., Kasahara M; Institute for Clinical and Translational Science, Nara Medical University Hospital, 840 Shijo-Cho, Kashihara, Nara, 634-8522, Japan., Hosoda K; Diabetes Center, Ijinkai Takeda General Hospital, 28-1 Ishidamoriminami-cho, Fushimi-ku, Kyoto, 601-1495, Japan.

المصدر: BMC endocrine disorders [BMC Endocr Disord] 2024 Aug 19; Vol. 24 (1), pp. 153. Date of Electronic Publication: 2024 Aug 19.

نوع المنشور: Journal Article; Comparative Study; Randomized Controlled Trial; Multicenter Study

بيانات الدورية: Publisher: BioMed Central Country of Publication: England NLM ID: 101088676 Publication Model: Electronic Cited Medium: Internet ISSN: 1472-6823 (Electronic) Linking ISSN: 14726823 NLM ISO Abbreviation: BMC Endocr Disord Subsets: MEDLINE

مواضيع طبية MeSH: Diabetes Mellitus, Type 2*/drug therapy , Canagliflozin*/therapeutic use , Thiazolidines*/therapeutic use , Pyrazoles*/therapeutic use , Energy Intake* , Body Weight*/drug effects , Sodium-Glucose Transporter 2 Inhibitors*/therapeutic use, Humans ; Male ; Female ; Middle Aged ; Aged ; Japan/epidemiology ; Hypoglycemic Agents/therapeutic use ; Blood Glucose/analysis ; Blood Glucose/metabolism ; Blood Glucose/drug effects ; Glycated Hemoglobin/analysis ; Glycated Hemoglobin/metabolism ; Dipeptidyl-Peptidase IV Inhibitors/therapeutic use ; East Asian People

المؤلفون: Shaik AR; Department of Pharmacology, School of Pharmaceutical Education and Research, Jamia Hamdard, Hamdard Nagar, New Delhi 110062, India., Kohli S; Department of Medicine, Hamdard Institute of Medical Sciences and Research, Jamia Hamdard, Hamdard Nagar, New Delhi 110062, India., Vohora D; Department of Pharmacology, School of Pharmaceutical Education and Research, Jamia Hamdard, Hamdard Nagar, New Delhi 110062, India. Electronic address: dvohora@jamiahamdard.ac.in.

المصدر: Diabetes research and clinical practice [Diabetes Res Clin Pract] 2024 Jul; Vol. 213, pp. 111744. Date of Electronic Publication: 2024 Jun 13.

نوع المنشور: Journal Article; Observational Study

بيانات الدورية: Publisher: Elsevier Scientific Publishers Country of Publication: Ireland NLM ID: 8508335 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-8227 (Electronic) Linking ISSN: 01688227 NLM ISO Abbreviation: Diabetes Res Clin Pract Subsets: MEDLINE

مواضيع طبية MeSH: Diabetes Mellitus, Type 2*/drug therapy , Diabetes Mellitus, Type 2*/blood , Metformin*/therapeutic use , Thiazolidines*/therapeutic use , Pyrazoles*/therapeutic use , Hypoglycemic Agents*/therapeutic use, Humans ; Male ; Female ; Middle Aged ; Follow-Up Studies ; Glycated Hemoglobin/metabolism ; Glycated Hemoglobin/analysis ; Drug Therapy, Combination ; Adult ; Interleukin-6/blood ; Bone Remodeling/drug effects ; Biomarkers/blood ; Aged ; Bone Resorption/drug therapy

المؤلفون: Zhou C; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China., Kong Y; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China., Zhang H; Key Laboratory of Integrated Management of Crop Diseases and Pests (Ministry of Education), College of Plant Protection, Nanjing Agricultural University, Nanjing 210095, China., Zhai N; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China., Li Z; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China., Qian X; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China.; School of Chemistry and Molecular Engineering, East China Normal University, Shanghai 200241, China., Liu Z; Key Laboratory of Integrated Management of Crop Diseases and Pests (Ministry of Education), College of Plant Protection, Nanjing Agricultural University, Nanjing 210095, China., Cheng J; Shanghai Key Laboratory of Chemical Biology, School of Pharmacy, East China University of Science and Technology, Shanghai 200237, China.

المصدر: Journal of agricultural and food chemistry [J Agric Food Chem] 2024 May 29; Vol. 72 (21), pp. 11968-11979. Date of Electronic Publication: 2024 May 17.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 0374755 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1520-5118 (Electronic) Linking ISSN: 00218561 NLM ISO Abbreviation: J Agric Food Chem Subsets: MEDLINE

مواضيع طبية MeSH: Insecticides*/chemistry , Insecticides*/toxicity , Neonicotinoids*/chemistry , Neonicotinoids*/toxicity , Thiazolidines*/chemistry , Thiazolidines*/toxicity, Animals ; Bees/drug effects ; Molecular Docking Simulation ; Insect Proteins/genetics ; Insect Proteins/chemistry ; Insect Proteins/metabolism ; Insect Proteins/toxicity ; Aphids/drug effects ; Aphids/genetics ; Structure-Activity Relationship ; Molecular Structure ; Receptors, Nicotinic/genetics ; Receptors, Nicotinic/metabolism ; Receptors, Nicotinic/chemistry

المؤلفون: Georgiou N; Laboratory of Organic Chemistry, Department of Chemistry, National and Kapodistrian University of Athens, Panepistimioupolis Zografou, 11571 Athens, Greece., Karta D; Laboratory of Organic Chemistry, Department of Chemistry, National and Kapodistrian University of Athens, Panepistimioupolis Zografou, 11571 Athens, Greece., Cheilari A; Department of Pharmacognosy and Natural Products Chemistry, Faculty of Pharmacy, National and Kapodistrian University of Athens, Panepistimiopolis Zografou, 15771 Athens, Greece., Merzel F; Theory Department, National Institute of Chemistry, 1000 Ljubljana, Slovenia., Tzeli D; Laboratory of Physical Chemistry, Department of Chemistry, National and Kapodistrian University of Athens, Panepistimioupolis Zografou, 11571 Athens, Greece.; Theoretical and Physical Chemistry Institute, National Hellenic Research Foundation, 48 Vassileos Constantinou Ave., 11635 Athens, Greece., Vassiliou S; Laboratory of Organic Chemistry, Department of Chemistry, National and Kapodistrian University of Athens, Panepistimioupolis Zografou, 11571 Athens, Greece., Mavromoustakos T; Laboratory of Organic Chemistry, Department of Chemistry, National and Kapodistrian University of Athens, Panepistimioupolis Zografou, 11571 Athens, Greece.

المصدر: Molecules (Basel, Switzerland) [Molecules] 2024 May 23; Vol. 29 (11). Date of Electronic Publication: 2024 May 23.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 100964009 Publication Model: Electronic Cited Medium: Internet ISSN: 1420-3049 (Electronic) Linking ISSN: 14203049 NLM ISO Abbreviation: Molecules Subsets: MEDLINE

مواضيع طبية MeSH: Molecular Docking Simulation* , Molecular Conformation* , Thiazolidines*/chemistry , Thiazolidines*/chemical synthesis, Isomerism ; Animals ; Acetylcholinesterase/chemistry ; Acetylcholinesterase/metabolism ; Zebrafish ; Magnetic Resonance Spectroscopy ; Janus Kinase 3/antagonists & inhibitors ; Janus Kinase 3/metabolism ; Janus Kinase 3/chemistry ; Molecular Structure

المؤلفون: Gamal MA; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Kasr El-Aini St, Cairo, 11562, Egypt., Fahim SH; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Kasr El-Aini St, Cairo, 11562, Egypt. Electronic address: samer.mohamed@pharma.cu.edu.eg., Giovannuzzi S; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Fouad MA; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Kasr El-Aini St, Cairo, 11562, Egypt; Pharmaceutical Chemistry Department, School of Pharmacy, Newgiza University, New Giza, km 22 Cairo-Alexandria Desert Road, Cairo, Egypt., Bonardi A; NEUROFARBA Department, Pharmaceutical and Nutraceutical Section, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Gratteri P; NEUROFARBA Department, Pharmaceutical and Nutraceutical Section, Laboratory of Molecular Modeling Cheminformatics & QSAR, University of Florence, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Supuran CT; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Via U. Schiff 6, 50019, Sesto Fiorentino, Firenze, Italy., Hassan GS; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Cairo University, Kasr El-Aini St, Cairo, 11562, Egypt; Pharmaceutical Chemistry Department, School of Pharmacy, Badr University in Cairo (BUC), Badr City, Egypt.

المصدر: European journal of medicinal chemistry [Eur J Med Chem] 2024 May 05; Vol. 271, pp. 116434. Date of Electronic Publication: 2024 Apr 20.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Editions Scientifiques Elsevier Country of Publication: France NLM ID: 0420510 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1768-3254 (Electronic) Linking ISSN: 02235234 NLM ISO Abbreviation: Eur J Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrase II*/antagonists & inhibitors , Carbonic Anhydrase II*/metabolism , Diabetes Mellitus, Type 2*/drug therapy , alpha-Glucosidases*/metabolism , Benzenesulfonamides* , Sulfonamides*/chemistry , Sulfonamides*/pharmacology , Sulfonamides*/chemical synthesis , Glycoside Hydrolase Inhibitors*/pharmacology , Glycoside Hydrolase Inhibitors*/chemistry , Glycoside Hydrolase Inhibitors*/chemical synthesis , Hypoglycemic Agents*/chemistry , Hypoglycemic Agents*/pharmacology , Hypoglycemic Agents*/chemical synthesis , Carbonic Anhydrase Inhibitors*/chemistry , Carbonic Anhydrase Inhibitors*/pharmacology , Carbonic Anhydrase Inhibitors*/chemical synthesis , Thiazolidines*/chemistry , Thiazolidines*/pharmacology , Thiazolidines*/chemical synthesis, Humans ; Structure-Activity Relationship ; Animals ; Ligands ; Molecular Structure ; Rats ; Dose-Response Relationship, Drug ; Molecular Docking Simulation ; Diabetes Mellitus, Experimental/drug therapy ; Male ; Rats, Wistar

المؤلفون: Desai NC; Division of Medicinal Chemistry, Department of Chemistry, Maharaja Krishnakumarsinhji Bhavnagar University, Mahatma Gandhi Campus, Bhavnagar, 364 002, India. dnisheeth@rediffmail.com., Jadeja DJ; Division of Medicinal Chemistry, Department of Chemistry, Maharaja Krishnakumarsinhji Bhavnagar University, Mahatma Gandhi Campus, Bhavnagar, 364 002, India., Jethawa AM; Division of Medicinal Chemistry, Department of Chemistry, Maharaja Krishnakumarsinhji Bhavnagar University, Mahatma Gandhi Campus, Bhavnagar, 364 002, India., Ahmad I; Division of Computer Aided Drug Design, Department of Pharmaceutical Chemistry, R. C. Patel Institute of Pharmaceutical Education and Research, Shirpur, Maharashtra, 425405, India., Patel H; Division of Computer Aided Drug Design, Department of Pharmaceutical Chemistry, R. C. Patel Institute of Pharmaceutical Education and Research, Shirpur, Maharashtra, 425405, India., Dave BP; School of Science, Indrashil University, Rajpur, Kadi, Gujarat, 382740, India.

المصدر: Molecular diversity [Mol Divers] 2024 Apr; Vol. 28 (2), pp. 693-709. Date of Electronic Publication: 2023 Feb 08.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: ESCOM Science Publishers Country of Publication: Netherlands NLM ID: 9516534 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1573-501X (Electronic) Linking ISSN: 13811991 NLM ISO Abbreviation: Mol Divers Subsets: MEDLINE

مواضيع طبية MeSH: DNA Gyrase*/chemistry , DNA Gyrase*/metabolism , Pyrazoles*/chemistry , Pyrazoles*/pharmacology , Pyrazoles*/chemical synthesis , Pyridines*/chemistry , Pyridines*/pharmacology , Thiazolidines*/chemistry , Thiazolidines*/pharmacology , Thiazolidines*/chemical synthesis , Topoisomerase II Inhibitors*/chemistry , Topoisomerase II Inhibitors*/pharmacology , Topoisomerase II Inhibitors*/chemical synthesis, Anti-Bacterial Agents/pharmacology ; Anti-Bacterial Agents/chemistry ; Anti-Bacterial Agents/chemical synthesis ; Antifungal Agents/pharmacology ; Antifungal Agents/chemistry ; Antifungal Agents/chemical synthesis ; Bacteria/drug effects ; Candida albicans/drug effects ; Drug Design ; Microbial Sensitivity Tests ; Molecular Docking Simulation ; Molecular Dynamics Simulation ; Structure-Activity Relationship