دورية أكاديمية
Caffeine regulates GABA transport via A 1 R blockade and cAMP signaling.
العنوان: | Caffeine regulates GABA transport via A |
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المؤلفون: | Borges-Martins VPP; Laboratório de Neurofarmacologia, Departamento de Fisiologia e Farmacologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: vladimirppbm@gmail.com., Ferreira DDP; Laboratório de Doenças Neurodegenerativas, Instituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro, Brazil. Electronic address: ferreiradanielle@id.uff.br., Souto AC; Laboratório de Neurofarmacologia, Departamento de Fisiologia e Farmacologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: arthursouto@id.uff.br., Oliveira Neto JG; Laboratório de Fisiologia Endócrina e Metabologia, Departamento de Fisiologia e Farmacologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: jgeisebel@gmail.com., Pereira-Figueiredo D; Laboratório de Neurobiologia da Retina, Departmento de Neurobiologia, Instituto de Biologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: dannifigueiredo12@gmail.com., da Costa Calaza K; Laboratório de Neurobiologia da Retina, Departmento de Neurobiologia, Instituto de Biologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: karincalaza@gmail.com., de Jesus Oliveira K; Laboratório de Fisiologia Endócrina e Metabologia, Departamento de Fisiologia e Farmacologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: karenoliveira@id.uff.br., Manhães AC; Laboratório de Neurofisiologia, Instituto de Biologia Roberto Alcantara Gomes, Universidade do Estado do Rio de Janeiro, Rio de Janeiro, Brazil. Electronic address: ac_manhaes@yahoo.com.br., de Melo Reis RA; Laboratório de Neuroquímica, Instituto de Biofísica Carlos Chagas Filho, Universidade Federal do Rio de Janeiro, Rio de Janeiro, Brazil. Electronic address: ramreis@biof.ufrj.br., Kubrusly RCC; Laboratório de Neurofarmacologia, Departamento de Fisiologia e Farmacologia, Universidade Federal Fluminense, Niterói, Brazil. Electronic address: reginakubrusly1@gmail.com.br. |
المصدر: | Neurochemistry international [Neurochem Int] 2019 Dec; Vol. 131, pp. 104550. Date of Electronic Publication: 2019 Sep 26. |
نوع المنشور: | Journal Article |
اللغة: | English |
بيانات الدورية: | Publisher: Pergamon Press Country of Publication: England NLM ID: 8006959 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1872-9754 (Electronic) Linking ISSN: 01970186 NLM ISO Abbreviation: Neurochem Int Subsets: MEDLINE |
أسماء مطبوعة: | Original Publication: Oxford [Elmsford, N. Y.] Pergamon Press. |
مواضيع طبية MeSH: | Angiotensin II Type 1 Receptor Blockers/*pharmacology , Angiotensin Receptor Antagonists/*pharmacology , Caffeine/*pharmacology , Central Nervous System Stimulants/*pharmacology , Cyclic AMP/*physiology , gamma-Aminobutyric Acid/*metabolism, Adenosine/analogs & derivatives ; Adenosine/pharmacology ; Amacrine Cells/drug effects ; Amacrine Cells/metabolism ; Animals ; Caffeine/antagonists & inhibitors ; Chick Embryo ; Cyclic AMP/metabolism ; Cyclic AMP-Dependent Protein Kinases/metabolism ; GABA Plasma Membrane Transport Proteins/metabolism ; Phenethylamines/pharmacology ; Receptor, Adenosine A1/drug effects ; Receptor, Adenosine A1/metabolism ; Receptor, Angiotensin, Type 1/drug effects ; Receptors, Adenosine A2/drug effects ; Receptors, Adenosine A2/metabolism ; Retina/drug effects ; Retina/embryology ; Retina/growth & development ; Signal Transduction/drug effects |
مستخلص: | Caffeine is the most consumed psychostimulant drug in the world, acting as a non-selective antagonist of adenosine receptors A (Copyright © 2019 Elsevier Ltd. All rights reserved.) |
فهرسة مساهمة: | Keywords: A1R; Caffeine; Chick; Development; GAT; Retina |
المشرفين على المادة: | 0 (Angiotensin II Type 1 Receptor Blockers) 0 (Angiotensin Receptor Antagonists) 0 (Central Nervous System Stimulants) 0 (GABA Plasma Membrane Transport Proteins) 0 (Phenethylamines) 0 (Receptor, Adenosine A1) 0 (Receptor, Angiotensin, Type 1) 0 (Receptors, Adenosine A2) 120225-54-9 (2-(4-(2-carboxyethyl)phenethylamino)-5'-N-ethylcarboxamidoadenosine) 36396-99-3 (N(6)-cyclohexyladenosine) 3G6A5W338E (Caffeine) 56-12-2 (gamma-Aminobutyric Acid) E0399OZS9N (Cyclic AMP) EC 2.7.11.11 (Cyclic AMP-Dependent Protein Kinases) K72T3FS567 (Adenosine) |
تواريخ الأحداث: | Date Created: 20190930 Date Completed: 20200903 Latest Revision: 20200903 |
رمز التحديث: | 20231215 |
DOI: | 10.1016/j.neuint.2019.104550 |
PMID: | 31563462 |
قاعدة البيانات: | MEDLINE |
تدمد: | 1872-9754 |
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DOI: | 10.1016/j.neuint.2019.104550 |