دورية أكاديمية
[ 18 F]Fluspidine-A PET Tracer for Imaging of σ 1 Receptors in the Central Nervous System.
العنوان: | [ 18 F]Fluspidine-A PET Tracer for Imaging of σ |
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المؤلفون: | Ludwig FA; Institute of Radiopharmaceutical Cancer Research, Department of Neuroradiopharmaceuticals, Helmholtz-Zentrum Dresden-Rossendorf, D-04318 Leipzig, Germany., Laurini E; Molecular Biology and Nanotechnology Laboratory (MolBNL@UniTS), DEA, University of Trieste, 34127 Trieste, Italy., Schmidt J; Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, D-48149 Münster, Germany., Pricl S; Molecular Biology and Nanotechnology Laboratory (MolBNL@UniTS), DEA, University of Trieste, 34127 Trieste, Italy.; Department of General Biophysics, Faculty of Biology and Environmental Protection, University of Lodz, 90-136 Lodz, Poland., Deuther-Conrad W; Institute of Radiopharmaceutical Cancer Research, Department of Neuroradiopharmaceuticals, Helmholtz-Zentrum Dresden-Rossendorf, D-04318 Leipzig, Germany., Wünsch B; Institut für Pharmazeutische und Medizinische Chemie, Universität Münster, Corrensstraße 48, D-48149 Münster, Germany.; GRK 2515, Chemical Biology of Ion Channels (Chembion), Universität Münster, Corrensstraße 48, D-48149 Münster, Germany. |
المصدر: | Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2024 Jan 28; Vol. 17 (2). Date of Electronic Publication: 2024 Jan 28. |
نوع المنشور: | Journal Article; Review |
اللغة: | English |
بيانات الدورية: | Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE |
أسماء مطبوعة: | Original Publication: Basel, Switzerland : MDPI, c2004- |
مستخلص: | σ |
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معلومات مُعتمدة: | Pilot applications), T.2.8 Centro Nazionale di Ricerca in Hihg-Performance Computing, Big Data, and Quantum Computing; WU 176 Deutsche Forschungsgemeinschaft |
فهرسة مساهمة: | Keywords: automated radiosynthesis; biodistribution; biotransformation; enantioselective synthesis; increased σ1 receptor density; irreversible binding of (R)-[18F]2; ligand–σ1 receptor interactions; logD7.4 value; major depressive disorder; molecular dynamics simulations; occupancy study with pridopidine; pharmacokinetics; plasma protein binding; radiometabolites; radiosynthesis; structure–affinity relationships; σ1 receptor ligands; σ1:σ2 selectivity |
تواريخ الأحداث: | Date Created: 20240224 Latest Revision: 20240227 |
رمز التحديث: | 20240227 |
مُعرف محوري في PubMed: | PMC10892410 |
DOI: | 10.3390/ph17020166 |
PMID: | 38399380 |
قاعدة البيانات: | MEDLINE |
تدمد: | 1424-8247 |
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DOI: | 10.3390/ph17020166 |