دورية أكاديمية
Attempting to Unmask the Inhibition of Sulfotransferase 1E1 in 17α-Ethinyl Estradiol Drug Interactions.
العنوان: | Attempting to Unmask the Inhibition of Sulfotransferase 1E1 in 17α-Ethinyl Estradiol Drug Interactions. |
---|---|
المؤلفون: | Rodrigues D; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA., Niosi M; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA., Eng H; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA., Healy C; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA., Lazzaro S; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA., Yang Q; Computational Chemistry, Internal Medicine, Medicine Design, Worldwide Research & Development, Cambridge, Massachusetts, USA., Cerny MA; Pharmacokinetics & Drug Metabolism, Medicine Design, Worldwide Research & Development, Pfizer Inc., Groton, Connecticut, USA. |
المصدر: | Journal of clinical pharmacology [J Clin Pharmacol] 2023 Aug; Vol. 63 (8), pp. 875-879. Date of Electronic Publication: 2023 Apr 27. |
نوع المنشور: | Journal Article |
اللغة: | English |
بيانات الدورية: | Publisher: Wiley Country of Publication: England NLM ID: 0366372 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1552-4604 (Electronic) Linking ISSN: 00912700 NLM ISO Abbreviation: J Clin Pharmacol Subsets: MEDLINE |
أسماء مطبوعة: | Publication: 2013- : Oxford : Wiley Original Publication: Stamford, Conn., Hall Associates. |
مواضيع طبية MeSH: | Ethinyl Estradiol*/pharmacology , Contraceptives, Oral, Combined*, Humans ; Female ; Drug Interactions ; Sulfotransferases ; Estradiol |
References: | Rodrigues AD. Drug interactions involving 17α-ethinylestradiol: considerations beyond cytochrome P450 3A induction and inhibition. Clin Pharmacol Ther. 2022;111(6):1212-1221. Helmer E, Karimian N, Van Assche K, et al. Ziritaxestat drug-drug interaction with oral contraceptives: role of SULT1E1 inhibition. Clin Pharmacol Ther. 2022;112(4):901-908. Wiesinger H, Berse M, Klein S, et al. Pharmacokinetic interaction between the CYP3A4 inhibitor ketoconazole and the hormone drospirenone in combination with ethinylestradiol or estradiol. Br J Clin Pharmacol. 2015;80(6):1399-1410. Schrag ML, Cui D, Rushmore TH, Shou M, Ma B, Rodrigues AD. Sulfotransferase 1E1 is a low km isoform mediating the 3-O-sulfation of ethinyl estradiol. Drug Metab Dispos. 2004;32(11):1299-1303. Schwartz J, Hunt T, Smith WB, et al. The effect of etoricoxib on the pharmacokinetics of oral contraceptives in healthy participants. J Clin Pharmacol. 2009;49(7):807-815. Kassahun K, McIntosh IS, Shou M, et al. Role of human liver cytochrome P4503A in the metabolism of etoricoxib, a novel cyclooxygenase-2 selective inhibitor. Drug Metab Dispos. 2001;29(6):813-820. Agrawal NG, Matthews CZ, Mazenko RS, et al. The effects of modifying in vivo cytochrome P450 3A (CYP3A) activity on etoricoxib pharmacokinetics and of etoricoxib administration on CYP3A activity. J Clin Pharmacol. 2004;44(10):1125-1131. Zhang H, Cui D, Wang B, et al. Pharmacokinetic drug interactions involving 17alpha-ethinylestradiol: a new look at an old drug. Clin Pharmacokinet. 2007;46(2):133-157. Kim WY, Benet LZ. P-glycoprotein (P-gp/MDR1)-mediated efflux of sex-steroid hormones and modulation of P-gp expression in vitro. Pharm Res. 2004;21(7):1284-1293. Peng R, Zhang H, Zhang Y, Wei DY. Effects of the ABCB1 (1199G >A) polymorphism on steroid sex hormone-induced P-glycoprotein expression, ATPase activity, and hormone efflux. Med Sci. 2015;3(4):124-137. Nwokolo N, Post E, Mageau AS, et al. Fostemsavir and ethinyl estradiol drug interaction: clinical recommendations for co-administration. HIV Med. 2022. https://doi.org/10.1111/hiv.13442. Ezuruike U, Humphries H, Dickins M, et al. Risk-benefit assessment of ethinyl estradiol using a physiologically based pharmacokinetic modeling approach. Clin Pharmacol Ther. 2018;104(6):1229-1239. Schwartz JI, Wong PH, Porras AG, et al. Effect of rofecoxib on the pharmacokinetics of chronically administered oral contraceptives in healthy female volunteers. J Clin Pharmacol. 2002;42(2):215-221. Liao M, Jeziorski KG, Tomaszewska-Kiecana M, et al. A phase 1, open-label, drug-drug interaction study of rucaparib with rosuvastatin and oral contraceptives in patients with advanced solid tumors. Cancer Chemother Pharmacol. 2021;88(5):887-897. Järvinen E, Deng F, Kiander W, et al. The role of uptake and efflux transporters in the disposition of glucuronide and sulfate conjugates. Front Pharmacol. 2022;12:802539. |
فهرسة مساهمة: | Keywords: 17α-ethinyl estradiol; drug interactions; oral contraceptives; sulfotransferase 1E1 |
المشرفين على المادة: | 423D2T571U (Ethinyl Estradiol) 0 (Contraceptives, Oral, Combined) EC 2.8.2.- (Sulfotransferases) 4TI98Z838E (Estradiol) |
تواريخ الأحداث: | Date Created: 20230315 Date Completed: 20230711 Latest Revision: 20230718 |
رمز التحديث: | 20230718 |
DOI: | 10.1002/jcph.2235 |
PMID: | 36919596 |
قاعدة البيانات: | MEDLINE |
تدمد: | 1552-4604 |
---|---|
DOI: | 10.1002/jcph.2235 |