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New Antibacterial 1,3,4-Thiadiazole Derivatives With Pyridine Moiety.

التفاصيل البيبلوغرافية
العنوان: New Antibacterial 1,3,4-Thiadiazole Derivatives With Pyridine Moiety.
المؤلفون: Şener N; Department of Chemistry, Faculty of Science, Kastamonu University, 37200, Kastamonu, Turkey., Aldwib AEO; Institute of Science, Kastamonu University, 37200, Kastamonu, Turkey.
المصدر: Chemistry & biodiversity [Chem Biodivers] 2024 Jun; Vol. 21 (6), pp. e202400522. Date of Electronic Publication: 2024 May 16.
نوع المنشور: Journal Article
اللغة: English
بيانات الدورية: Publisher: Verlag Helvetica Chimica Acta Country of Publication: Switzerland NLM ID: 101197449 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1612-1880 (Electronic) Linking ISSN: 16121872 NLM ISO Abbreviation: Chem Biodivers Subsets: MEDLINE
أسماء مطبوعة: Original Publication: Zürich, Switzerland : Hoboken, NJ : Verlag Helvetica Chimica Acta ; Distributed in the USA by Wiley, c2004-
مواضيع طبية MeSH: Anti-Bacterial Agents*/pharmacology , Anti-Bacterial Agents*/chemistry , Anti-Bacterial Agents*/chemical synthesis , Thiadiazoles*/chemistry , Thiadiazoles*/pharmacology , Thiadiazoles*/chemical synthesis , Pyridines*/chemistry , Pyridines*/pharmacology , Pyridines*/chemical synthesis , Microbial Sensitivity Tests* , Klebsiella pneumoniae*/drug effects , Escherichia coli*/drug effects, Molecular Structure ; Structure-Activity Relationship
مستخلص: 1,3,4-Thiadiazole compounds were synthesized using pyridine carboxylic acid derivatives and thiosemicarbazide derivatives. The molecular structures of the resulting compounds were characterized by spectroscopic methods such as ATR-FTIR, 1 H-NMR, and elemental analysis. Its compounds were also examined for their antibacterial properties against some strains of bacteria. Five synthesized compounds showed varying antibacterial effects on Escherichia coli, Salmonella kentucky, Bacillus substilis and Klebsiella pneumoniae. This result revealed that some of the resulting compounds could be antibacterial agents.
(© 2024 Wiley-VHCA AG, Zurich, Switzerland.)
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معلومات مُعتمدة: KÜBAP-01/2020-52 Kastamonu University
فهرسة مساهمة: Keywords: 1,3,4-thiadiazole; Pyridine; antibacterial
المشرفين على المادة: 0 (Anti-Bacterial Agents)
0 (Thiadiazoles)
0 (Pyridines)
14IAC3GH7G (1,3,4-thiadiazole)
NH9L3PP67S (pyridine)
تواريخ الأحداث: Date Created: 20240412 Date Completed: 20240618 Latest Revision: 20240621
رمز التحديث: 20240622
DOI: 10.1002/cbdv.202400522
PMID: 38606431
قاعدة البيانات: MEDLINE
الوصف
تدمد:1612-1880
DOI:10.1002/cbdv.202400522