دورية أكاديمية
New Antibacterial 1,3,4-Thiadiazole Derivatives With Pyridine Moiety.
العنوان: | New Antibacterial 1,3,4-Thiadiazole Derivatives With Pyridine Moiety. |
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المؤلفون: | Şener N; Department of Chemistry, Faculty of Science, Kastamonu University, 37200, Kastamonu, Turkey., Aldwib AEO; Institute of Science, Kastamonu University, 37200, Kastamonu, Turkey. |
المصدر: | Chemistry & biodiversity [Chem Biodivers] 2024 Jun; Vol. 21 (6), pp. e202400522. Date of Electronic Publication: 2024 May 16. |
نوع المنشور: | Journal Article |
اللغة: | English |
بيانات الدورية: | Publisher: Verlag Helvetica Chimica Acta Country of Publication: Switzerland NLM ID: 101197449 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1612-1880 (Electronic) Linking ISSN: 16121872 NLM ISO Abbreviation: Chem Biodivers Subsets: MEDLINE |
أسماء مطبوعة: | Original Publication: Zürich, Switzerland : Hoboken, NJ : Verlag Helvetica Chimica Acta ; Distributed in the USA by Wiley, c2004- |
مواضيع طبية MeSH: | Anti-Bacterial Agents*/pharmacology , Anti-Bacterial Agents*/chemistry , Anti-Bacterial Agents*/chemical synthesis , Thiadiazoles*/chemistry , Thiadiazoles*/pharmacology , Thiadiazoles*/chemical synthesis , Pyridines*/chemistry , Pyridines*/pharmacology , Pyridines*/chemical synthesis , Microbial Sensitivity Tests* , Klebsiella pneumoniae*/drug effects , Escherichia coli*/drug effects, Molecular Structure ; Structure-Activity Relationship |
مستخلص: | 1,3,4-Thiadiazole compounds were synthesized using pyridine carboxylic acid derivatives and thiosemicarbazide derivatives. The molecular structures of the resulting compounds were characterized by spectroscopic methods such as ATR-FTIR, 1 H-NMR, and elemental analysis. Its compounds were also examined for their antibacterial properties against some strains of bacteria. Five synthesized compounds showed varying antibacterial effects on Escherichia coli, Salmonella kentucky, Bacillus substilis and Klebsiella pneumoniae. This result revealed that some of the resulting compounds could be antibacterial agents. (© 2024 Wiley-VHCA AG, Zurich, Switzerland.) |
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معلومات مُعتمدة: | KÜBAP-01/2020-52 Kastamonu University |
فهرسة مساهمة: | Keywords: 1,3,4-thiadiazole; Pyridine; antibacterial |
المشرفين على المادة: | 0 (Anti-Bacterial Agents) 0 (Thiadiazoles) 0 (Pyridines) 14IAC3GH7G (1,3,4-thiadiazole) NH9L3PP67S (pyridine) |
تواريخ الأحداث: | Date Created: 20240412 Date Completed: 20240618 Latest Revision: 20240621 |
رمز التحديث: | 20240622 |
DOI: | 10.1002/cbdv.202400522 |
PMID: | 38606431 |
قاعدة البيانات: | MEDLINE |
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