دورية أكاديمية

Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model.

التفاصيل البيبلوغرافية
العنوان: Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model.
المؤلفون: Carcache, David A., Vulpetti, Anna, Kallen, Joerg, Mattes, Henri, Orain, David, Stringer, Rowan, Vangrevelinghe, Eric, Wolf, Romain M., Kaupmann, Klemens, Ottl, Johannes, Dawson, Janet, Cooke, Nigel G., Hoegenauer, Klemens, Billich, Andreas, Wagner, Juergen, Guntermann, Christine, Hintermann, Samuel
المصدر: Journal of Medicinal Chemistry; 8/9/2018, Vol. 61 Issue 15, p6724-6735, 12p
قاعدة البيانات: Supplemental Index
الوصف
تدمد:00222623
DOI:10.1021/acs.jmedchem.8b00529