التفاصيل البيبلوغرافية
العنوان: |
JDQ443, a Structurally Novel, Pyrazole-Based, Covalent Inhibitor of KRASG12C for the Treatment of Solid Tumors |
المؤلفون: |
Edwige Lorthiois, Marc Gerspacher, Kim S. Beyer, Andrea Vaupel, Catherine Leblanc, Rowan Stringer, Andreas Weiss, Rainer Wilcken, Daniel A. Guthy, Andreas Lingel, Claudio Bomio-Confaglia, Rainer Machauer, Pascal Rigollier, Johannes Ottl, Dorothee Arz, Pascal Bernet, Gaëlle Desjonqueres, Solene Dussauge, Malika Kazic-Legueux, Marie-Anne Lozac’h, Christophe Mura, Mickaël Sorge, Milen Todorov, Nicolas Warin, Florence Zink, Hans Voshol, Frederic J. Zecri, Richard C. Sedrani, Nils Ostermann, Saskia M. Brachmann, Simona Cotesta |
المصدر: |
Journal of Medicinal Chemistry. 65:16173-16203 |
بيانات النشر: |
American Chemical Society (ACS), 2022. |
سنة النشر: |
2022 |
مصطلحات موضوعية: |
Drug Discovery, Molecular Medicine |
تدمد: |
1520-4804 0022-2623 |
URL الوصول: |
https://explore.openaire.eu/search/publication?articleId=doi_________::ad7ccf3634960d3fbc0cb2fa59a10551 https://doi.org/10.1021/acs.jmedchem.2c01438 |
حقوق: |
CLOSED |
رقم الأكسشن: |
edsair.doi...........ad7ccf3634960d3fbc0cb2fa59a10551 |
قاعدة البيانات: |
OpenAIRE |