Practical Synthesis of [18F]Pitavastatin and Evaluation of Hepatobiliary Transport Activity in Rats by Positron Emission Tomography
العنوان: | Practical Synthesis of [18F]Pitavastatin and Evaluation of Hepatobiliary Transport Activity in Rats by Positron Emission Tomography |
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المؤلفون: | Takayoshi Nakaoka, Ken-ichi Kaneko, Yuichi Sugiyama, Yoshie Suezaki, Takamitsu Hosoya, Natsumi Otsuka, Hidenori Ochiai, Satsuki Irie, Hiroyuki Kusuhara, Takashi Niwa, Emi Hayashinaka, Yilong Cui, Yasuyoshi Watanabe, Yuta Uetake, Kazuya Maeda, Yasuhiro Wada |
المصدر: | Molecular Pharmaceutics. 17:1884-1898 |
بيانات النشر: | American Chemical Society (ACS), 2020. |
سنة النشر: | 2020 |
مصطلحات موضوعية: | Nuclear magnetic resonance, medicine.diagnostic_test, Chemistry, Transport activity, Positron emission tomography, Drug Discovery, medicine, Pharmaceutical Science, Molecular Medicine, Pitavastatin, medicine.drug |
الوصف: | We developed a practical synthetic method for fluorine-18 (18F)-labeled pitavastatin ([18F]PTV) as a positron emission tomography (PET) tracer to assess hepatobiliary transporter activity and condu... |
تدمد: | 1543-8392 1543-8384 |
URL الوصول: | https://explore.openaire.eu/search/publication?articleId=doi_________::c1c7535ecb3ce9aa67fbdefdc914e3be https://doi.org/10.1021/acs.molpharmaceut.9b01284 |
حقوق: | CLOSED |
رقم الأكسشن: | edsair.doi...........c1c7535ecb3ce9aa67fbdefdc914e3be |
قاعدة البيانات: | OpenAIRE |
تدمد: | 15438392 15438384 |
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