Practical Synthesis of [18F]Pitavastatin and Evaluation of Hepatobiliary Transport Activity in Rats by Positron Emission Tomography

التفاصيل البيبلوغرافية
العنوان: Practical Synthesis of [18F]Pitavastatin and Evaluation of Hepatobiliary Transport Activity in Rats by Positron Emission Tomography
المؤلفون: Takayoshi Nakaoka, Ken-ichi Kaneko, Yuichi Sugiyama, Yoshie Suezaki, Takamitsu Hosoya, Natsumi Otsuka, Hidenori Ochiai, Satsuki Irie, Hiroyuki Kusuhara, Takashi Niwa, Emi Hayashinaka, Yilong Cui, Yasuyoshi Watanabe, Yuta Uetake, Kazuya Maeda, Yasuhiro Wada
المصدر: Molecular Pharmaceutics. 17:1884-1898
بيانات النشر: American Chemical Society (ACS), 2020.
سنة النشر: 2020
مصطلحات موضوعية: Nuclear magnetic resonance, medicine.diagnostic_test, Chemistry, Transport activity, Positron emission tomography, Drug Discovery, medicine, Pharmaceutical Science, Molecular Medicine, Pitavastatin, medicine.drug
الوصف: We developed a practical synthetic method for fluorine-18 (18F)-labeled pitavastatin ([18F]PTV) as a positron emission tomography (PET) tracer to assess hepatobiliary transporter activity and condu...
تدمد: 1543-8392
1543-8384
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::c1c7535ecb3ce9aa67fbdefdc914e3be
https://doi.org/10.1021/acs.molpharmaceut.9b01284
حقوق: CLOSED
رقم الأكسشن: edsair.doi...........c1c7535ecb3ce9aa67fbdefdc914e3be
قاعدة البيانات: OpenAIRE