Supplementary Data 2 from Discovery of JNJ-63576253, a Next-Generation Androgen Receptor Antagonist Active Against Wild-Type and Clinically Relevant Ligand Binding Domain Mutations in Metastatic Castration-Resistant Prostate Cancer

التفاصيل البيبلوغرافية
العنوان: Supplementary Data 2 from Discovery of JNJ-63576253, a Next-Generation Androgen Receptor Antagonist Active Against Wild-Type and Clinically Relevant Ligand Binding Domain Mutations in Metastatic Castration-Resistant Prostate Cancer
المؤلفون: Gilles Bignan, Marco M. Gottardis, Yolanda T. Chong, Christopher J. Parrett, Kathryn Packman, Lieven Meerpoel, Geert Van Hecke, Georges Habineza, James R. Bischoff, Steffen Jaensch, Janine Ondrus, Ian Hickson, Zhuming Zhang, Peter J. Connolly, Vineet Pande, Tammy L. Bush, Jonathan R. Branch
بيانات النشر: American Association for Cancer Research (AACR), 2023.
سنة النشر: 2023
الوصف: Enzalutamide activates AR signaling in the absence of androgen in HepG2 transiently transfected with AR F877L and AR F877L/T878A constructs but not AR T878A only
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::69f427283d55abb76e964cda4ea0a4f9
https://doi.org/10.1158/1535-7163.22522980
حقوق: OPEN
رقم الأكسشن: edsair.doi.dedup.....69f427283d55abb76e964cda4ea0a4f9
قاعدة البيانات: OpenAIRE