دورية أكاديمية

Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer

التفاصيل البيبلوغرافية
العنوان: Discovery and optimization of 1-(1H-indol-1-yl)ethanone derivatives as CBP/EP300 bromodomain inhibitors for the treatment of castration-resistant prostate cancer
المؤلفون: Xiang, Qiuping, Wang, Chao, Zhang, Yan, Xue, Xiaoqian, Song, Ming, Zhang, Cheng, Li, Chenchang, Wu, Chun, Li, Kuai, Hui, Xiaoyan, Zhou, Yulai, Smaill, Jeff B., Patterson, Adam V., Wu, Donghai, Ding, Ke, Xu, Yong
المصدر: In European Journal of Medicinal Chemistry 10 March 2018 147:238-252
قاعدة البيانات: ScienceDirect
الوصف
تدمد:02235234
DOI:10.1016/j.ejmech.2018.01.087