دورية أكاديمية

The advantages of describing covalent inhibitor in vitro potencies by IC50 at a fixed time point. IC50 determination of covalent inhibitors provides meaningful data to medicinal chemistry for SAR optimization

التفاصيل البيبلوغرافية
العنوان: The advantages of describing covalent inhibitor in vitro potencies by IC50 at a fixed time point. IC50 determination of covalent inhibitors provides meaningful data to medicinal chemistry for SAR optimization
المؤلفون: Thorarensen, Atli, Balbo, Paul, Banker, Mary E., Czerwinski, Robert M., Kuhn, Max, Maurer, Tristan S., Telliez, Jean-Baptiste, Vincent, Fabien, Wittwer, Arthur J.
المصدر: In Bioorganic & Medicinal Chemistry 1 January 2021 29
قاعدة البيانات: ScienceDirect
الوصف
تدمد:09680896
DOI:10.1016/j.bmc.2020.115865